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Results: 1 to 20 of 97

1.

[Design, synthesis and activity assessment of aryl-substituent benzyl acid targeting HIV gp41].

Wang H, Chen Z, Qiu J, Yu X, Xie Y, Liu S.

Nan Fang Yi Ke Da Xue Xue Bao. 2013 Feb;33(2):221-4. Chinese.

PMID:
23443776
[PubMed - indexed for MEDLINE]
Free Article
2.

Design, synthesis, and structure-activity relationship of a novel series of 2-aryl 5-(4-oxo-3-phenethyl-2-thioxothiazolidinylidenemethyl)furans as HIV-1 entry inhibitors.

Katritzky AR, Tala SR, Lu H, Vakulenko AV, Chen QY, Sivapackiam J, Pandya K, Jiang S, Debnath AK.

J Med Chem. 2009 Dec 10;52(23):7631-9. doi: 10.1021/jm900450n.

PMID:
19746983
[PubMed - indexed for MEDLINE]
Free PMC Article
3.

Design, synthesis, and biological activity of a novel series of 2,5-disubstituted furans/pyrroles as HIV-1 fusion inhibitors targeting gp41.

Jiang S, Tala SR, Lu H, Zou P, Avan I, Ibrahim TS, Abo-Dya NE, Abdelmajeid A, Debnath AK, Katritzky AR.

Bioorg Med Chem Lett. 2011 Nov 15;21(22):6895-8. doi: 10.1016/j.bmcl.2011.08.081. Epub 2011 Sep 5.

PMID:
21978673
[PubMed - indexed for MEDLINE]
4.

Tannin inhibits HIV-1 entry by targeting gp41.

Lü L, Liu SW, Jiang SB, Wu SG.

Acta Pharmacol Sin. 2004 Feb;25(2):213-8.

PMID:
14769212
[PubMed - indexed for MEDLINE]
Free Article
5.

Design, synthesis, and evaluation of indole compounds as novel inhibitors targeting Gp41.

Zhou G, Wu D, Hermel E, Balogh E, Gochin M.

Bioorg Med Chem Lett. 2010 Mar 1;20(5):1500-3. doi: 10.1016/j.bmcl.2010.01.111. Epub 2010 Jan 25.

PMID:
20153190
[PubMed - indexed for MEDLINE]
Free PMC Article
6.

Hydroxyl may not be indispensable for raltegravir: Design, synthesis and SAR Studies of raltegravir derivatives as HIV-1 inhibitors.

Wang Z, Wang M, Yao X, Li Y, Qiao W, Geng Y, Liu Y, Wang Q.

Eur J Med Chem. 2012 Apr;50:361-9. doi: 10.1016/j.ejmech.2012.02.015. Epub 2012 Feb 13.

PMID:
22369862
[PubMed - indexed for MEDLINE]
7.

Theaflavin derivatives in black tea and catechin derivatives in green tea inhibit HIV-1 entry by targeting gp41.

Liu S, Lu H, Zhao Q, He Y, Niu J, Debnath AK, Wu S, Jiang S.

Biochim Biophys Acta. 2005 May 25;1723(1-3):270-81. Epub 2005 Mar 24. Erratum in: Biochim Biophys Acta. 2007 Feb;1770(2):312.

PMID:
15823507
[PubMed - indexed for MEDLINE]
Free Article
8.

Synthesis and anti-HIV-1 activity of new MKC-442 analogues with an alkynyl-substituted 6-benzyl group.

Aly YL, Pedersen EB, La Colla P, Loddo R.

Arch Pharm (Weinheim). 2007 May;340(5):225-35.

PMID:
17464964
[PubMed - indexed for MEDLINE]
9.

Synthesis and antiviral activity of 4-benzyl pyridinone derivatives as potent and selective non-nucleoside human immunodeficiency virus type 1 reverse transcriptase inhibitors.

Dollé V, Nguyen CH, Legraverend M, Aubertin AM, Kirn A, Andreola ML, Ventura M, Tarrago-Litvak L, Bisagni E.

J Med Chem. 2000 Oct 19;43(21):3949-62.

PMID:
11052800
[PubMed - indexed for MEDLINE]
10.

Synthesis and anti-HIV activity evaluation of novel 2,4-disubstituted 7-methyl-1,1,3-trioxo-2,4-dihydro-pyrazolo-[4,5-e][1,2]thiadiazines.

Liu XY, Yan RZ, Wang Y, Zhan P, De Clercq E, Pannecouque C, Witvrouw M, Molina MT, Vega S.

Arch Pharm (Weinheim). 2008 Apr;341(4):216-22. doi: 10.1002/ardp.200700216.

PMID:
18266290
[PubMed - indexed for MEDLINE]
11.

Structure-activity relationships: analogues of the dicaffeoylquinic and dicaffeoyltartaric acids as potent inhibitors of human immunodeficiency virus type 1 integrase and replication.

King PJ, Ma G, Miao W, Jia Q, McDougall BR, Reinecke MG, Cornell C, Kuan J, Kim TR, Robinson WE Jr.

J Med Chem. 1999 Feb 11;42(3):497-509.

PMID:
9986720
[PubMed - indexed for MEDLINE]
12.

Anti-AIDS agents 90. novel C-28 modified bevirimat analogues as potent HIV maturation inhibitors.

Qian K, Bori ID, Chen CH, Huang L, Lee KH.

J Med Chem. 2012 Sep 27;55(18):8128-36. Epub 2012 Sep 14.

PMID:
22978745
[PubMed - indexed for MEDLINE]
Free PMC Article
13.

Synthesis of 2-(aminocarbonylmethylthio)-1H-imidazoles as novel Capravirine analogues.

Loksha YM, el-Barbary AA, el-Badawi MA, Nielsen C, Pedersen EB.

Bioorg Med Chem. 2005 Jul 1;13(13):4209-20.

PMID:
15896963
[PubMed - indexed for MEDLINE]
14.

Identification of inhibitors of the HIV-1 gp41 six-helix bundle formation from extracts of Chinese medicinal herbs Prunella vulgaris and Rhizoma cibotte.

Liu S, Jiang S, Wu Z, Lv L, Zhang J, Zhu Z, Wu S.

Life Sci. 2002 Aug 30;71(15):1779-91.

PMID:
12151056
[PubMed - indexed for MEDLINE]
15.

Computer-aided design, synthesis, and biological activity evaluation of potent fusion inhibitors targeting HIV-1 gp41.

Tan JJ, Zhang B, Cong XJ, Yang LF, Liu B, Kong R, Kui ZY, Wang CX, Hu LM.

Med Chem. 2011 Jul;7(4):309-16.

PMID:
21568877
[PubMed - indexed for MEDLINE]
16.

Anti-HIV-1 activity of anionic polymers: a comparative study of candidate microbicides.

Neurath AR, Strick N, Li YY.

BMC Infect Dis. 2002 Nov 21;2:27. Epub 2002 Nov 21.

PMID:
12445331
[PubMed - indexed for MEDLINE]
Free PMC Article
17.

[Isolation and characterization of the anti-HIV active component from Eucommia ulmoides].

Lv L, Sun YR, Xu W, Liu SW, Rao JJ, Wu SG.

Zhong Yao Cai. 2008 Jun;31(6):847-50. Chinese.

PMID:
18998566
[PubMed - indexed for MEDLINE]
18.

Design and properties of N(CCG)-gp41, a chimeric gp41 molecule with nanomolar HIV fusion inhibitory activity.

Louis JM, Bewley CA, Clore GM.

J Biol Chem. 2001 Aug 3;276(31):29485-9. Epub 2001 Jun 19.

PMID:
11418583
[PubMed - indexed for MEDLINE]
Free Article
19.

A natural theaflavins preparation inhibits HIV-1 infection by targeting the entry step: potential applications for preventing HIV-1 infection.

Yang J, Li L, Tan S, Jin H, Qiu J, Mao Q, Li R, Xia C, Jiang ZH, Jiang S, Liu S.

Fitoterapia. 2012 Mar;83(2):348-55. doi: 10.1016/j.fitote.2011.11.016. Epub 2011 Dec 3.

PMID:
22155187
[PubMed - indexed for MEDLINE]
20.

HIV-1 gp41 fusion intermediate: a target for HIV therapeutics.

Pan C, Liu S, Jiang S.

J Formos Med Assoc. 2010 Feb;109(2):94-105. doi: 10.1016/S0929-6646(10)60029-0. Review.

PMID:
20206833
[PubMed - indexed for MEDLINE]

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