J Med Chem. 1996 Apr 26;39(9):1760-2.
2(S)-((3,5-bis(trifluoromethyl)benzyl)-oxy)-3(S)-phenyl-4- ((3-oxo-1,2,4-triazol-5-yl)methyl)morpholine (1): a potent, orally active, morpholine-based human neurokinin-1 receptor antagonist.
Hale JJ, Mills SG, MacCoss M, Shah SK, Qi H, Mathre DJ, Cascieri MA, Sadowski S, Strader CD, MacIntyre DE, Metzger JM.
Merck Research Laboratories, Rahway, New Jersey 07065, USA.
PMID: 8627597 [PubMed - indexed for MEDLINE]