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Results: 1 to 20 of 97

1.

Synthesis and evaluation of hybrid drugs for a potential HIV/AIDS-malaria combination therapy.

Aminake MN, Mahajan A, Kumar V, Hans R, Wiesner L, Taylor D, de Kock C, Grobler A, Smith PJ, Kirschner M, Rethwilm A, Pradel G, Chibale K.

Bioorg Med Chem. 2012 Sep 1;20(17):5277-89. doi: 10.1016/j.bmc.2012.06.038. Epub 2012 Jun 29.

PMID:
22858300
[PubMed - indexed for MEDLINE]
2.

New chimeric antimalarials with 4-aminoquinoline moiety linked to a tetraoxane skeleton.

Opsenica I, Opsenica D, Lanteri CA, Anova L, Milhous WK, Smith KS, Solaja BA.

J Med Chem. 2008 Oct 9;51(19):6216-9. doi: 10.1021/jm8006905. Epub 2008 Sep 6.

PMID:
18774792
[PubMed - indexed for MEDLINE]
3.

Synthesis and evaluation of sulfonylurea derivatives as novel antimalarials.

León C, Rodrigues J, Gamboa de Domínguez N, Charris J, Gut J, Rosenthal PJ, Domínguez JN.

Eur J Med Chem. 2007 Jun;42(6):735-42. Epub 2007 Jan 14.

PMID:
17321641
[PubMed - indexed for MEDLINE]
4.

4-anilinoquinoline triazines: a novel class of hybrid antimalarial agents.

Kumar A, Srivastava K, Kumar SR, Siddiqi MI, Puri SK, Sexana JK, Chauhan PM.

Eur J Med Chem. 2011 Feb;46(2):676-90. doi: 10.1016/j.ejmech.2010.12.003. Epub 2010 Dec 9.

PMID:
21194812
[PubMed - indexed for MEDLINE]
5.

Antimalarial and antiplasmodial activities of norneolignans. Syntheses and SAR.

Skytte DM, Nielsen SF, Chen M, Zhai L, Olsen CE, Christensen SB.

J Med Chem. 2006 Jan 12;49(1):436-40.

PMID:
16392829
[PubMed - indexed for MEDLINE]
6.

Antimalarial dual drugs based on potent inhibitors of glutathione reductase from Plasmodium falciparum.

Friebolin W, Jannack B, Wenzel N, Furrer J, Oeser T, Sanchez CP, Lanzer M, Yardley V, Becker K, Davioud-Charvet E.

J Med Chem. 2008 Mar 13;51(5):1260-77. doi: 10.1021/jm7009292. Epub 2008 Feb 9.

PMID:
18260613
[PubMed - indexed for MEDLINE]
7.

Antiparasitic activities of two sesquiterpenic lactones isolated from Acanthospermum hispidum D.C.

Ganfon H, Bero J, Tchinda AT, Gbaguidi F, Gbenou J, Moudachirou M, Frédérich M, Quetin-Leclercq J.

J Ethnopharmacol. 2012 May 7;141(1):411-7. doi: 10.1016/j.jep.2012.03.002. Epub 2012 Mar 13.

PMID:
22440261
[PubMed - indexed for MEDLINE]
8.

Anti-HIV and antiplasmodial activity of original flavonoid derivatives.

Casano G, Dumètre A, Pannecouque C, Hutter S, Azas N, Robin M.

Bioorg Med Chem. 2010 Aug 15;18(16):6012-23. doi: 10.1016/j.bmc.2010.06.067. Epub 2010 Jun 25.

PMID:
20638854
[PubMed - indexed for MEDLINE]
9.

Synergy of the antiretroviral protease inhibitor indinavir and chloroquine against malaria parasites in vitro and in vivo.

Li X, He Z, Chen L, Li Y, Li Q, Zhao S, Tao Z, Hu W, Qin L, Chen X.

Parasitol Res. 2011 Dec;109(6):1519-24. doi: 10.1007/s00436-011-2427-z. Epub 2011 May 3.

PMID:
21537980
[PubMed - indexed for MEDLINE]
10.

Squaric acid/4-aminoquinoline conjugates: novel potent antiplasmodial agents.

Ribeiro CJ, Kumar SP, Gut J, Gonçalves LM, Rosenthal PJ, Moreira R, Santos MM.

Eur J Med Chem. 2013 Nov;69:365-72. doi: 10.1016/j.ejmech.2013.08.037. Epub 2013 Sep 13.

PMID:
24077527
[PubMed - indexed for MEDLINE]
11.

Traditional herbal antimalarial therapy in Kilifi district, Kenya.

Gathirwa JW, Rukunga GM, Mwitari PG, Mwikwabe NM, Kimani CW, Muthaura CN, Kiboi DM, Nyangacha RM, Omar SA.

J Ethnopharmacol. 2011 Mar 24;134(2):434-42. doi: 10.1016/j.jep.2010.12.043. Epub 2011 Jan 4.

PMID:
21211554
[PubMed - indexed for MEDLINE]
12.

Novel orally active antimalarial thiazoles.

González Cabrera D, Douelle F, Feng TS, Nchinda AT, Younis Y, White KL, Wu Q, Ryan E, Burrows JN, Waterson D, Witty MJ, Wittlin S, Charman SA, Chibale K.

J Med Chem. 2011 Nov 10;54(21):7713-9. doi: 10.1021/jm201108k. Epub 2011 Oct 11.

PMID:
21966980
[PubMed - indexed for MEDLINE]
13.

Short synthesis and antimalarial activity of fagaronine.

Rivaud M, Mendoza A, Sauvain M, Valentin A, Jullian V.

Bioorg Med Chem. 2012 Aug 1;20(15):4856-61. doi: 10.1016/j.bmc.2012.05.061. Epub 2012 Jun 5.

PMID:
22766218
[PubMed - indexed for MEDLINE]
14.

In vitro and in vivo antimalarial activity of derivatives of 1,10-phenanthroline framework.

Yapi AD, Valentin A, Chezal JM, Chavignon O, Chaillot B, Gerhardt R, Teulade JC, Blache Y.

Arch Pharm (Weinheim). 2006 Apr;339(4):201-6.

PMID:
16586427
[PubMed - indexed for MEDLINE]
15.

Antimalarial activity of betulinic acid and derivatives in vitro against Plasmodium falciparum and in vivo in P. berghei-infected mice.

de Sá MS, Costa JF, Krettli AU, Zalis MG, Maia GL, Sette IM, Câmara Cde A, Filho JM, Giulietti-Harley AM, Ribeiro Dos Santos R, Soares MB.

Parasitol Res. 2009 Jul;105(1):275-9. doi: 10.1007/s00436-009-1394-0. Epub 2009 Apr 15.

PMID:
19367418
[PubMed - indexed for MEDLINE]
16.

Ketotifen is an antimalarial prodrug of norketotifen with blood schizonticidal and liver-stage efficacy.

Milner E, Sousa J, Pybus B, Auschwitz J, Caridha D, Gardner S, Grauer K, Harris E, Hickman M, Kozar MP, Lee P, Leed S, Li Q, Melendez V, Moon J, Ngundam F, O'Neil M, Parriott S, Potter B, Sciotti R, Tangteung A, Dow GS.

Eur J Drug Metab Pharmacokinet. 2012 Mar;37(1):17-22.

PMID:
22314893
[PubMed - indexed for MEDLINE]
17.

Synthesis and structure-activity relationships of 4-pyridones as potential antimalarials.

Yeates CL, Batchelor JF, Capon EC, Cheesman NJ, Fry M, Hudson AT, Pudney M, Trimming H, Woolven J, Bueno JM, Chicharro J, Fernández E, Fiandor JM, Gargallo-Viola D, Gómez de las Heras F, Herreros E, León ML.

J Med Chem. 2008 May 8;51(9):2845-52. doi: 10.1021/jm0705760. Epub 2008 Apr 9.

PMID:
18396855
[PubMed - indexed for MEDLINE]
18.

Antimalarial activity of endoperoxide compound 6-(1,2,6,7-tetraoxaspiro[7.11]nonadec-4-yl)hexan-1-ol.

Sato A, Hiramoto A, Morita M, Matsumoto M, Komich Y, Nakase Y, Tanigawa N, Hiraoka O, Hiramoto K, Hayatsu H, Higaki K, Kawai S, Masuyama A, Nojima M, Wataya Y, Kim HS.

Parasitol Int. 2011 Sep;60(3):270-3. doi: 10.1016/j.parint.2011.04.001. Epub 2011 Apr 8.

PMID:
21501696
[PubMed - indexed for MEDLINE]
19.

Synthesis and antiplasmodial activity of new indolone N-oxide derivatives.

Nepveu F, Kim S, Boyer J, Chatriant O, Ibrahim H, Reybier K, Monje MC, Chevalley S, Perio P, Lajoie BH, Bouajila J, Deharo E, Sauvain M, Tahar R, Basco L, Pantaleo A, Turini F, Arese P, Valentin A, Thompson E, Vivas L, Petit S, Nallet JP.

J Med Chem. 2010 Jan 28;53(2):699-714. doi: 10.1021/jm901300d.

PMID:
20014857
[PubMed - indexed for MEDLINE]
20.

In vitro and in vivo properties of ellagic acid in malaria treatment.

Soh PN, Witkowski B, Olagnier D, Nicolau ML, Garcia-Alvarez MC, Berry A, Benoit-Vical F.

Antimicrob Agents Chemother. 2009 Mar;53(3):1100-6. doi: 10.1128/AAC.01175-08. Epub 2008 Nov 17.

PMID:
19015354
[PubMed - indexed for MEDLINE]
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