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Results: 1 to 20 of 90

1.

Grassypeptolides as natural inhibitors of dipeptidyl peptidase 8 and T-cell activation.

Kwan JC, Liu Y, Ratnayake R, Hatano R, Kuribara A, Morimoto C, Ohnuma K, Paul VJ, Ye T, Luesch H.

Chembiochem. 2014 Apr 14;15(6):799-804. doi: 10.1002/cbic.201300762. Epub 2014 Mar 3.

PMID:
24591193
[PubMed - in process]
2.

Dipeptidyl peptidase IV inhibition for the treatment of type 2 diabetes: potential importance of selectivity over dipeptidyl peptidases 8 and 9.

Lankas GR, Leiting B, Roy RS, Eiermann GJ, Beconi MG, Biftu T, Chan CC, Edmondson S, Feeney WP, He H, Ippolito DE, Kim D, Lyons KA, Ok HO, Patel RA, Petrov AN, Pryor KA, Qian X, Reigle L, Woods A, Wu JK, Zaller D, Zhang X, Zhu L, Weber AE, Thornberry NA.

Diabetes. 2005 Oct;54(10):2988-94.

PMID:
16186403
[PubMed - indexed for MEDLINE]
Free Article
3.

DPP8 and DPP9 expression in cynomolgus monkey and Sprague Dawley rat tissues.

Harstad EB, Rosenblum JS, Gorrell MD, Achanzar WE, Minimo L, Wu J, Rosini-Marthaler L, Gullo R, Ordway ND, Kirby MS, Chadwick KD, Cosma GN, Moyer CF.

Regul Pept. 2013 Sep 10;186:26-35. doi: 10.1016/j.regpep.2013.07.003. Epub 2013 Jul 12.

PMID:
23850796
[PubMed - indexed for MEDLINE]
4.

Docking-based 3D-QSAR study for selectivity of DPP4, DPP8, and DPP9 inhibitors.

Kang NS, Ahn JH, Kim SS, Chae CH, Yoo SE.

Bioorg Med Chem Lett. 2007 Jul 1;17(13):3716-21. Epub 2007 Apr 13.

PMID:
17462890
[PubMed - indexed for MEDLINE]
5.

Dipeptidyl peptidase inhibitors, an emerging drug class for inflammatory disease?

Yazbeck R, Howarth GS, Abbott CA.

Trends Pharmacol Sci. 2009 Nov;30(11):600-7. doi: 10.1016/j.tips.2009.08.003. Review.

PMID:
19837468
[PubMed - indexed for MEDLINE]
6.

Dipeptidyl peptidase 8/9-like activity in human leukocytes.

Maes MB, Dubois V, Brandt I, Lambeir AM, Van der Veken P, Augustyns K, Cheng JD, Chen X, Scharpé S, De Meester I.

J Leukoc Biol. 2007 May;81(5):1252-7. Epub 2007 Feb 7.

PMID:
17287297
[PubMed - indexed for MEDLINE]
Free Article
7.

Cloning and characterization of dipeptidyl peptidase 10, a new member of an emerging subgroup of serine proteases.

Qi SY, Riviere PJ, Trojnar J, Junien JL, Akinsanya KO.

Biochem J. 2003 Jul 1;373(Pt 1):179-89.

PMID:
12662155
[PubMed - indexed for MEDLINE]
Free PMC Article
8.

Regulation of dipeptidyl peptidase 8 and 9 expression in activated lymphocytes and injured liver.

Chowdhury S, Chen Y, Yao TW, Ajami K, Wang XM, Popov Y, Schuppan D, Bertolino P, McCaughan GW, Yu DM, Gorrell MD.

World J Gastroenterol. 2013 May 21;19(19):2883-93. doi: 10.3748/wjg.v19.i19.2883.

PMID:
23704821
[PubMed - indexed for MEDLINE]
Free PMC Article
9.

Glutamic acid analogues as potent dipeptidyl peptidase IV and 8 inhibitors.

Lu IL, Lee SJ, Tsu H, Wu SY, Kao KH, Chien CH, Chang YY, Chen YS, Cheng JH, Chang CN, Chen TW, Chang SP, Chen X, Jiaang WT.

Bioorg Med Chem Lett. 2005 Jul 1;15(13):3271-5.

PMID:
15927466
[PubMed - indexed for MEDLINE]
10.

Current advances and therapeutic potential of agents targeting dipeptidyl peptidases-IV, -II, 8/9 and fibroblast activation protein.

Chen SJ, Jiaang WT.

Curr Top Med Chem. 2011;11(12):1447-63. Review.

PMID:
21510839
[PubMed - indexed for MEDLINE]
11.

Structure-activity relationship studies on isoindoline inhibitors of dipeptidyl peptidases 8 and 9 (DPP8, DPP9): is DPP8-selectivity an attainable goal?

Van Goethem S, Matheeussen V, Joossens J, Lambeir AM, Chen X, De Meester I, Haemers A, Augustyns K, Van der Veken P.

J Med Chem. 2011 Aug 25;54(16):5737-46. doi: 10.1021/jm200383j. Epub 2011 Aug 2.

PMID:
21711053
[PubMed - indexed for MEDLINE]
12.

Pharmacological profile of ASP8497, a novel, selective, and competitive dipeptidyl peptidase-IV inhibitor, in vitro and in vivo.

Someya Y, Tahara A, Nakano R, Matsuyama-Yokono A, Nagase I, Fukunaga Y, Takasu T, Hayakawa M, Shibasaki M.

Naunyn Schmiedebergs Arch Pharmacol. 2008 May;377(3):209-17. doi: 10.1007/s00210-008-0277-8. Epub 2008 Apr 9.

PMID:
18398600
[PubMed - indexed for MEDLINE]
13.

Potency, selectivity and prolonged binding of saxagliptin to DPP4: maintenance of DPP4 inhibition by saxagliptin in vitro and ex vivo when compared to a rapidly-dissociating DPP4 inhibitor.

Wang A, Dorso C, Kopcho L, Locke G, Langish R, Harstad E, Shipkova P, Marcinkeviciene J, Hamann L, Kirby MS.

BMC Pharmacol. 2012 Apr 4;12:2. doi: 10.1186/1471-2210-12-2.

PMID:
22475049
[PubMed - indexed for MEDLINE]
Free PMC Article
14.

Expression and spatial heterogeneity of dipeptidyl peptidases in endothelial cells of conduct vessels and capillaries.

Matheeussen V, Baerts L, De Meyer G, De Keulenaer G, Van der Veken P, Augustyns K, Dubois V, Scharpé S, De Meester I.

Biol Chem. 2011 Mar;392(3):189-98. doi: 10.1515/BC.2011.002.

PMID:
21194356
[PubMed - indexed for MEDLINE]
15.

Cloning, expression and chromosomal localization of a novel human dipeptidyl peptidase (DPP) IV homolog, DPP8.

Abbott CA, Yu DM, Woollatt E, Sutherland GR, McCaughan GW, Gorrell MD.

Eur J Biochem. 2000 Oct;267(20):6140-50.

PMID:
11012666
[PubMed - indexed for MEDLINE]
Free Article
16.

The SUMO1-E67 interacting loop peptide is an allosteric inhibitor of the dipeptidyl peptidases 8 and 9.

Pilla E, Kilisch M, Lenz C, Urlaub H, Geiss-Friedlander R.

J Biol Chem. 2013 Nov 8;288(45):32787-96. doi: 10.1074/jbc.M113.489179. Epub 2013 Sep 26.

PMID:
24072711
[PubMed - indexed for MEDLINE]
17.

Prolyl peptidases related to dipeptidyl peptidase IV: potential of specific inhibitors in drug discovery.

Van der Veken P, Haemers A, Augustyns K.

Curr Top Med Chem. 2007;7(6):621-35. Review.

PMID:
17352682
[PubMed - indexed for MEDLINE]
18.

Recent insights into the role of dipeptidyl aminopeptidase IV (DPIV) and aminopeptidase N (APN) families in immune functions.

Ansorge S, Bank U, Heimburg A, Helmuth M, Koch G, Tadje J, Lendeckel U, Wolke C, Neubert K, Faust J, Fuchs P, Reinhold D, Thielitz A, Täger M.

Clin Chem Lab Med. 2009;47(3):253-61. doi: 10.1515/CCLM.2009.063. Review.

PMID:
19327105
[PubMed - indexed for MEDLINE]
19.

Inhibitors of dipeptidyl peptidase 8 and dipeptidyl peptidase 9. Part 2: isoindoline containing inhibitors.

Van Goethem S, Van der Veken P, Dubois V, Soroka A, Lambeir AM, Chen X, Haemers A, Scharpé S, De Meester I, Augustyns K.

Bioorg Med Chem Lett. 2008 Jul 15;18(14):4159-62. doi: 10.1016/j.bmcl.2008.05.079. Epub 2008 May 24.

PMID:
18556198
[PubMed - indexed for MEDLINE]
20.

Dipeptidyl peptidase IV: development, design, synthesis and biological evaluation of inhibitors.

Borloo M, De Meester I.

Verh K Acad Geneeskd Belg. 1994;56(1):57-88. Review.

PMID:
7911611
[PubMed - indexed for MEDLINE]

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