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Year Number of Results
2002 1
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2005 2
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Your search was processed without automatic term mapping because it retrieved zero results.
The following terms were not found in PubMed: 7-tetrahydrobenzothiophen-2-yl, benzimidazol-1-ylthio
Unknown fields were ignored: [1,2,4], [4,3-a]
Page 1
The role of the adenosinergic system in lung fibrosis.
Della Latta V, Cabiati M, Rocchiccioli S, Del Ry S, Morales MA. Della Latta V, et al. Pharmacol Res. 2013 Oct;76:182-9. doi: 10.1016/j.phrs.2013.08.004. Epub 2013 Aug 28. Pharmacol Res. 2013. PMID: 23994158 Review.
Design, Synthesis and Anticancer Activity of New Polycyclic: Imidazole, Thiazine, Oxathiine, Pyrrolo-Quinoxaline and Thienotriazolopyrimidine Derivatives.
Abu-Hashem AA, Al-Hussain SA, Zaki MEA. Abu-Hashem AA, et al. Molecules. 2021 Apr 2;26(7):2031. doi: 10.3390/molecules26072031. Molecules. 2021. PMID: 33918322 Free PMC article.
In this article, we showed the synthesis of new polycyclic aromatic compounds, such as thienotriazolopyrimidinones, N-(thienotriazolopyrimidine) acetamide, 2-mercapto-thienotriazolo-pyrimidinones, 2-(((thieno-triazolopyrimidine) methyl) thio) thieno-tr …
In this article, we showed the synthesis of new polycyclic aromatic compounds, such as thienotriazolopyrimidinones, N-(thienotriazolo …
2-Chloro-N(6)-cyclopentyladenosine, adenosine A(1) receptor agonist, antagonizes the adenosine A(3) receptor.
Gao ZG, Jacobson KA. Gao ZG, et al. Eur J Pharmacol. 2002 May 17;443(1-3):39-42. doi: 10.1016/s0014-2999(02)01552-2. Eur J Pharmacol. 2002. PMID: 12044789 Free PMC article.
CCPA competitively antagonized the effects of agonist Cl-IB-MECA (2-chloro-N(6)-(3-iodobenzyl)-5'-N-methylcarbamoyladenosine) with K(B) value of 5.0 nM. CPA competition curves versus the A(3) antagonist radioligand [3H]PSB-11 (8-ethyl- …
CCPA competitively antagonized the effects of agonist Cl-IB-MECA (2-chloro-N(6)-(3-iodobenzyl)-5'-N-methy …
In vitro and in vivo trypanocidal evaluation of nickel complexes with an azapurine derivative against Trypanosoma cruzi.
Maldonado CR, Marín C, Olmo F, Huertas O, Quirós M, Sánchez-Moreno M, Rosales MJ, Salas JM. Maldonado CR, et al. J Med Chem. 2010 Oct 14;53(19):6964-72. doi: 10.1021/jm100581z. J Med Chem. 2010. PMID: 20812723
Seven ternary nickel(II) complexes (three previously described and four firstly described here) with an azapurine derivative (the anionic form of 4,6-dimethyl-1,2,3-triazolo[4,5-d]pyrimidin-5,7-dione) have been synthesized and spec …
Seven ternary nickel(II) complexes (three previously described and four firstly described here) with an azapurine derivative (the anionic fo …
Afferent arteriolar vasodilator effect of adenosine predominantly involves adenosine A2B receptor activation.
Feng MG, Navar LG. Feng MG, et al. Am J Physiol Renal Physiol. 2010 Aug;299(2):F310-5. doi: 10.1152/ajprenal.00149.2010. Epub 2010 May 12. Am J Physiol Renal Physiol. 2010. PMID: 20462966 Free PMC article.
Adenosine (10 micromol/l) caused modest constriction and subsequent superfusion with SCH-58261 (SCH), an A(2A) receptor blocker, at concentrations up 10 micromol/l elicited only slight additional decreases in afferent arteriolar diameter with maximum effect at a concentration of …
Adenosine (10 micromol/l) caused modest constriction and subsequent superfusion with SCH-58261 (SCH), an A(2A) receptor blocker, at concentr …
Determination of adenosine effects and adenosine receptors in murine corpus cavernosum.
Tostes RC, Giachini FR, Carneiro FS, Leite R, Inscho EW, Webb RC. Tostes RC, et al. J Pharmacol Exp Ther. 2007 Aug;322(2):678-85. doi: 10.1124/jpet.107.122705. Epub 2007 May 9. J Pharmacol Exp Ther. 2007. PMID: 17494861
Relaxation to 2-chloroadenosine was inhibited, in a concentration-dependent manner, by 2-(2-furanyl)-7-(2-phenylethyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine (SCH58261; A2(A) antagonist; 10(- …
Relaxation to 2-chloroadenosine was inhibited, in a concentration-dependent manner, by 2-(2-furanyl)-7-(2-phenyl …
Adenosine receptors involved in modulation of noradrenaline release in isolated rat tail artery.
Diniz C, Fresco P, Leal S, Gonçalves J. Diniz C, et al. Eur J Pharmacol. 2004 Nov 3;504(1-2):17-25. doi: 10.1016/j.ejphar.2004.09.048. Eur J Pharmacol. 2004. PMID: 15507216
Adenosine receptors involved in the modulation of noradrenaline release from postganglionic sympathetic nerves in rat tail artery were characterized by studying the effects of adenosine-receptor agonists and antagonists on electrically evoked tritium overflow (100 pulses, 5 …
Adenosine receptors involved in the modulation of noradrenaline release from postganglionic sympathetic nerves in rat tail artery were chara …
Characterization of adenosine receptors in the human bladder carcinoma T24 cell line.
Phelps PT, Anthes JC, Correll CC. Phelps PT, et al. Eur J Pharmacol. 2006 Apr 24;536(1-2):28-37. doi: 10.1016/j.ejphar.2006.02.046. Epub 2006 Mar 3. Eur J Pharmacol. 2006. PMID: 16581066
This rank order of potency is typical of adenosine A2B receptors. In addition, select adenosine receptor antagonists N-(4-acetylphenyl)-2-[4-(2,3,6,7-tetrahydro-2,6 dioxo-1,3-dipropyl-1H-purin-8-yl)phenoxy]acetamid …
This rank order of potency is typical of adenosine A2B receptors. In addition, select adenosine receptor antagonists N-(4-acet …
Adenosine A(2) receptor activation ameliorates mitochondrial oxidative stress upon reperfusion through the posttranslational modification of NDUFV2 subunit of complex I in the heart.
Xu J, Bian X, Liu Y, Hong L, Teng T, Sun Y, Xu Z. Xu J, et al. Free Radic Biol Med. 2017 May;106:208-218. doi: 10.1016/j.freeradbiomed.2017.02.036. Epub 2017 Feb 20. Free Radic Biol Med. 2017. PMID: 28219781
This study probed the mitochondrial events associated with the cardioprotective effect of 5'-(N-ethylcarboxamido) adenosine (NECA), an adenosine A(2) receptor agonist. ...Both the adenosine A(2A) receptor antagonist SCH58261 and A(2B) receptor antagonist MRS1 …
This study probed the mitochondrial events associated with the cardioprotective effect of 5'-(N-ethylcarboxamido) adenosine (N …
ZM241385, DPCPX, MRS1706 are inverse agonists with different relative intrinsic efficacies on constitutively active mutants of the human adenosine A2B receptor.
Li Q, Ye K, Blad CC, den Dulk H, Brouwer J, Ijzerman AP, Beukers MW. Li Q, et al. J Pharmacol Exp Ther. 2007 Feb;320(2):637-45. doi: 10.1124/jpet.106.111203. Epub 2006 Oct 31. J Pharmacol Exp Ther. 2007. PMID: 17077318
In the current study, three known A(2B) receptor antagonists, 4-{2-[7-amino-2-(2-furyl)[1,2,4]triazolo-[2,3-a][1,3,5]triazin-5-yl-amino]ethyl}phenol (ZM241385), 8-cyclopentyl-1,3-dipropylxanthine (DPCPX), and …
In the current study, three known A(2B) receptor antagonists, 4-{2-[7-amino-2-(2-furyl)[1,2,4]t …
20 results