Format
Items per page
Sort by

Send to:

Choose Destination

Results: 1 to 20 of 77

Similar articles for PubMed (Select 23462137)

1.

Structural basis for vitamin D receptor agonism by novel non-secosteroidal ligands.

Asano L, Ito I, Kuwabara N, Waku T, Yanagisawa J, Miyachi H, Shimizu T.

FEBS Lett. 2013 Apr 2;587(7):957-63. doi: 10.1016/j.febslet.2013.02.028. Epub 2013 Feb 24.

2.

Structural basis for the accommodation of bis- and tris-aromatic derivatives in vitamin D nuclear receptor.

Ciesielski F, Sato Y, Chebaro Y, Moras D, Dejaegere A, Rochel N.

J Med Chem. 2012 Oct 11;55(19):8440-9. doi: 10.1021/jm300858s. Epub 2012 Sep 19.

PMID:
22957834
3.

Critical role of helix 12 of the vitamin D(3) receptor for the partial agonism of carboxylic ester antagonists.

Väisänen S, Peräkylä M, Kärkkäinen JI, Steinmeyer A, Carlberg C.

J Mol Biol. 2002 Jan 11;315(2):229-38.

PMID:
11779241
4.

Synthetically accessible non-secosteroidal hybrid molecules combining vitamin D receptor agonism and histone deacetylase inhibition.

Fischer J, Wang TT, Kaldre D, Rochel N, Moras D, White JH, Gleason JL.

Chem Biol. 2012 Aug 24;19(8):963-71. doi: 10.1016/j.chembiol.2012.05.024.

6.

Corepressor excess shifts the two-side chain vitamin D analog Gemini from an agonist to an inverse agonist of the vitamin D receptor.

Gonzalez MM, Samenfeld P, Peräkylä M, Carlberg C.

Mol Endocrinol. 2003 Oct;17(10):2028-38. Epub 2003 Jul 3.

PMID:
12843209
7.

A structural basis for the species-specific antagonism of 26,23-lactones on vitamin D signaling.

Peräkylä M, Molnár F, Carlberg C.

Chem Biol. 2004 Aug;11(8):1147-56.

PMID:
15324816
8.

Crystal structures of rat vitamin D receptor bound to adamantyl vitamin D analogs: structural basis for vitamin D receptor antagonism and partial agonism.

Nakabayashi M, Yamada S, Yoshimoto N, Tanaka T, Igarashi M, Ikura T, Ito N, Makishima M, Tokiwa H, DeLuca HF, Shimizu M.

J Med Chem. 2008 Sep 11;51(17):5320-9. doi: 10.1021/jm8004477. Epub 2008 Aug 19.

PMID:
18710208
10.

Ligand binding domain of vitamin D receptors.

Rochel N, Moras D.

Curr Top Med Chem. 2006;6(12):1229-41. Review.

PMID:
16848737
11.

Effects of fluorines on nonsecosteroidal vitamin D receptor agonists.

Kashiwagi H, Ohta M, Ono Y, Morikami K, Itoh S, Sato H, Takahashi T.

Bioorg Med Chem. 2013 Feb 1;21(3):712-21. doi: 10.1016/j.bmc.2012.11.029. Epub 2012 Dec 2.

PMID:
23266184
12.

Ligand recognition by the vitamin D receptor.

Choi M, Yamamoto K, Masuno H, Nakashima K, Taga T, Yamada S.

Bioorg Med Chem. 2001 Jul;9(7):1721-30.

PMID:
11425573
13.

Three-dimensional modeling of and ligand docking to vitamin D receptor ligand binding domain.

Yamamoto K, Masuno H, Choi M, Nakashima K, Taga T, Ooizumi H, Umesono K, Sicinska W, VanHooke J, DeLuca HF, Yamada S.

Proc Natl Acad Sci U S A. 2000 Feb 15;97(4):1467-72.

14.

Adaptability of the Vitamin D nuclear receptor to the synthetic ligand Gemini: remodelling the LBP with one side chain rotation.

Ciesielski F, Rochel N, Moras D.

J Steroid Biochem Mol Biol. 2007 Mar;103(3-5):235-42. Epub 2007 Jan 10.

PMID:
17218092
15.

Hydrogen/deuterium exchange reveals distinct agonist/partial agonist receptor dynamics within vitamin D receptor/retinoid X receptor heterodimer.

Zhang J, Chalmers MJ, Stayrook KR, Burris LL, Garcia-Ordonez RD, Pascal BD, Burris TP, Dodge JA, Griffin PR.

Structure. 2010 Oct 13;18(10):1332-41. doi: 10.1016/j.str.2010.07.007.

16.

Applications of the Vitamin D sterol-Vitamin D receptor (VDR) conformational ensemble model.

Mizwicki MT, Bishop JE, Norman AW.

Steroids. 2005 May-Jun;70(5-7):464-71. Epub 2005 Apr 8.

PMID:
15862832
17.

Combination of triple bond and adamantane ring on the vitamin D side chain produced partial agonists for vitamin D receptor.

Kudo T, Ishizawa M, Maekawa K, Nakabayashi M, Watarai Y, Uchida H, Tokiwa H, Ikura T, Ito N, Makishima M, Yamada S.

J Med Chem. 2014 May 22;57(10):4073-87. doi: 10.1021/jm401989c. Epub 2014 May 7.

PMID:
24773565
18.

A mixed population of antagonist and agonist binding conformers in a single crystal explains partial agonism against vitamin D receptor: active vitamin D analogues with 22R-alkyl group.

Anami Y, Itoh T, Egawa D, Yoshimoto N, Yamamoto K.

J Med Chem. 2014 May 22;57(10):4351-67. doi: 10.1021/jm500392t. Epub 2014 Apr 29.

PMID:
24742174
19.

Design and synthesis of tetraol derivatives of 1,12-dicarba-closo-dodecaborane as non-secosteroidal vitamin D analogs.

Fujii S, Kano A, Masuno H, Songkram C, Kawachi E, Hirano T, Tanatani A, Kagechika H.

Bioorg Med Chem Lett. 2014 Sep 15;24(18):4515-9. doi: 10.1016/j.bmcl.2014.07.075. Epub 2014 Aug 6.

PMID:
25149512
20.

Structural basis of the histidine-mediated vitamin D receptor agonistic and antagonistic mechanisms of (23S)-25-dehydro-1alpha-hydroxyvitamin D3-26,23-lactone.

Kakuda S, Ishizuka S, Eguchi H, Mizwicki MT, Norman AW, Takimoto-Kamimura M.

Acta Crystallogr D Biol Crystallogr. 2010 Aug;66(Pt 8):918-26. doi: 10.1107/S0907444910020810. Epub 2010 Jul 10.

PMID:
20693691
Format
Items per page
Sort by

Send to:

Choose Destination

Supplemental Content

Write to the Help Desk