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Items: 1 to 20 of 108

1.

Dose-dependent sigma-1 receptor occupancy by donepezil in rat brain can be assessed with (11)C-SA4503 and microPET.

Ramakrishnan NK, Visser AK, Schepers M, Luurtsema G, Nyakas CJ, Elsinga PH, Ishiwata K, Dierckx RA, van Waarde A.

Psychopharmacology (Berl). 2014 Oct;231(20):3997-4006. doi: 10.1007/s00213-014-3533-2. Epub 2014 Mar 18. Erratum in: Psychopharmacology (Berl). 2014 Oct;231(20):4085.

PMID:
24639047
2.

High occupancy of sigma1 receptors in the human brain after single oral administration of donepezil: a positron emission tomography study using [11C]SA4503.

Ishikawa M, Sakata M, Ishii K, Kimura Y, Oda K, Toyohara J, Wu J, Ishiwata K, Iyo M, Hashimoto K.

Int J Neuropsychopharmacol. 2009 Sep;12(8):1127-31. doi: 10.1017/S1461145709990204. Epub 2009 Jul 2.

PMID:
19573265
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5.

Distribution of intravenously administered acetylcholinesterase inhibitor and acetylcholinesterase activity in the adrenal gland: 11C-donepezil PET study in the normal rat.

Watabe T, Naka S, Ikeda H, Horitsugi G, Kanai Y, Isohashi K, Ishibashi M, Kato H, Shimosegawa E, Watabe H, Hatazawa J.

PLoS One. 2014 Sep 16;9(9):e107427. doi: 10.1371/journal.pone.0107427. eCollection 2014.

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In vivo visualization of donepezil binding in the brain of patients with Alzheimer's disease.

Okamura N, Funaki Y, Tashiro M, Kato M, Ishikawa Y, Maruyama M, Ishikawa H, Meguro K, Iwata R, Yanai K.

Br J Clin Pharmacol. 2008 Apr;65(4):472-9. Epub 2007 Dec 7.

8.

Cutamesine Overcomes REM Sleep Deprivation-Induced Memory Loss: Relationship to Sigma-1 Receptor Occupancy.

Ramakrishnan NK, Schepers M, Luurtsema G, Nyakas CJ, Elsinga PH, Ishiwata K, Dierckx RA, van Waarde A.

Mol Imaging Biol. 2015 Jun;17(3):364-72. doi: 10.1007/s11307-014-0808-2.

PMID:
25449772
10.

Safety and tolerability of donepezil at doses up to 20 mg/day: results from a pilot study in patients with Alzheimer's disease.

Doody RS, Corey-Bloom J, Zhang R, Li H, Ieni J, Schindler R.

Drugs Aging. 2008;25(2):163-74.

PMID:
18257603
11.

Evaluation of the binding characteristics of [5-(11)C-methoxy]Donepezil in the rat brain for in vivo visualization of acetylcholinesterase.

Funaki Y, Kato M, Iwata R, Sakurai E, Sakurai E, Tashiro M, Ido T, Yanai K.

J Pharmacol Sci. 2003 Feb;91(2):105-12.

12.

Pridopidine selectively occupies sigma-1 rather than dopamine D2 receptors at behaviorally active doses.

Sahlholm K, Sijbesma JW, Maas B, Kwizera C, Marcellino D, Ramakrishnan NK, Dierckx RA, Elsinga PH, van Waarde A.

Psychopharmacology (Berl). 2015 Sep;232(18):3443-53. doi: 10.1007/s00213-015-3997-8. Epub 2015 Jul 11.

13.

Pharmacokinetic and pharmacodynamic properties of cholinesterase inhibitors donepezil, tacrine, and galantamine in aged and young Lister hooded rats.

Goh CW, Aw CC, Lee JH, Chen CP, Browne ER.

Drug Metab Dispos. 2011 Mar;39(3):402-11. doi: 10.1124/dmd.110.035964. Epub 2010 Dec 8.

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Small-animal PET with a σ-ligand, 11C-SA4503, detects spontaneous pituitary tumors in aged rats.

Ramakrishnan NK, Rybczynska AA, Visser AK, Marosi K, Nyakas CJ, Kwizera C, Sijbesma JW, Elsinga PH, Ishiwata K, Pruim J, Dierckx RA, van Waarde A.

J Nucl Med. 2013 Aug;54(8):1377-83. doi: 10.2967/jnumed.112.115931. Epub 2013 Jun 19.

16.

Estimation of plasma IC50 of donepezil hydrochloride for brain acetylcholinesterase inhibition in monkey using N-[11C]methylpiperidin-4-yl acetate ([11C]MP4A) and PET.

Shiraishi T, Kikuchi T, Fukushi K, Shinotoh H, Nagatsuka S, Tanaka N, Ota T, Sato K, Hirano S, Tanada S, Iyo M, Irie T.

Neuropsychopharmacology. 2005 Dec;30(12):2154-61.

17.

Pharmacokinetic and pharmacodynamic profile of donepezil HCl following single oral doses.

Rogers SL, Friedhoff LT.

Br J Clin Pharmacol. 1998 Nov;46 Suppl 1:1-6.

18.

High occupancy of sigma-1 receptors in the human brain after single oral administration of fluvoxamine: a positron emission tomography study using [11C]SA4503.

Ishikawa M, Ishiwata K, Ishii K, Kimura Y, Sakata M, Naganawa M, Oda K, Miyatake R, Fujisaki M, Shimizu E, Shirayama Y, Iyo M, Hashimoto K.

Biol Psychiatry. 2007 Oct 15;62(8):878-83. Epub 2007 Jul 30.

PMID:
17662961
19.

Quantitative analysis of donepezil binding to acetylcholinesterase using positron emission tomography and [5-(11)C-methoxy]donepezil.

Hiraoka K, Okamura N, Funaki Y, Watanuki S, Tashiro M, Kato M, Hayashi A, Hosokai Y, Yamasaki H, Fujii T, Mori E, Yanai K, Watabe H.

Neuroimage. 2009 Jul 1;46(3):616-23. doi: 10.1016/j.neuroimage.2009.03.006. Epub 2009 Mar 12.

PMID:
19286462
20.

Binding properties of SA4503, a novel and selective sigma 1 receptor agonist.

Matsuno K, Nakazawa M, Okamoto K, Kawashima Y, Mita S.

Eur J Pharmacol. 1996 Jun 13;306(1-3):271-9.

PMID:
8813641
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