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Results: 1 to 20 of 112

1.

Importance of recognition loops B and D in the activation of human 5-HT₃ receptors by 5-HT and meta-chlorophenylbiguanide.

Michaelson SD, Paulsen IM, Kozuska JL, Martin IL, Dunn SM.

Neuropharmacology. 2013 Oct;73:398-403. doi: 10.1016/j.neuropharm.2013.06.017. Epub 2013 Jun 26.

PMID:
23810831
[PubMed - indexed for MEDLINE]
2.

The loop C region of the murine 5-HT3A receptor contributes to the differential actions of 5-hydroxytryptamine and m-chlorophenylbiguanide.

Suryanarayanan A, Joshi PR, Bikádi Z, Mani M, Kulkarni TR, Gaines C, Schulte MK.

Biochemistry. 2005 Jun 28;44(25):9140-9.

PMID:
15966738
[PubMed - indexed for MEDLINE]
3.

A single channel mutation alters agonist efficacy at 5-HT3A and 5-HT3AB receptors.

Thompson AJ, Lummis SC.

Br J Pharmacol. 2013 Sep;170(2):391-402. doi: 10.1111/bph.12287.

PMID:
23822584
[PubMed - indexed for MEDLINE]
Free PMC Article
4.

General anesthetic-induced channel gating enhancement of 5-hydroxytryptamine type 3 receptors depends on receptor subunit composition.

Solt K, Stevens RJ, Davies PA, Raines DE.

J Pharmacol Exp Ther. 2005 Nov;315(2):771-6. Epub 2005 Aug 4.

PMID:
16081679
[PubMed - indexed for MEDLINE]
Free Article
5.

Subunit-dependent inhibition and potentiation of 5-HT3 receptor by the anticancer drug, topotecan.

Nakamura Y, Ishida Y, Yamada T, Kondo M, Shimada S.

J Neurochem. 2013 Apr;125(1):7-15. doi: 10.1111/jnc.12146. Epub 2013 Jan 31.

PMID:
23305320
[PubMed - indexed for MEDLINE]
6.

Modular design of Cys-loop ligand-gated ion channels: functional 5-HT3 and GABA rho1 receptors lacking the large cytoplasmic M3M4 loop.

Jansen M, Bali M, Akabas MH.

J Gen Physiol. 2008 Feb;131(2):137-46. doi: 10.1085/jgp.200709896.

PMID:
18227272
[PubMed - indexed for MEDLINE]
Free PMC Article
7.

Molecular cloning and pharmacological characterization of serotonin 5-HT(3A) receptor subtype in dog.

Jensen TN, Nielsen J, Frederiksen K, Ebert B.

Eur J Pharmacol. 2006 May 24;538(1-3):23-31. Epub 2006 Mar 27.

PMID:
16647053
[PubMed - indexed for MEDLINE]
8.

Co-expression of the 5-HT3B serotonin receptor subunit alters the biophysics of the 5-HT3 receptor.

Hapfelmeier G, Tredt C, Haseneder R, Zieglgänsberger W, Eisensamer B, Rupprecht R, Rammes G.

Biophys J. 2003 Mar;84(3):1720-33.

PMID:
12609874
[PubMed - indexed for MEDLINE]
Free PMC Article
9.

Agonists and antagonists bind to an A-A interface in the heteromeric 5-HT3AB receptor.

Lochner M, Lummis SC.

Biophys J. 2010 Apr 21;98(8):1494-502. doi: 10.1016/j.bpj.2009.12.4313.

PMID:
20409468
[PubMed - indexed for MEDLINE]
Free PMC Article
10.

The 5-hydroxytryptamine type 3 (5-HT3) receptor reveals a novel determinant of single-channel conductance.

Peters JA, Kelley SP, Dunlop JI, Kirkness EF, Hales TG, Lambert JJ.

Biochem Soc Trans. 2004 Jun;32(Pt3):547-52. Review.

PMID:
15157181
[PubMed - indexed for MEDLINE]
11.

Subunit-dependent modulation of the 5-hydroxytryptamine type 3 receptor open-close equilibrium by n-alcohols.

Rüsch D, Musset B, Wulf H, Schuster A, Raines DE.

J Pharmacol Exp Ther. 2007 Jun;321(3):1069-74. Epub 2007 Mar 7.

PMID:
17360702
[PubMed - indexed for MEDLINE]
Free Article
12.

Modulation of human 5-hydroxytryptamine type 3AB receptors by volatile anesthetics and n-alcohols.

Stevens R, Rüsch D, Solt K, Raines DE, Davies PA.

J Pharmacol Exp Ther. 2005 Jul;314(1):338-45. Epub 2005 Apr 14.

PMID:
15831437
[PubMed - indexed for MEDLINE]
Free Article
13.

Different efficacy of specific agonists at 5-HT3 receptor splice variants: the role of the extra six amino acid segment.

Niemeyer MI, Lummis SC.

Br J Pharmacol. 1998 Feb;123(4):661-6.

PMID:
9517385
[PubMed - indexed for MEDLINE]
Free PMC Article
14.

RIC-3 exclusively enhances the surface expression of human homomeric 5-hydroxytryptamine type 3A (5-HT3A) receptors despite direct interactions with 5-HT3A, -C, -D, and -E subunits.

Walstab J, Hammer C, Lasitschka F, Möller D, Connolly CN, Rappold G, Brüss M, Bönisch H, Niesler B.

J Biol Chem. 2010 Aug 27;285(35):26956-65. doi: 10.1074/jbc.M110.122838. Epub 2010 Jun 3.

PMID:
20522555
[PubMed - indexed for MEDLINE]
Free PMC Article
15.

Role of aspartate 298 in mouse 5-HT3A receptor gating and modulation by extracellular Ca2+.

Hu XQ, Lovinger DM.

J Physiol. 2005 Oct 15;568(Pt 2):381-96. Epub 2005 Aug 11.

PMID:
16096341
[PubMed - indexed for MEDLINE]
Free PMC Article
16.

A comprehensive study on the 5-hydroxytryptamine(3A) receptor binding of agonists serotonin and m-chlorophenylbiguanidine.

Hazai E, Joshi P, Skoviak EC, Suryanarayanan A, Schulte MK, Bikadi Z.

Bioorg Med Chem. 2009 Aug 15;17(16):5796-805. doi: 10.1016/j.bmc.2009.07.022. Epub 2009 Jul 16.

PMID:
19640719
[PubMed - indexed for MEDLINE]
17.

Introduction of the 5-HT3B subunit alters the functional properties of 5-HT3 receptors native to neuroblastoma cells.

Stewart A, Davies PA, Kirkness EF, Safa P, Hales TG.

Neuropharmacology. 2003 Feb;44(2):214-23.

PMID:
12623220
[PubMed - indexed for MEDLINE]
18.

The minimum M3-M4 loop length of neurotransmitter-activated pentameric receptors is critical for the structural integrity of cytoplasmic portals.

Baptista-Hon DT, Deeb TZ, Lambert JJ, Peters JA, Hales TG.

J Biol Chem. 2013 Jul 26;288(30):21558-68. doi: 10.1074/jbc.M113.481689. Epub 2013 Jun 5.

PMID:
23740249
[PubMed - indexed for MEDLINE]
Free PMC Article
19.

Isomerization of the proline in the M2-M3 linker is not required for activation of the human 5-HT3A receptor.

Paulsen IM, Martin IL, Dunn SM.

J Neurochem. 2009 Aug;110(3):870-8. doi: 10.1111/j.1471-4159.2009.06180.x. Epub 2009 May 18.

PMID:
19457066
[PubMed - indexed for MEDLINE]
20.

Identification of a domain affecting agonist potency of meta-chlorophenylbiguanide in 5-HT3 receptors.

Mochizuki S, Miyake A, Furuichi K.

Eur J Pharmacol. 1999 Mar 12;369(1):125-32.

PMID:
10204690
[PubMed - indexed for MEDLINE]

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