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Results: 1 to 20 of 101

1.

Design, synthesis and molecular modelling studies of novel 3-acetamido-4-methyl benzoic acid derivatives as inhibitors of protein tyrosine phosphatase 1B.

Rakse M, Karthikeyan C, Deora GS, Moorthy NS, Rathore V, Rawat AK, Srivastava AK, Trivedi P.

Eur J Med Chem. 2013 Dec;70:469-76. doi: 10.1016/j.ejmech.2013.10.030. Epub 2013 Oct 23.

PMID:
24185377
[PubMed - in process]
2.

Docking of oxalyl aryl amino benzoic acid derivatives into PTP1B.

Verma N, Mittal M, Verma RK.

Bioinformation. 2008;3(2):83-8. Epub 2008 Oct 25.

PMID:
19238234
[PubMed]
Free PMC Article
3.

Synthesis and biological evaluation of 2,4,6-trihydroxychalcone derivatives as novel protein tyrosine phosphatase 1B inhibitors.

Sun LP, Gao LX, Ma WP, Nan FJ, Li J, Piao HR.

Chem Biol Drug Des. 2012 Oct;80(4):584-90. doi: 10.1111/j.1747-0285.2012.01431.x. Epub 2012 Jul 13.

PMID:
22805439
[PubMed - indexed for MEDLINE]
4.

A novel strategy for the development of selective active-site inhibitors of the protein tyrosine phosphatase-like proteins islet-cell antigen 512 (IA-2) and phogrin (IA-2beta).

Drake PG, Peters GH, Andersen HS, Hendriks W, Møller NP.

Biochem J. 2003 Jul 15;373(Pt 2):393-401.

PMID:
12697028
[PubMed - indexed for MEDLINE]
Free PMC Article
5.

Synthesis and biological evaluation of oleanolic acid derivatives as inhibitors of protein tyrosine phosphatase 1B.

Qian S, Li H, Chen Y, Zhang W, Yang S, Wu Y.

J Nat Prod. 2010 Nov 29;73(11):1743-50. doi: 10.1021/np100064m. Epub 2010 Oct 21.

PMID:
20964318
[PubMed - indexed for MEDLINE]
6.

Molecular docking and high-throughput screening for novel inhibitors of protein tyrosine phosphatase-1B.

Doman TN, McGovern SL, Witherbee BJ, Kasten TP, Kurumbail R, Stallings WC, Connolly DT, Shoichet BK.

J Med Chem. 2002 May 23;45(11):2213-21.

PMID:
12014959
[PubMed - indexed for MEDLINE]
7.

Design, synthesis and docking study of 5-(substituted benzylidene)thiazolidine-2,4-dione derivatives as inhibitors of protein tyrosine phosphatase 1B.

Wang Z, Liu Z, Lee W, Kim SN, Yoon G, Cheon SH.

Bioorg Med Chem Lett. 2014 Aug 1;24(15):3337-40. doi: 10.1016/j.bmcl.2014.05.099. Epub 2014 Jun 6.

PMID:
24953600
[PubMed - in process]
8.

1H-2,3-dihydroperimidine derivatives: a new class of potent protein tyrosine phosphatase 1B inhibitors.

Wang WL, Yang DL, Gao LX, Tang CL, Ma WP, Ye HH, Zhang SQ, Zhao YN, Xu HJ, Hu Z, Chen X, Fan WH, Chen HJ, Li JY, Nan FJ, Li J, Feng B.

Molecules. 2013 Dec 23;19(1):102-21. doi: 10.3390/molecules19010102.

PMID:
24366088
[PubMed - in process]
Free Article
9.

Design, synthesis, and evaluation of bromo-retrochalcone derivatives as protein tyrosine phosphatase 1B inhibitors.

Liu Z, Lee W, Kim SN, Yoon G, Cheon SH.

Bioorg Med Chem Lett. 2011 Jun 15;21(12):3755-8. doi: 10.1016/j.bmcl.2011.04.057. Epub 2011 Apr 23.

PMID:
21555221
[PubMed - indexed for MEDLINE]
10.

Synthesis and biological evaluation of 4,4-dimethyl lithocholic acid derivatives as novel inhibitors of protein tyrosine phosphatase 1B.

He HB, Gao LX, Deng QF, Ma WP, Tang CL, Qiu WW, Tang J, Li JY, Li J, Yang F.

Bioorg Med Chem Lett. 2012 Dec 1;22(23):7237-42. doi: 10.1016/j.bmcl.2012.09.040. Epub 2012 Sep 21.

PMID:
23067554
[PubMed - indexed for MEDLINE]
11.

Synthesis and biological evaluation of heterocyclic ring-substituted maslinic acid derivatives as novel inhibitors of protein tyrosine phosphatase 1B.

Qiu WW, Shen Q, Yang F, Wang B, Zou H, Li JY, Li J, Tang J.

Bioorg Med Chem Lett. 2009 Dec 1;19(23):6618-22. doi: 10.1016/j.bmcl.2009.10.017. Epub 2009 Oct 8.

PMID:
19846303
[PubMed - indexed for MEDLINE]
12.

Synthesis and evaluation of oxovanadium(IV) complexes of Schiff-base condensates from 5-substituted-2-hydroxybenzaldehyde and 2-substituted-benzenamine as selective inhibitors of protein tyrosine phosphatase 1B.

Han H, Lu L, Wang Q, Zhu M, Yuan C, Xing S, Fu X.

Dalton Trans. 2012 Aug 28;41(36):11116-24. doi: 10.1039/c2dt30198a.

PMID:
22864521
[PubMed - indexed for MEDLINE]
13.

Design, synthesis, and biological evaluation of bromophenol derivatives as protein tyrosine phosphatase 1B inhibitors.

Jiang B, Shi D, Cui Y, Guo S.

Arch Pharm (Weinheim). 2012 Jun;345(6):444-53. doi: 10.1002/ardp.201100373. Epub 2012 Feb 3.

PMID:
22307562
[PubMed - indexed for MEDLINE]
14.

Molecular docking and 3D-QSAR on 2-(oxalylamino) benzoic acid and its analogues as protein tyrosine phosphatase 1B inhibitors.

Zhou M, Ji M.

Bioorg Med Chem Lett. 2005 Dec 15;15(24):5521-5. Epub 2005 Oct 17.

PMID:
16230012
[PubMed - indexed for MEDLINE]
15.

Design, synthesis, and discovery of stilbene derivatives based on lithospermic acid B as potent protein tyrosine phosphatase 1B inhibitors.

Jung M, Lee Y, Park M, Kim H, Kim H, Lim E, Tak J, Sim M, Lee D, Park N, Oh WK, Hur KY, Kang ES, Lee HC.

Bioorg Med Chem Lett. 2007 Aug 15;17(16):4481-6. Epub 2007 Jun 8.

PMID:
17596944
[PubMed - indexed for MEDLINE]
16.

[Design, synthesis and evaluation of malonic acid-based PTP1B inhibitors].

Du X, Zhang SE, Liu JZ, Nie FL, Ye F, Tian JY, Xiao ZY.

Yao Xue Xue Bao. 2012 Mar;47(3):367-73. Chinese.

PMID:
22645761
[PubMed - indexed for MEDLINE]
17.

Preparation of triazole-linked glycosylated α-ketocarboxylic acid derivatives as new PTP1B inhibitors.

Song Z, He XP, Li C, Gao LX, Wang ZX, Tang Y, Xie J, Li J, Chen GR.

Carbohydr Res. 2011 Jan 3;346(1):140-5. doi: 10.1016/j.carres.2010.10.023. Epub 2010 Oct 30.

PMID:
21111404
[PubMed - indexed for MEDLINE]
18.

Synthesis and acrosin inhibitory activity of methyl 5-substituted-1H-benzo[d]imidazol-2-yl carbamate derivatives.

Liu X, Chen Q, Zhu J, Fan Y, Ding L, Zhao J, Han G, Tian W, Qi J, Zhou Y, Lv J.

Bioorg Med Chem Lett. 2012 May 15;22(10):3554-9. doi: 10.1016/j.bmcl.2012.03.042. Epub 2012 Mar 21.

PMID:
22507960
[PubMed - indexed for MEDLINE]
19.

Potent α-glucosidase and protein tyrosine phosphatase 1B inhibitors from Artemisia capillaris.

Nurul Islam M, Jung HA, Sohn HS, Kim HM, Choi JS.

Arch Pharm Res. 2013 May;36(5):542-52. doi: 10.1007/s12272-013-0069-7. Epub 2013 Feb 24.

PMID:
23435948
[PubMed - indexed for MEDLINE]
20.

Synthesis and biological evaluation of (±)-3-(2-(2-fluorobenzyloxy) naphthalen-6-yl)-2-aminopropanoic acid derivatives as novel PTP1B inhibitors.

Sun LP, Shen Q, Piao HH, Ma WP, Gao LX, Zhang W, Nan FJ, Li J, Piao HR.

Eur J Med Chem. 2011 Sep;46(9):3630-8. doi: 10.1016/j.ejmech.2011.05.027. Epub 2011 May 20.

PMID:
21680062
[PubMed - indexed for MEDLINE]

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