PubMed

Adenylyl cyclases as innovative therapeutic goals.

Pavan B, Biondi C, Dalpiaz A.

Drug Discov Today. 2009 Oct;14(19-20):982-91. Epub 2009 Jul 26.PMID: 19638320 [PubMed - in process]Related articles

Fabrication via a nonaqueous nanoprecipitation method, characterization and in vitro biological behavior of N(6)-cyclopentyladenosine-loaded nanoparticles.

Dalpiaz A, Vighi E, Pavan B, Leo E.

J Pharm Sci. 2009 Nov;98(11):4272-84.PMID: 19283768 [PubMed - in process]Related articles

Zolpidem-induced sleep-driving.

Doane JA, Dalpiaz AS.

Am J Med. 2008 Nov;121(11):e5. No abstract available. PMID: 18954831 [PubMed - indexed for MEDLINE]Related articles

An RPE cell line as a useful in vitro model for studying retinoic acid receptor beta: expression and affinity.

Pavan B, Dalpiaz A, Biondi C, Nieddu M, De Luca A, Prasad PD, Paganetto G, Favaloro B.

Biosci Rep. 2008 Dec;28(6):327-34.PMID: 18673301 [PubMed - indexed for MEDLINE]Related articles

Progress in drug delivery to the central nervous system by the prodrug approach.

Pavan B, Dalpiaz A, Ciliberti N, Biondi C, Manfredini S, Vertuani S.

Molecules. 2008 May 1;13(5):1035-65. Review.PMID: 18560328 [PubMed - indexed for MEDLINE]Related articles

Treatment of non-alcoholic fatty liver disease.

Tolman KG, Dalpiaz AS.

Ther Clin Risk Manag. 2007 Dec;3(6):1153-63.PMID: 18516264 [PubMed - in process]Related articlesFree article

Brain uptake of an anti-ischemic agent by nasal administration of microparticles.

Dalpiaz A, Gavini E, Colombo G, Russo P, Bortolotti F, Ferraro L, Tanganelli S, Scatturin A, Menegatti E, Giunchedi P.

J Pharm Sci. 2008 Nov;97(11):4889-903.PMID: 18300305 [PubMed - indexed for MEDLINE]Related articles

Solid lipid microparticles for the stability enhancement of the polar drug N6-cyclopentyladenosine.

Dalpiaz A, Mezzena M, Scatturin A, Scalia S.

Int J Pharm. 2008 May 1;355(1-2):81-6. Epub 2007 Nov 29.PMID: 18178347 [PubMed - indexed for MEDLINE]Related articles

Metabolic flux analysis using stoichiometric models for Aspergillus niger: comparison under glucoamylase-producing and non-producing conditions.

Melzer G, Dalpiaz A, Grote A, Kucklick M, Göcke Y, Jonas R, Dersch P, Franco-Lara E, Nörtemann B, Hempel DC.

J Biotechnol. 2007 Dec 1;132(4):405-17. Epub 2007 Aug 26.PMID: 17931730 [PubMed - indexed for MEDLINE]Related articles

Selection of reference genes for normalisation of specific gene quantification data of Aspergillus niger.

Bohle K, Jungebloud A, Göcke Y, Dalpiaz A, Cordes C, Horn H, Hempel DC.

J Biotechnol. 2007 Dec 1;132(4):353-8. Epub 2007 Aug 7.PMID: 17868942 [PubMed - indexed for MEDLINE]Related articles

Complementary use of flow and sedimentation field-flow fractionation techniques for size characterizing biodegradable poly(lactic acid) nanospheres.

Contado C, Dalpiaz A, Leo E, Zborowski M, Williams PS.

J Chromatogr A. 2007 Jul 20;1157(1-2):321-35. Epub 2007 Apr 21.PMID: 17482199 [PubMed - indexed for MEDLINE]Related articles

Spectrum of liver disease in type 2 diabetes and management of patients with diabetes and liver disease.

Tolman KG, Fonseca V, Dalpiaz A, Tan MH.

Diabetes Care. 2007 Mar;30(3):734-43. Review. No abstract available. PMID: 17327353 [PubMed - indexed for MEDLINE]Related articlesFree article

Molecular mechanism involved in the transport of a prodrug dopamine glycosyl conjugate.

Dalpiaz A, Filosa R, de Caprariis P, Conte G, Bortolotti F, Biondi C, Scatturin A, Prasad PD, Pavan B.

Int J Pharm. 2007 May 4;336(1):133-9. Epub 2006 Nov 28.PMID: 17184941 [PubMed - indexed for MEDLINE]Related articles

Nuclear retinoic acid receptor beta as a tool in chemoprevention trials.

Pavan B, Biondi C, Dalpiaz A.

Curr Med Chem. 2006;13(29):3553-63. Review.PMID: 17168722 [PubMed - indexed for MEDLINE]Related articles

Expression and characterization of vitamin C transporter in the human trophoblast cell line HTR-8/SVneo: effect of steroids, flavonoids and NSAIDs.

Biondi C, Pavan B, Dalpiaz A, Medici S, Lunghi L, Vesce F.

Mol Hum Reprod. 2007 Jan;13(1):77-83. Epub 2006 Nov 8.PMID: 17092984 [PubMed - indexed for MEDLINE]Related articlesFree article

Polymeric nanoparticles as drug controlled release systems: a new formulation strategy for drugs with small or large molecular weight.

Leo E, Scatturin A, Vighi E, Dalpiaz A.

J Nanosci Nanotechnol. 2006 Sep-Oct;6(9-10):3070-9.PMID: 17048520 [PubMed - indexed for MEDLINE]Related articles

Cationic liposomes as potential carriers for ocular administration of peptides with anti-herpetic activity.

Cortesi R, Argnani R, Esposito E, Dalpiaz A, Scatturin A, Bortolotti F, Lufino M, Guerrini R, Cavicchioni G, Incorvaia C, Menegatti E, Manservigi R.

Int J Pharm. 2006 Jul 6;317(1):90-100. Epub 2006 Apr 5.PMID: 16600535 [PubMed - indexed for MEDLINE]Related articles

Allosteric modulation, thermodynamics and binding to wild-type and mutant (T277A) adenosine A1 receptors of LUF5831, a novel nonadenosine-like agonist.

Heitman LH, Mulder-Krieger T, Spanjersberg RF, von Frijtag Drabbe Künzel JK, Dalpiaz A, IJzerman AP.

Br J Pharmacol. 2006 Mar;147(5):533-41.PMID: 16444290 [PubMed - indexed for MEDLINE]Related articlesFree article

Nanoparticle formulation may affect the stabilization of an antiischemic prodrug.

Leo E, Contado C, Bortolotti F, Pavan B, Scatturin A, Tosi G, Manfredini S, Angusti A, Dalpiaz A.

Int J Pharm. 2006 Jan 3;307(1):103-13. Epub 2005 Nov 14.PMID: 16289882 [PubMed - indexed for MEDLINE]Related articles

Evidence for the presence of N-formyl-methionyl-leucyl-phenylalanine (fMLP) receptor ligands in human amniotic fluid and fMLP receptor modulation by physiological labour.

Biondi C, Pavan B, Dalpiaz A, Valerio A, Spisani S, Vesce F.

J Reprod Immunol. 2005 Dec;68(1-2):71-83. Epub 2005 Oct 19.PMID: 16236365 [PubMed - indexed for MEDLINE]Related articles

Caffeine intake induces an alteration in human neutrophil A2A adenosine receptors.

Varani K, Portaluppi F, Gessi S, Merighi S, Vincenzi F, Cattabriga E, Dalpiaz A, Bortolotti F, Belardinelli L, Borea PA.

Cell Mol Life Sci. 2005 Oct;62(19-20):2350-8.PMID: 16143823 [PubMed - indexed for MEDLINE]Related articles

Synthesis and biological evaluation of pro-drugs of GW196771, a potent glycine antagonist acting at the NMDA receptor.

Angusti A, Durini E, Vertuani S, Dalpiaz A, Ruffo A, Di Fabio R, Donati D, Pentassuglia G, Vitulli G, Barnaby RJ, Manfredini S.

Farmaco. 2005 May;60(5):393-7.PMID: 15885689 [PubMed - indexed for MEDLINE]Related articles

Parecoxib: a shift in pain management?

Dalpiaz AS, Peterson D.

Expert Rev Neurother. 2004 Mar;4(2):165-77. Review.PMID: 15853557 [PubMed - indexed for MEDLINE]Related articles

Binding thermodynamics as a tool to investigate the mechanisms of drug-receptor interactions: thermodynamics of cytoplasmic steroid/nuclear receptors in comparison with membrane receptors.

Gilli P, Gilli G, Borea PA, Varani K, Scatturin A, Dalpiaz A.

J Med Chem. 2005 Mar 24;48(6):2026-35.PMID: 15771445 [PubMed - indexed for MEDLINE]Related articles

Ascorbic and 6-Br-ascorbic acid conjugates as a tool to increase the therapeutic effects of potentially central active drugs.

Dalpiaz A, Pavan B, Vertuani S, Vitali F, Scaglianti M, Bortolotti F, Biondi C, Scatturin A, Tanganelli S, Ferraro L, Marzola G, Prasad P, Manfredini S.

Eur J Pharm Sci. 2005 Mar;24(4):259-69. Epub 2004 Dec 19.PMID: 15734292 [PubMed - indexed for MEDLINE]Related articles

Vitamin C and 6-amino-vitamin C conjugates of diclofenac: synthesis and evaluation.

Dalpiaz A, Pavan B, Scaglianti M, Vitali F, Bortolotti F, Biondi C, Scatturin A, Manfredini S.

Int J Pharm. 2005 Mar 3;291(1-2):171-81. Epub 2004 Dec 30.PMID: 15707744 [PubMed - indexed for MEDLINE]Related articles

Narrative review: hepatobiliary disease in type 2 diabetes mellitus.

Tolman KG, Fonseca V, Tan MH, Dalpiaz A.

Ann Intern Med. 2004 Dec 21;141(12):946-56. Review.PMID: 15611492 [PubMed - indexed for MEDLINE]Related articlesFree article

Development and characterization of biodegradable nanospheres as delivery systems of anti-ischemic adenosine derivatives.

Dalpiaz A, Leo E, Vitali F, Pavan B, Scatturin A, Bortolotti F, Manfredini S, Durini E, Forni F, Brina B, Vandelli MA.

Biomaterials. 2005 Apr;26(11):1299-306.PMID: 15475060 [PubMed - indexed for MEDLINE]Related articles

Design, synthesis and in vitro evaluation on HRPE cells of ascorbic and 6-bromoascorbic acid conjugates with neuroactive molecules.

Manfredini S, Vertuani S, Pavan B, Vitali F, Scaglianti M, Bortolotti F, Biondi C, Scatturin A, Prasad P, Dalpiaz A.

Bioorg Med Chem. 2004 Oct 15;12(20):5453-63.PMID: 15388172 [PubMed - indexed for MEDLINE]Related articles

Topical lidocaine patch therapy for myofascial pain.

Dalpiaz AS, Lordon SP, Lipman AG.

J Pain Palliat Care Pharmacother. 2004;18(3):15-34.PMID: 15364629 [PubMed - indexed for MEDLINE]Related articles

Conformational aspects of human formyl-peptide receptor agonists.

Dalpiaz A, Vertuani G, Scatturin A, Vitali F, Varani K, Spisani S.

Arzneimittelforschung. 2003;53(11):793-8.PMID: 14677376 [PubMed - indexed for MEDLINE]Related articles

Transporter-mediated effects of diclofenamic acid and its ascorbyl pro-drug in the in vivo neurotropic activity of ascorbyl nipecotic acid conjugate.

Dalpiaz A, Pavan B, Scaglianti M, Vitali F, Bortolotti F, Biondi C, Scatturin A, Tanganelli S, Ferraro L, Prasad P, Manfredini S.

J Pharm Sci. 2004 Jan;93(1):78-85.PMID: 14648638 [PubMed - indexed for MEDLINE]Related articles

Myofascial pain response to topical lidocaine patch therapy: case report.

Dalpiaz AS, Dodds TA.

J Pain Palliat Care Pharmacother. 2002;16(1):99-104.PMID: 14650453 [PubMed - indexed for MEDLINE]Related articles

Preparation and characterization of starch/cyclodextrin bioadhesive microspheres as platform for nasal administration of Gabexate Mesylate (Foy) in allergic rhinitis treatment.

Fundueanu G, Constantin M, Dalpiaz A, Bortolotti F, Cortesi R, Ascenzi P, Menegatti E.

Biomaterials. 2004 Jan;25(1):159-70.PMID: 14580919 [PubMed - indexed for MEDLINE]Related articles

Peptide derivatives as agonists or antagonists of formylpeptide receptors: analysis of their effects on neutrophils.

Dalpiaz A, Scatturin A.

Mini Rev Med Chem. 2003 May;3(3):167-73. Review.PMID: 12570833 [PubMed - indexed for MEDLINE]Related articles

Studies on human neutrophil biological functions by means of formyl-peptide receptor agonists and antagonists.

Dalpiaz A, Spisani S, Biondi C, Fabbri E, Nalli M, Ferretti ME.

Curr Drug Targets Immune Endocr Metabol Disord. 2003 Mar;3(1):33-42. Review.PMID: 12570724 [PubMed - indexed for MEDLINE]Related articles

Adenosine A(1) receptor: analysis of the potential therapeutic effects obtained by its activation in the central nervous system.

Dalpiaz A, Manfredini S.

Curr Med Chem. 2002 Nov;9(21):1923-37. Review.PMID: 12369876 [PubMed - indexed for MEDLINE]Related articles

Poly(lactic acid) microspheres for the sustained release of antiischemic agents.

Dalpiaz A, Scatturin A, Pavan B, Biondi C, Vandelli MA, Forni F.

Int J Pharm. 2002 Aug 21;242(1-2):115-20.PMID: 12176233 [PubMed - indexed for MEDLINE]Related articles

Temperature dependence of the affinity enhancement of selective adenosine A1 receptor agonism: a thermodynamic analysis.

Dalpiaz A, Pavan B, Ngos FN, Franchetti P, IJzerman AP.

Eur J Pharmacol. 2002 Jul 19;448(2-3):123-31.PMID: 12144931 [PubMed - indexed for MEDLINE]Related articles

C- and N-terminal residue effect on peptide derivatives' antagonism toward the formyl-peptide receptor.

Dalpiaz A, Ferretti ME, Vertuani G, Traniello S, Scatturin A, Spisani S.

Eur J Pharmacol. 2002 Feb 2;436(3):187-96.PMID: 11858798 [PubMed - indexed for MEDLINE]Related articles

Design, synthesis and activity of ascorbic acid prodrugs of nipecotic, kynurenic and diclophenamic acids, liable to increase neurotropic activity.

Manfredini S, Pavan B, Vertuani S, Scaglianti M, Compagnone D, Biondi C, Scatturin A, Tanganelli S, Ferraro L, Prasad P, Dalpiaz A.

J Med Chem. 2002 Jan 31;45(3):559-62.PMID: 11806707 [PubMed - indexed for MEDLINE]Related articles

Poly(lactic acid) microspheres for the sustained release of a selective A1 receptor agonist.

Dalpiaz A, Scatturin A, Pavan B, Biondi C, Vandelli MA, Forni F.

J Control Release. 2001 Jun 15;73(2-3):303-13.PMID: 11516507 [PubMed - indexed for MEDLINE]Related articles

Synthesis and study of 5'-ester prodrugs of N6-cyclopentyladenosine, a selective A1 receptor agonist.

Dalpiaz A, Scatturin A, Menegatti E, Bortolotti F, Pavan B, Biondi C, Durini E, Manfredini S.

Pharm Res. 2001 Apr;18(4):531-6.PMID: 11451042 [PubMed - indexed for MEDLINE]Related articles

Determination of the adenosine A(1) agonist N(6)-cyclopentyladenosine in rat blood by solid-phase extraction and HPLC.

Scalia S, Simeoni S, Dalpiaz A, Villani S.

J Pharm Biomed Anal. 2001 Mar;24(5-6):1131-6.PMID: 11248509 [PubMed - indexed for MEDLINE]Related articles

Met-Ile-Phe-Leu derivatives: full and partial agonists of human neutrophil formylpeptide receptors.

Dalpiaz A, Scatturin A, Vertuani G, Pecoraro R, Borea PA, Varani K, Traniello S, Spisani S.

Eur J Pharmacol. 2001 Jan 12;411(3):327-33.PMID: 11164392 [PubMed - indexed for MEDLINE]Related articles

Can thermodynamic measurements of receptor binding yield information on drug affinity and efficacy?

Borea PA, Dalpiaz A, Varani K, Gilli P, Gilli G.

Biochem Pharmacol. 2000 Dec 1;60(11):1549-56. Review.PMID: 11077036 [PubMed - indexed for MEDLINE]Related articles

Binding thermodynamics and intrinsic activity of adenosine A1 receptor ligands.

Dalpiaz A, Scatturin A, Varani K, Pecoraro R, Pavan B, Borea PA.

Life Sci. 2000 Aug 11;67(12):1517-24.PMID: 10983847 [PubMed - indexed for MEDLINE]Related articles

Conformational aspects of human formylpeptide receptor antagonists.

Scatturin A, Vertuani G, Pecoraro R, Dalpiaz A, Boggian M, Ferretti ME, Spisani S.

Arzneimittelforschung. 1999 Oct;49(10):873-7.PMID: 10554666 [PubMed - indexed for MEDLINE]Related articles

Thermodynamic in vitro studies as a method to investigate the pharmacodynamic behavior of adenosine A1 receptor ligands.

Dalpiaz A, Scatturin A, Pavan B, Varani K, IJzerman AP, Andrea Borea P.

Pharm Res. 1999 Jul;16(7):1054-8.PMID: 10450930 [PubMed - indexed for MEDLINE]Related articles

Formylpeptide receptor antagonists: structure and activity.

Dalpiaz A, Pecoraro R, Vertuani G, Spisani S, Rizzuti O, Fabbri E, Scatturin A.

Boll Chim Farm. 1999 Mar;138(3):44-8. No abstract available. PMID: 10394703 [PubMed - indexed for MEDLINE]Related articles