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Items: 1 to 20 of 93

1.

Lithium Halomethylcarbenoids: Preparation and Use in the Homologation of Carbon Electrophiles.

Pace V, Holzer W, De Kimpe N.

Chem Rec. 2016 Jul 6. doi: 10.1002/tcr.201600011. [Epub ahead of print]

PMID:
27381551
2.

Highly efficient synthesis of functionalized α-oxyketones via Weinreb amides homologation with α-oxygenated organolithiums.

Pace V, Murgia I, Westermayer S, Langer T, Holzer W.

Chem Commun (Camb). 2016 Jun 18;52(48):7584-7. doi: 10.1039/c6cc03532a. Epub 2016 May 25.

PMID:
27220327
3.

Compounds from Caesalpinia sappan with anti-inflammatory properties in macrophages and chondrocytes.

Mueller M, Weinmann D, Toegel S, Holzer W, Unger FM, Viernstein H.

Food Funct. 2016 Mar;7(3):1671-9. doi: 10.1039/c5fo01256b.

PMID:
26951869
4.

Bromomethyllithium-mediated chemoselective homologation of disulfides to dithioacetals.

Pace V, Pelosi A, Antermite D, Rosati O, Curini M, Holzer W.

Chem Commun (Camb). 2016 Feb 11;52(12):2639-42. doi: 10.1039/c5cc10280d. Epub 2016 Jan 11.

PMID:
26750866
5.

A Robust, Eco-Friendly Access to Secondary Thioamides through the Addition of Organolithium Reagents to Isothiocyanates in Cyclopentyl Methyl Ether (CPME).

Pace V, Castoldi L, Monticelli S, Safranek S, Roller A, Langer T, Holzer W.

Chemistry. 2015 Dec 21;21(52):18966-70. doi: 10.1002/chem.201504247. Epub 2015 Nov 20.

PMID:
26507565
6.

Synthesis and in silico evaluation of novel compounds for PET-based investigations of the norepinephrine transporter.

Neudorfer C, Seddik A, Shanab K, Jurik A, Rami-Mark C, Holzer W, Ecker G, Mitterhauser M, Wadsak W, Spreitzer H.

Molecules. 2015 Jan 20;20(1):1712-30. doi: 10.3390/molecules20011712.

7.

Chemoselective efficient synthesis of functionalized β-oxonitriles through cyanomethylation of Weinreb amides.

Mamuye AD, Castoldi L, Azzena U, Holzer W, Pace V.

Org Biomol Chem. 2015 Feb 21;13(7):1969-73. doi: 10.1039/c4ob02398f.

PMID:
25535702
8.

Chemoenzymatic synthesis of carbohydrates as antidiabetic and anticancer drugs.

Alcántara AR, Pace V, Hoyos P, Sandoval M, Holzer W, Hernáiz MJ.

Curr Top Med Chem. 2014;14(23):2694-711. Review.

PMID:
25515749
9.

Synthesis of trifluoromethyl-substituted pyrazolo[4,3-c]pyridines - sequential versus multicomponent reaction approach.

Palka B, Di Capua A, Anzini M, Vilkauskaité G, Sačkus A, Holzer W.

Beilstein J Org Chem. 2014 Jul 31;10:1759-64. doi: 10.3762/bjoc.10.183. eCollection 2014.

10.

Development of potential selective and reversible pyrazoline based MAO-B inhibitors as MAO-B PET tracer precursors and reference substances for the early detection of Alzheimer's disease.

Neudorfer C, Shanab K, Jurik A, Schreiber V, Neudorfer C, Vraka C, Schirmer E, Holzer W, Ecker G, Mitterhauser M, Wadsak W, Spreitzer H.

Bioorg Med Chem Lett. 2014 Sep 15;24(18):4490-5. doi: 10.1016/j.bmcl.2014.07.085. Epub 2014 Aug 7.

PMID:
25127869
11.

Use of activated enol ethers in the synthesis of pyrazoles: reactions with hydrazine and a study of pyrazole tautomerism.

Tarabová D, Soralová S, Breza M, Fronc M, Holzer W, Milata V.

Beilstein J Org Chem. 2014 Apr 1;10:752-60. doi: 10.3762/bjoc.10.70. eCollection 2014.

12.

A one-step microwave-assisted synthetic method for an O/S-chemoselective route to derivatives of the first adenosine A3 PET radiotracer.

Shanab K, Neudorfer C, Holzer W, Mitterhauser M, Wadsak W, Spreitzer H.

Molecules. 2014 Apr 2;19(4):4076-82. doi: 10.3390/molecules19044076.

13.

Azido derivatives of cellobiose: oxidation at C1 with cellobiose dehydrogenase from Sclerotium rolfsii.

Mulla D, Kracher D, Ludwig R, Nagy G, Grandits M, Holzer W, Saber Y, Gabra N, Viernstein H, Unger FM.

Carbohydr Res. 2013 Dec 15;382:86-94. doi: 10.1016/j.carres.2013.09.004. Epub 2013 Sep 16.

PMID:
24211370
14.

Synthesis and antiproliferative activity of new cytotoxic tri- and tetraazabenzo[3,2-a]fluorene-5,6-dione derivatives.

Leepasert T, Shahabi M, Shanab K, Schirmer E, Holzer W, Spreitzer H, Aicher B, Müller G, Günther E.

Bioorg Med Chem Lett. 2013 Oct 1;23(19):5264-6. doi: 10.1016/j.bmcl.2013.08.021. Epub 2013 Aug 13.

PMID:
23988351
15.

Addition of lithium carbenoids to isocyanates: a direct access to synthetically useful N-substituted 2-haloacetamides.

Pace V, Castoldi L, Holzer W.

Chem Commun (Camb). 2013 Sep 28;49(75):8383-5. doi: 10.1039/c3cc44255a.

PMID:
23938607
16.

Synthesis of α,β-unsaturated α'-haloketones through the chemoselective addition of halomethyllithiums to Weinreb amides.

Pace V, Castoldi L, Holzer W.

J Org Chem. 2013 Aug 2;78(15):7764-70. doi: 10.1021/jo401236t. Epub 2013 Jul 16.

PMID:
23805887
17.

Chemoselective CaO-mediated acylation of alcohols and amines in 2-methyltetrahydrofuran.

Pace V, Hoyos P, Alcántara AR, Holzer W.

ChemSusChem. 2013 May;6(5):905-10. doi: 10.1002/cssc.201200922. Epub 2013 Mar 26.

PMID:
23532956
18.

Synthesis and biological evaluation of new cytotoxic indazolo[4,3-gh]isoquinolinone derivatives.

Shahabi M, Schirmer E, Shanab K, Leepasert T, Ruzicka J, Holzer W, Spreitzer H, Aicher B, Schmidt P, Blumenstein L, Müller G, Günther E.

Bioorg Med Chem Lett. 2013 Mar 15;23(6):1846-52. doi: 10.1016/j.bmcl.2013.01.022. Epub 2013 Jan 23.

PMID:
23395656
19.

Dipyrazolo[1,5-a:4',3'-c]pyridines - a new heterocyclic system accessed via multicomponent reaction.

Holzer W, Vilkauskaitė G, Arbačiauskienė E, Sačkus A.

Beilstein J Org Chem. 2012;8:2223-9. doi: 10.3762/bjoc.8.251. Epub 2012 Dec 27.

20.

Highly efficient and chemoselective α-iodination of acrylate esters through Morita-Baylis-Hillman-type chemistry.

Pace V, Vilkauskaitė G, Šačkus A, Holzer W.

Org Biomol Chem. 2013 Feb 21;11(7):1085-8. doi: 10.1039/c2ob27341a.

PMID:
23303274
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