Format
Items per page
Sort by

Send to:

Choose Destination

Links from PubMed

Items: 1 to 20 of 139

1.

Direct comparison of [(18) F]MH.MZ and [(18) F] altanserin for 5-HT2A receptor imaging with PET.

Hansen HD, Ettrup A, Herth MM, Dyssegaard A, Ratner C, Gillings N, Knudsen GM.

Synapse. 2013 Jun;67(6):328-37. doi: 10.1002/syn.21643. Epub 2013 Mar 7.

PMID:
23390031
2.

Binding characteristics of the 5-HT2A receptor antagonists altanserin and MDL 100907.

Kristiansen H, Elfving B, Plenge P, Pinborg LH, Gillings N, Knudsen GM.

Synapse. 2005 Dec 15;58(4):249-57.

PMID:
16206185
3.

18F-labeling and evaluation of novel MDL 100907 derivatives as potential 5-HT2A antagonists for molecular imaging.

Debus F, Herth MM, Piel M, Buchholz HG, Bausbacher N, Kramer V, Lüddens H, Rösch F.

Nucl Med Biol. 2010 May;37(4):487-95. doi: 10.1016/j.nucmedbio.2010.02.002. Epub 2010 Apr 8.

PMID:
20447561
4.

Preliminary in vivo and ex vivo evaluation of the 5-HT2A imaging probe [(18)F]MH.MZ.

Herth MM, Piel M, Debus F, Schmitt U, Lüddens H, Rösch F.

Nucl Med Biol. 2009 May;36(4):447-54. doi: 10.1016/j.nucmedbio.2009.01.012. Epub 2009 Mar 26.

PMID:
19423013
5.

P-glycoprotein influence on the brain uptake of a 5-HT(2A) ligand: [(18)F]MH.MZ.

Schmitt U, Lee DE, Herth MM, Piel M, Buchholz HG, Roesch F, Hiemke C, Lueddens H, Debus F.

Neuropsychobiology. 2011;63(3):183-90. doi: 10.1159/000321594. Epub 2011 Feb 8.

PMID:
21304228
6.

Characterization of radioactive metabolites of 5-HT2A receptor PET ligand [18F]altanserin in human and rodent.

Tan PZ, Baldwin RM, Van Dyck CH, Al-Tikriti M, Roth B, Khan N, Charney DS, Innis RB.

Nucl Med Biol. 1999 Aug;26(6):601-8.

PMID:
10587097
7.

Synthesis and in vitro affinities of various MDL 100907 derivatives as potential 18F-radioligands for 5-HT2A receptor imaging with PET.

Herth MM, Kramer V, Piel M, Palner M, Riss PJ, Knudsen GM, Rösch F.

Bioorg Med Chem. 2009 Apr 15;17(8):2989-3002. doi: 10.1016/j.bmc.2009.03.021. Epub 2009 Mar 14.

PMID:
19329329
8.

Analyses of [(18)F]altanserin bolus injection PET data. II: consideration of radiolabeled metabolites in humans.

Price JC, Lopresti BJ, Meltzer CC, Smith GS, Mason NS, Huang Y, Holt DP, Gunn RN, Mathis CA.

Synapse. 2001 Jul;41(1):11-21.

PMID:
11354009
9.

Analyses of [(18)F] altanserin bolus injection PET data. I: consideration of radiolabeled metabolites in baboons.

Price JC, Lopresti BJ, Mason NS, Holt DP, Huang Y, Mathis CA.

Synapse. 2001 Jul;41(1):1-10.

PMID:
11354008
10.

A PET [18F]altanserin study of 5-HT2A receptor binding in the human brain and responses to painful heat stimulation.

Kupers R, Frokjaer VG, Naert A, Christensen R, Budtz-Joergensen E, Kehlet H, Knudsen GM.

Neuroimage. 2009 Feb 1;44(3):1001-7. doi: 10.1016/j.neuroimage.2008.10.011. Epub 2008 Oct 28.

PMID:
19007894
11.

Suitability of [18F]altanserin and PET to determine 5-HT2A receptor availability in the rat brain: in vivo and in vitro validation of invasive and non-invasive kinetic models.

Kroll T, Elmenhorst D, Matusch A, Wedekind F, Weisshaupt A, Beer S, Bauer A.

Mol Imaging Biol. 2013 Aug;15(4):456-67. doi: 10.1007/s11307-013-0621-3. Epub 2013 Mar 1.

PMID:
23456885
12.

[¹⁸F]Altanserin and small animal PET: impact of multidrug efflux transporters on ligand brain uptake and subsequent quantification of 5-HT₂A receptor densities in the rat brain.

Kroll T, Elmenhorst D, Matusch A, Celik AA, Wedekind F, Weisshaupt A, Beer S, Bauer A.

Nucl Med Biol. 2014 Jan;41(1):1-9. doi: 10.1016/j.nucmedbio.2013.09.001. Epub 2013 Oct 9.

PMID:
24120220
13.

Extended characterisation of the serotonin 2A (5-HT2A) receptor-selective PET radiotracer 11C-MDL100907 in humans: quantitative analysis, test-retest reproducibility, and vulnerability to endogenous 5-HT tone.

Talbot PS, Slifstein M, Hwang DR, Huang Y, Scher E, Abi-Dargham A, Laruelle M.

Neuroimage. 2012 Jan 2;59(1):271-85. doi: 10.1016/j.neuroimage.2011.07.001. Epub 2011 Jul 18.

14.

Test-retest variability of serotonin 5-HT2A receptor binding measured with positron emission tomography and [18F]altanserin in the human brain.

Smith GS, Price JC, Lopresti BJ, Huang Y, Simpson N, Holt D, Mason NS, Meltzer CC, Sweet RA, Nichols T, Sashin D, Mathis CA.

Synapse. 1998 Dec;30(4):380-92.

PMID:
9826230
15.

Visualisation of loss of 5-HT2A receptors with age in healthy volunteers using [18F]altanserin and positron emission tomographic imaging.

Rosier A, Dupont P, Peuskens J, Bormans G, Vandenberghe R, Maes M, de Groot T, Schiepers C, Verbruggen A, Mortelmans L.

Psychiatry Res. 1996 Nov 25;68(1):11-22.

PMID:
9027929
16.

Reproducibility of 5-HT2A receptor measurements and sample size estimations with [18F]altanserin PET using a bolus/infusion approach.

Haugbøl S, Pinborg LH, Arfan HM, Frøkjaer VM, Madsen J, Dyrby TB, Svarer C, Knudsen GM.

Eur J Nucl Med Mol Imaging. 2007 Jun;34(6):910-5. Epub 2006 Dec 29.

PMID:
17195073
17.

Time-efficient and convenient synthesis of [(18)F]altanserin for human PET imaging by a new work-up procedure.

Massarweh G, Kovacevic M, Rosa-Neto P, Evans AC, Diksic M, Schirrmacher R.

Appl Radiat Isot. 2009 Nov;67(11):2040-3. doi: 10.1016/j.apradiso.2009.07.020. Epub 2009 Aug 4.

PMID:
19692252
18.

Equilibrium modeling of 5-HT(2A) receptors with [18F]deuteroaltanserin and PET: feasibility of a constant infusion paradigm.

van Dyck CH, Soares JC, Tan PZ, Staley JK, Baldwin RM, Amici LA, Fu X, Garg PK, Seibyl JP, Charney DS, Innis RB.

Nucl Med Biol. 2000 Nov;27(8):715-22.

PMID:
11150702
19.

Validation and quantification of [18F]altanserin binding in the rat brain using blood input and reference tissue modeling.

Riss PJ, Hong YT, Williamson D, Caprioli D, Sitnikov S, Ferrari V, Sawiak SJ, Baron JC, Dalley JW, Fryer TD, Aigbirhio FI.

J Cereb Blood Flow Metab. 2011 Dec;31(12):2334-42. doi: 10.1038/jcbfm.2011.94. Epub 2011 Jul 13.

20.

Characterization of [(11)C]Cimbi-36 as an agonist PET radioligand for the 5-HT(2A) and 5-HT(2C) receptors in the nonhuman primate brain.

Finnema SJ, Stepanov V, Ettrup A, Nakao R, Amini N, Svedberg M, Lehmann C, Hansen M, Knudsen GM, Halldin C.

Neuroimage. 2014 Jan 1;84:342-53. doi: 10.1016/j.neuroimage.2013.08.035. Epub 2013 Aug 28.

PMID:
23994452
Format
Items per page
Sort by

Send to:

Choose Destination

Supplemental Content

Write to the Help Desk