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Results: 1 to 20 of 131

1.

Radiosynthesis of N-(4-chloro-3-[(11)C]methoxyphenyl)-2-picolinamide ([(11)C]ML128) as a PET radiotracer for metabotropic glutamate receptor subtype 4 (mGlu4).

Kil KE, Zhang Z, Jokivarsi K, Gong C, Choi JK, Kura S, Brownell AL.

Bioorg Med Chem. 2013 Oct 1;21(19):5955-62. doi: 10.1016/j.bmc.2013.07.046. Epub 2013 Aug 2.

PMID:
23978356
[PubMed - indexed for MEDLINE]
Free PMC Article
2.

Radiosynthesis and evaluation of an 18F-labeled positron emission tomography (PET) radioligand for metabotropic glutamate receptor subtype 4 (mGlu4).

Kil KE, Poutiainen P, Zhang Z, Zhu A, Choi JK, Jokivarsi K, Brownell AL.

J Med Chem. 2014 Nov 13;57(21):9130-8. doi: 10.1021/jm501245b. Epub 2014 Oct 27.

PMID:
25330258
[PubMed - in process]
Free PMC Article
3.

Radiosynthesis and preclinical evaluation of 11C-ABP688 as a probe for imaging the metabotropic glutamate receptor subtype 5.

Ametamey SM, Kessler LJ, Honer M, Wyss MT, Buck A, Hintermann S, Auberson YP, Gasparini F, Schubiger PA.

J Nucl Med. 2006 Apr;47(4):698-705.

PMID:
16595505
[PubMed - indexed for MEDLINE]
Free Article
4.

Synthesis and preliminary biological evaluation of 3-[(18)F]fluoro-5-(2-pyridinylethynyl)benzonitrile as a PET radiotracer for imaging metabotropic glutamate receptor subtype 5.

Wang JQ, Tueckmantel W, Zhu A, Pellegrino D, Brownell AL.

Synapse. 2007 Dec;61(12):951-61.

PMID:
17787003
[PubMed - indexed for MEDLINE]
5.

Radiolabeling and in vitro and in vivo evaluation of [18F]-FE-DABP688 as a PET radioligand for the metabotropic glutamate receptor subtype 5.

Honer M, Stoffel A, Kessler LJ, Schubiger PA, Ametamey SM.

Nucl Med Biol. 2007 Nov;34(8):973-80. Epub 2007 Sep 19.

PMID:
17998101
[PubMed - indexed for MEDLINE]
6.

Radiosynthesis of PET radiotracer as a prodrug for imaging group II metabotropic glutamate receptors in vivo.

Wang JQ, Zhang Z, Kuruppu D, Brownell AL.

Bioorg Med Chem Lett. 2012 Mar 1;22(5):1958-62. doi: 10.1016/j.bmcl.2012.01.039. Epub 2012 Jan 21.

PMID:
22318160
[PubMed - indexed for MEDLINE]
Free PMC Article
7.

A PET imaging agent with fast kinetics: synthesis and in vivo evaluation of the serotonin transporter ligand [11C]2-[2-dimethylaminomethylphenylthio)]-5-fluorophenylamine ([11C]AFA).

Huang Y, Narendran R, Bae SA, Erritzoe D, Guo N, Zhu Z, Hwang DR, Laruelle M.

Nucl Med Biol. 2004 Aug;31(6):727-38.

PMID:
15246363
[PubMed - indexed for MEDLINE]
8.
9.

In vitro and in vivo evaluation of [11C]MPEPy as a potential PET ligand for mGlu5 receptors.

Severance AJ, Parsey RV, Kumar JS, Underwood MD, Arango V, Majo VJ, Prabhakaran J, Simpson NR, Van Heertum RL, Mann JJ.

Nucl Med Biol. 2006 Nov;33(8):1021-7.

PMID:
17127176
[PubMed - indexed for MEDLINE]
10.

Radiosynthesis and ex vivo evaluation of [11C]-SIB-1553A as a PET radiotracer for beta4 selective subtype nicotinic acetylcholine receptor.

Sobrio F, Quentin T, Dhilly M, Bourdier T, Tymciu S, Debruyne D, Barré L.

Nucl Med Biol. 2008 Apr;35(3):377-85. doi: 10.1016/j.nucmedbio.2007.11.011. Epub 2008 Jan 30.

PMID:
18355694
[PubMed - indexed for MEDLINE]
11.

The new PET imaging agent [11C]AFE is a selective serotonin transporter ligand with fast brain uptake kinetics.

Zhu Z, Guo N, Narendran R, Erritzoe D, Ekelund J, Hwang DR, Bae SA, Laruelle M, Huang Y.

Nucl Med Biol. 2004 Nov;31(8):983-94.

PMID:
15607480
[PubMed - indexed for MEDLINE]
12.

Synthesis, in vitro and in vivo evaluation of [11C]MMTP: a potential PET ligand for mGluR1 receptors.

Prabhakaran J, Majo VJ, Milak MS, Kassir SA, Palner M, Savenkova L, Mali P, Arango V, Mann JJ, Parsey RV, Kumar JS.

Bioorg Med Chem Lett. 2010 Jun 15;20(12):3499-501. doi: 10.1016/j.bmcl.2010.04.146. Epub 2010 May 5.

PMID:
20494576
[PubMed - indexed for MEDLINE]
Free PMC Article
13.

Radiosynthesis and evaluation of [11C]-(+)-4-propyl-3,4,4a,5,6,10b-hexahydro-2H-naphtho[1,2-b][1,4]oxazin-9-ol as a potential radiotracer for in vivo imaging of the dopamine D2 high-affinity state with positron emission tomography.

Wilson AA, McCormick P, Kapur S, Willeit M, Garcia A, Hussey D, Houle S, Seeman P, Ginovart N.

J Med Chem. 2005 Jun 16;48(12):4153-60.

PMID:
15943487
[PubMed - indexed for MEDLINE]
14.

Methoxyphenylethynyl, methoxypyridylethynyl and phenylethynyl derivatives of pyridine: synthesis, radiolabeling and evaluation of new PET ligands for metabotropic glutamate subtype 5 receptors.

Yu M, Tueckmantel W, Wang X, Zhu A, Kozikowski AP, Brownell AL.

Nucl Med Biol. 2005 Aug;32(6):631-40.

PMID:
16026710
[PubMed - indexed for MEDLINE]
15.

In vitro and in vivo evaluation of [18F]-FDEGPECO as a PET tracer for imaging the metabotropic glutamate receptor subtype 5 (mGluR5).

Wanger-Baumann CA, Mu L, Honer M, Belli S, Alf MF, Schubiger PA, Krämer SD, Ametamey SM.

Neuroimage. 2011 Jun 1;56(3):984-91. doi: 10.1016/j.neuroimage.2011.03.024. Epub 2011 Mar 21.

PMID:
21406237
[PubMed - indexed for MEDLINE]
16.

Synthesis, evaluation, and radiolabeling of new potent positive allosteric modulators of the metabotropic glutamate receptor 2 as potential tracers for positron emission tomography imaging.

Andrés JI, Alcázar J, Cid JM, De Angelis M, Iturrino L, Langlois X, Lavreysen H, Trabanco AA, Celen S, Bormans G.

J Med Chem. 2012 Oct 25;55(20):8685-99. doi: 10.1021/jm300912k. Epub 2012 Oct 11.

PMID:
22992024
[PubMed - indexed for MEDLINE]
17.

Discovery of a novel metabotropic glutamate receptor 4 (mGlu4) positive allosteric modulator (PAM) extended probe: Characterization of ML292, a potent and selective mGlu4 PAM which produces efficacy alone or in combination with L-DOPA in preclinical rodent models of Parkinson's disease.

Engers DW, Jones CK, Bubser M, Thompson AD, Blobaum AL, Sheffler DJ, Zamorano R, Carrington SJS, Bridges TM, Morrison RD, Daniels JS, Conn PJ, Lindsley CW, Niswender CM, Hopkins CR.

Probe Reports from the NIH Molecular Libraries Program [Internet]. Bethesda (MD): National Center for Biotechnology Information (US); 2010-.
2012 Apr 02 [updated 2013 Feb 25].

18.

Synthesis and characterization of two PET radioligands for the metabotropic glutamate 1 (mGlu1) receptor.

Huang Y, Narendran R, Bischoff F, Guo N, Bae SA, Hwang DR, Lesage AS, Laruelle M.

Synapse. 2012 Dec;66(12):1002-14. doi: 10.1002/syn.21606. Epub 2012 Sep 29. Erratum in: Synapse. 2013 Feb;67(2):109.

PMID:
22927303
[PubMed - indexed for MEDLINE]
19.

Radiosynthesis and evaluation of [11C]YM-202074 as a PET ligand for imaging the metabotropic glutamate receptor type 1.

Yanamoto K, Konno F, Odawara C, Yamasaki T, Kawamura K, Hatori A, Yui J, Wakizaka H, Nengaki N, Takei M, Zhang MR.

Nucl Med Biol. 2010 Jul;37(5):615-24. doi: 10.1016/j.nucmedbio.2010.03.002. Epub 2010 Apr 24.

PMID:
20610166
[PubMed - indexed for MEDLINE]
20.

Development of new carbon-11 labelled radiotracers for imaging GABAA- and GABAB-benzodiazepine receptors.

Moran MD, Wilson AA, Elmore CS, Parkes J, Ng A, Sadovski O, Graff A, Daskalakis ZJ, Houle S, Chapdelaine MJ, Vasdev N.

Bioorg Med Chem. 2012 Jul 15;20(14):4482-8. doi: 10.1016/j.bmc.2012.05.046. Epub 2012 May 24.

PMID:
22717238
[PubMed - indexed for MEDLINE]
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