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The following terms were not found in PubMed: -1-methylquinuclidin-1-ium-3-yl
Page 1
5+1-Heterocyclization as preparative approach for carboxy-containing triazolo[1,5-c]quinazolines with anti-inflammatory activity.
Krasovska N, Berest G, Belenichev I, Severina H, Nosulenko I, Voskoboinik O, Okovytyy S, Kovalenko S. Krasovska N, et al. Eur J Med Chem. 2024 Feb 15;266:116137. doi: 10.1016/j.ejmech.2024.116137. Epub 2024 Jan 11. Eur J Med Chem. 2024. PMID: 38237343
In vivo study on the model of acute aseptic inflammation (carrageenan test) have been revealed that synthesized compounds expose anti-inflammatory activity in the range of 0.94-52.66%. 4-(2-(Ethoxycarbonyl)-5,6-dihydro-[1,2,4]triazolo[1,5-c]quinazolin-5-yl)benzoic acid …
In vivo study on the model of acute aseptic inflammation (carrageenan test) have been revealed that synthesized compounds expose anti-inflam …
Metabolite Profiling and Characterization of LW6, a Novel HIF-1α Inhibitor, as an Antitumor Drug Candidate in Mice.
Lee K, Lee JY, Lee K, Jung CR, Kim MJ, Kim JA, Yoo DG, Shin EJ, Oh SJ. Lee K, et al. Molecules. 2021 Mar 30;26(7):1951. doi: 10.3390/molecules26071951. Molecules. 2021. PMID: 33808438 Free PMC article.
A novel HIF (hypoxia-inducible factor)-1alpha inhibitor, the (aryloxyacetylamino)benzoic acid derivative LW6, is an anticancer agent that inhibits the accumulation of HIF-1alpha. ...From this study, 2-(4-((3r,5r,7r)-adamantan-1-yl)phenoxy)acetic acid ( …
A novel HIF (hypoxia-inducible factor)-1alpha inhibitor, the (aryloxyacetylamino)benzoic acid derivative LW6, is an anticancer …
Structure-based optimization of novel azepane derivatives as PKB inhibitors.
Breitenlechner CB, Wegge T, Berillon L, Graul K, Marzenell K, Friebe WG, Thomas U, Schumacher R, Huber R, Engh RA, Masjost B. Breitenlechner CB, et al. J Med Chem. 2004 Mar 11;47(6):1375-90. doi: 10.1021/jm0310479. J Med Chem. 2004. PMID: 14998327
The original (-)-balanol-derived lead structure (4R)-4-(2-fluoro-6-hydroxy-3-methoxy-benzoyl)-benzoic acid (3R)-3-[(pyridine-4-carbonyl)amino]-azepan-4-yl ester (1) (IC(50) (PKB-alpha) = 5 nM) which contains an ester moiety was found to be plasm …
The original (-)-balanol-derived lead structure (4R)-4-(2-fluoro-6-hydroxy-3-methoxy-benzoyl)-benzoic acid (3R)-3-[(pyr …
Differentiation of natural and synthetic phenylalanine and tyrosine through natural abundance 2H nuclear magnetic resonance.
Brenna E, Fronza G, Fuganti C, Pinciroli M. Brenna E, et al. J Agric Food Chem. 2003 Aug 13;51(17):4866-72. doi: 10.1021/jf0302759. J Agric Food Chem. 2003. PMID: 12903937
The study, which includes also the NMR examination of benzoic acid (5) from 2 and of tyrosol (7) from 1, substantially fails in providing the required information because the mode of deuterium labeling of tyrosine samples of different origins is quite similar but in …
The study, which includes also the NMR examination of benzoic acid (5) from 2 and of tyrosol (7) from 1, substantially fails i …
Synthesis, structural characterization, and some properties of 2-acylmethyl-6-ester group-difunctionalized pyridine-containing iron complexes related to the active site of [Fe]-hydrogenase.
Song LC, Hu FQ, Wang MM, Xie ZJ, Xu KK, Song HB. Song LC, et al. Dalton Trans. 2014 Jun 7;43(21):8062-71. doi: 10.1039/c4dt00335g. Epub 2014 Apr 10. Dalton Trans. 2014. PMID: 24718303
As biomimetic models for [Fe]-hydrogenase, the 2-acylmethyl-6-ester group-difunctionalized pyridine-containing iron(II) complexes 1-4 have been successfully prepared via the following three separate steps. In the first step, the acylation or esterification of difunctionali …
As biomimetic models for [Fe]-hydrogenase, the 2-acylmethyl-6-ester group-difunctionalized pyridine-containing iron(II) complexes 1-4 …