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Results: 1 to 20 of 135

1.

Design and synthesis of 2-aminothiazole based antimicrobials targeting MRSA.

Annadurai S, Martinez R, Canney DJ, Eidem T, Dunman PM, Abou-Gharbia M.

Bioorg Med Chem Lett. 2012 Dec 15;22(24):7719-25. doi: 10.1016/j.bmcl.2012.09.095. Epub 2012 Oct 3.

PMID:
23116888
[PubMed - indexed for MEDLINE]
2.

The chemical synthesis and antibiotic activity of a diverse library of 2-aminobenzimidazole small molecules against MRSA and multidrug-resistant A. baumannii.

Huigens RW 3rd, Reyes S, Reed CS, Bunders C, Rogers SA, Steinhauer AT, Melander C.

Bioorg Med Chem. 2010 Jan 15;18(2):663-74. doi: 10.1016/j.bmc.2009.12.003. Epub 2009 Dec 6.

PMID:
20044260
[PubMed - indexed for MEDLINE]
3.

Exploration of the activity of 7-pyrrolidino-8-methoxyisothiazoloquinolones against methicillin-resistant Staphylococcus aureus (MRSA).

Kim HY, Wiles JA, Wang Q, Pais GC, Lucien E, Hashimoto A, Nelson DM, Thanassi JA, Podos SD, Deshpande M, Pucci MJ, Bradbury BJ.

J Med Chem. 2011 May 12;54(9):3268-82. doi: 10.1021/jm101604v. Epub 2011 Apr 15.

PMID:
21425851
[PubMed - indexed for MEDLINE]
4.

Ureas of 5-aminopyrazole and 2-aminothiazole inhibit growth of gram-positive bacteria.

Kane JL Jr, Hirth BH, Liang B, Gourlie BB, Nahill S, Barsomian G.

Bioorg Med Chem Lett. 2003 Dec 15;13(24):4463-6.

PMID:
14643347
[PubMed - indexed for MEDLINE]
5.

The synthesis of phenylalanine-derived C5-substituted rhodanines and their activity against selected methicillin-resistant Staphylococcus aureus (MRSA) strains.

Hardej D, Ashby CR Jr, Khadtare NS, Kulkarni SS, Singh S, Talele TT.

Eur J Med Chem. 2010 Dec;45(12):5827-32. doi: 10.1016/j.ejmech.2010.09.045. Epub 2010 Sep 25.

PMID:
20947220
[PubMed - indexed for MEDLINE]
6.

Marinopyrrole derivatives as potential antibiotic agents against methicillin-resistant Staphylococcus aureus (II).

Cheng C, Liu Y, Song H, Pan L, Li J, Qin Y, Li R.

Mar Drugs. 2013 Aug 15;11(8):2927-48. doi: 10.3390/md11082927.

PMID:
23955285
[PubMed - indexed for MEDLINE]
Free PMC Article
7.

Evaluation of 4,5-disubstituted-2-aminoimidazole-triazole conjugates for antibiofilm/antibiotic resensitization activity against MRSA and Acinetobacter baumannii.

Su Z, Peng L, Worthington RJ, Melander C.

ChemMedChem. 2011 Dec 9;6(12):2243-51. doi: 10.1002/cmdc.201100316. Epub 2011 Sep 16.

PMID:
21928438
[PubMed - indexed for MEDLINE]
8.

Synthesis and evaluation of novel sulfenamides as novel anti Methicillin-resistant Staphylococcus aureus agents.

Shang JL, Guo H, Li ZS, Ren B, Li ZM, Dai HQ, Zhang LX, Wang JG.

Bioorg Med Chem Lett. 2013 Feb 1;23(3):724-7. doi: 10.1016/j.bmcl.2012.11.103. Epub 2012 Dec 3.

PMID:
23265879
[PubMed - indexed for MEDLINE]
9.

Riccardin C derivatives as anti-MRSA agents: structure-activity relationship of a series of hydroxylated bis(bibenzyl)s.

Sawada H, Okazaki M, Morita D, Kuroda T, Matsuno K, Hashimoto Y, Miyachi H.

Bioorg Med Chem Lett. 2012 Dec 15;22(24):7444-7. doi: 10.1016/j.bmcl.2012.10.052. Epub 2012 Oct 17.

PMID:
23122868
[PubMed - indexed for MEDLINE]
10.

Synthesis and biological evaluation of novel 1,3,5-triazine derivatives as antimicrobial agents.

Zhou C, Min J, Liu Z, Young A, Deshazer H, Gao T, Chang YT, Kallenbach NR.

Bioorg Med Chem Lett. 2008 Feb 15;18(4):1308-11. doi: 10.1016/j.bmcl.2008.01.031. Epub 2008 Jan 11.

PMID:
18226902
[PubMed - indexed for MEDLINE]
11.

Synthesis and biological evaluation of some thiazolylpyrazole derivatives as dual anti-inflammatory antimicrobial agents.

Bekhit AA, Fahmy HT, Rostom SA, El-Din A Bekhit A.

Eur J Med Chem. 2010 Dec;45(12):6027-38. doi: 10.1016/j.ejmech.2010.10.001. Epub 2010 Oct 20.

PMID:
20970223
[PubMed - indexed for MEDLINE]
12.

A multivalent approach to drug discovery for novel antibiotics.

Long DD, Aggen JB, Christensen BG, Judice JK, Hegde SS, Kaniga K, Krause KM, Linsell MS, Moran EJ, Pace JL.

J Antibiot (Tokyo). 2008 Oct;61(10):595-602. doi: 10.1038/ja.2008.79.

PMID:
19168973
[PubMed - indexed for MEDLINE]
13.

N-thiolated beta-lactams: novel antibacterial agents for methicillin-resistant Staphylococcus aureus.

Turos E, Long TE, Konaklieva MI, Coates C, Shim JY, Dickey S, Lim DV, Cannons A.

Bioorg Med Chem Lett. 2002 Aug 19;12(16):2229-31.

PMID:
12127544
[PubMed - indexed for MEDLINE]
14.

High-throughput identification of antibacterials against methicillin-resistant Staphylococcus aureus (MRSA) and the transglycosylase.

Cheng TJ, Wu YT, Yang ST, Lo KH, Chen SK, Chen YH, Huang WI, Yuan CH, Guo CW, Huang LY, Chen KT, Shih HW, Cheng YS, Cheng WC, Wong CH.

Bioorg Med Chem. 2010 Dec 15;18(24):8512-29. doi: 10.1016/j.bmc.2010.10.036. Epub 2010 Oct 21.

PMID:
21075637
[PubMed - indexed for MEDLINE]
15.

Synthesis and potent antimicrobial activity of some novel 4-(5, 6-dichloro-1H-benzimidazol-2-yl)-N-substituted benzamides.

Ozden S, Karataş H, Yildiz S, Göker H.

Arch Pharm (Weinheim). 2004 Oct;337(10):556-62.

PMID:
15476288
[PubMed - indexed for MEDLINE]
16.

Development of novel antibacterial agents against methicillin-resistant Staphylococcus aureus.

Chiu HC, Lee SL, Kapuriya N, Wang D, Chen YR, Yu SL, Kulp SK, Teng LJ, Chen CS.

Bioorg Med Chem. 2012 Aug 1;20(15):4653-60. doi: 10.1016/j.bmc.2012.06.018. Epub 2012 Jun 15.

PMID:
22750009
[PubMed - indexed for MEDLINE]
Free PMC Article
17.

Design, synthesis and antibacterial activity studies of thiazole derivatives as potent ecKAS III inhibitors.

Cheng K, Xue JY, Zhu HL.

Bioorg Med Chem Lett. 2013 Jul 15;23(14):4235-8. doi: 10.1016/j.bmcl.2013.05.006. Epub 2013 May 10.

PMID:
23731945
[PubMed - indexed for MEDLINE]
18.

The synthesis and SAR study of phenylalanine-derived (Z)-5-arylmethylidene rhodanines as anti-methicillin-resistant Staphylococcus aureus (MRSA) compounds.

Patel BA, Ashby CR Jr, Hardej D, Talele TT.

Bioorg Med Chem Lett. 2013 Oct 15;23(20):5523-7. doi: 10.1016/j.bmcl.2013.08.059. Epub 2013 Aug 20.

PMID:
24012180
[PubMed - indexed for MEDLINE]
19.

Restoring methicillin-resistant Staphylococcus aureus susceptibility to β-lactam antibiotics.

Tan CM, Therien AG, Lu J, Lee SH, Caron A, Gill CJ, Lebeau-Jacob C, Benton-Perdomo L, Monteiro JM, Pereira PM, Elsen NL, Wu J, Deschamps K, Petcu M, Wong S, Daigneault E, Kramer S, Liang L, Maxwell E, Claveau D, Vaillancourt J, Skorey K, Tam J, Wang H, Meredith TC, Sillaots S, Wang-Jarantow L, Ramtohul Y, Langlois E, Landry F, Reid JC, Parthasarathy G, Sharma S, Baryshnikova A, Lumb KJ, Pinho MG, Soisson SM, Roemer T.

Sci Transl Med. 2012 Mar 21;4(126):126ra35. doi: 10.1126/scitranslmed.3003592.

PMID:
22440737
[PubMed - indexed for MEDLINE]
Free Article
20.

Design, synthesis, and structure-activity relationship studies of conformationally restricted mutilin 14-carbamates.

Fu L, Liu X, Ling C, Cheng J, Guo X, He H, Ding S, Yang Y.

Bioorg Med Chem Lett. 2012 Jan 15;22(2):814-9. doi: 10.1016/j.bmcl.2011.12.063. Epub 2011 Dec 20.

PMID:
22209487
[PubMed - indexed for MEDLINE]

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