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Items: 1 to 20 of 104

1.

A tetradecapeptide somatostatin dicarba-analog: Synthesis, structural impact and biological activity.

Martín-Gago P, Ramón R, Aragón E, Fernández-Carneado J, Martin-Malpartida P, Verdaguer X, López-Ruiz P, Colás B, Cortes MA, Ponsati B, Macias MJ, Riera A.

Bioorg Med Chem Lett. 2014 Jan 1;24(1):103-7. doi: 10.1016/j.bmcl.2013.11.065. Epub 2013 Dec 3.

PMID:
24342240
2.

Human somatostatin receptor specificity of backbone-cyclic analogues containing novel sulfur building units.

Gazal S, Gelerman G, Ziv O, Karpov O, Litman P, Bracha M, Afargan M, Gilon C.

J Med Chem. 2002 Apr 11;45(8):1665-71.

PMID:
11931620
3.

Identification of potent non-peptide somatostatin antagonists with sst(3) selectivity.

Poitout L, Roubert P, Contour-Galcéra MO, Moinet C, Lannoy J, Pommier J, Plas P, Bigg D, Thurieau C.

J Med Chem. 2001 Aug 30;44(18):2990-3000.

PMID:
11520208
4.

Lanthionine-somatostatin analogs: synthesis, characterization, biological activity, and enzymatic stability studies.

Osapay G, Prokai L, Kim HS, Medzihradszky KF, Coy DH, Liapakis G, Reisine T, Melacini G, Zhu Q, Wang SH, Mattern RH, Goodman M.

J Med Chem. 1997 Jul 4;40(14):2241-51.

PMID:
9216843
5.

Novel sst5-selective somatostatin dicarba-analogues: synthesis and conformation-affinity relationships.

D'Addona D, Carotenuto A, Novellino E, Piccand V, Reubi JC, Di Cianni A, Gori F, Papini AM, Ginanneschi M.

J Med Chem. 2008 Feb 14;51(3):512-20. doi: 10.1021/jm070886i. Epub 2008 Jan 23.

PMID:
18210999
6.

Highly potent and subtype selective ligands derived by N-methyl scan of a somatostatin antagonist.

Rajeswaran WG, Hocart SJ, Murphy WA, Taylor JE, Coy DH.

J Med Chem. 2001 Apr 12;44(8):1305-11.

PMID:
11312929
7.

A bicyclic and hsst2 selective somatostatin analogue: design, synthesis, conformational analysis and binding.

Falb E, Salitra Y, Yechezkel T, Bracha M, Litman P, Olender R, Rosenfeld R, Senderowitz H, Jiang S, Goodman M.

Bioorg Med Chem. 2001 Dec;9(12):3255-64.

PMID:
11711301
8.

SSTR1- and SSTR3-selective somatostatin analogues.

Ramón R, Martín-Gago P, Verdaguer X, Macias MJ, Martin-Malpartida P, Fernández-Carneado J, Gomez-Caminals M, Ponsati B, López-Ruiz P, Cortés MA, Colás B, Riera A.

Chembiochem. 2011 Mar 7;12(4):625-32. doi: 10.1002/cbic.201000597. Epub 2011 Jan 21.

PMID:
21259412
9.

Cloned somatostatin receptors: identification of subtype-selective peptides and demonstration of high affinity binding of linear peptides.

Raynor K, Murphy WA, Coy DH, Taylor JE, Moreau JP, Yasuda K, Bell GI, Reisine T.

Mol Pharmacol. 1993 Jun;43(6):838-44.

PMID:
8100350
10.

Synthesis and biological activity of a cyclic pseudohexapeptide analog of somatostatin.

Gero TW, Spatola AF, Torres-Aleman I, Schally AV.

Biochem Biophys Res Commun. 1984 May 16;120(3):840-5.

PMID:
6145411
12.

A bioactive somatostatin analog without a type II' beta-turn: synthesis and conformational analysis in solution.

Jiang S, Gazal S, Gelerman G, Ziv O, Karpov O, Litman P, Bracha M, Afargan M, Gilon C, Goodman M.

J Pept Sci. 2001 Oct;7(10):521-8.

PMID:
11695647
13.

Design, synthesis, and biological activities of potent and selective somatostatin analogues incorporating novel peptoid residues.

Tran TA, Mattern RH, Afargan M, Amitay O, Ziv O, Morgan BA, Taylor JE, Hoyer D, Goodman M.

J Med Chem. 1998 Jul 16;41(15):2679-85.

PMID:
9667958
14.

Cyclic hexapeptide analogs of somatostatin containing bridge modifications. Syntheses and conformational analyses.

Huang Z, Pröbstl A, Spencer JR, Yamazaki T, Goodman M.

Int J Pept Protein Res. 1993 Oct;42(4):352-65.

PMID:
7902342
15.
16.

Potent somatostatin undecapeptide agonists selective for somatostatin receptor 1 (sst1).

Rivier JE, Hoeger C, Erchegyi J, Gulyas J, DeBoard R, Craig AG, Koerber SC, Wenger S, Waser B, Schaer JC, Reubi JC.

J Med Chem. 2001 Jun 21;44(13):2238-46.

PMID:
11405660
17.

Novel sst(4)-selective somatostatin (SRIF) agonists. 2. Analogues with beta-methyl-3-(2-naphthyl)alanine substitutions at position 8.

Erchegyi J, Penke B, Simon L, Michaelson S, Wenger S, Waser B, Cescato R, Schaer JC, Reubi JC, Rivier J.

J Med Chem. 2003 Dec 18;46(26):5587-96.

PMID:
14667213
18.

Discovery of iodinated somatostatin analogues selective for hsst2 and hsst5 with excellent inhibition of growth hormone and prolactin release from rat pituitary cells.

Moore SB, van der Hoek J, de Capua A, van Koetsveld PM, Hofland LJ, Lamberts SW, Goodman M.

J Med Chem. 2005 Oct 20;48(21):6643-52.

PMID:
16220980
19.

Synthesis of somatostatin mimetics based on the 1-deoxymannojirimycin scaffold.

Gouin SG, Murphy PV.

J Org Chem. 2005 Oct 14;70(21):8527-32.

PMID:
16209603
20.

A light-activated beta-turn scaffold within a somatostatin analog: NMR structure and biological activity.

Ulysse LG Jr, Chmielewski J.

Chem Biol Drug Des. 2006 Feb;67(2):127-36.

PMID:
16492160
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