Display Settings:

Format
Items per page
Sort by

Send to:

Choose Destination

Results: 1 to 20 of 98

1.

Shape-based reprofiling of FDA-approved drugs for the H₁ histamine receptor.

Vasudevan SR, Moore JB, Schymura Y, Churchill GC.

J Med Chem. 2012 Aug 23;55(16):7054-60. doi: 10.1021/jm300671m. Epub 2012 Aug 6.

PMID:
22793499
[PubMed - indexed for MEDLINE]
2.

In vivo and in vitro interaction of the novel selective histamine H1 receptor antagonist mizolastine with H1 receptors in the rodent.

Benavides J, Schoemaker H, Dana C, Claustre Y, Delahaye M, Prouteau M, Manoury P, Allen J, Scatton B, Langer SZ, et al.

Arzneimittelforschung. 1995 May;45(5):551-8.

PMID:
7612054
[PubMed - indexed for MEDLINE]
3.

Effects of antidepressant drugs on histamine-H1 receptors in the brain.

Hall H, Ogren SO.

Life Sci. 1984 Feb 6;34(6):597-605.

PMID:
6141518
[PubMed - indexed for MEDLINE]
4.

The suppression of olfactory bulbectomy-induced muricide by antidepressants and antihistamines via histamine H1 receptor blocking.

Noguchi S, Inukai T, Kuno T, Tanaka C.

Physiol Behav. 1992 Jun;51(6):1123-7.

PMID:
1353628
[PubMed - indexed for MEDLINE]
5.

Analytical method for simultaneously measuring ex vivo drug receptor occupancy and dissociation rate: application to (R)-dimethindene occupancy of central histamine H1 receptors.

Malany S, Hernandez LM, Smith WF, Crowe PD, Hoare SR.

J Recept Signal Transduct Res. 2009;29(2):84-93. doi: 10.1080/10799890902721339.

PMID:
19308787
[PubMed - indexed for MEDLINE]
6.

Intact cell binding for in vitro prediction of sedative and non-sedative histamine H1-receptor antagonists based on receptor internalization.

Hishinuma S, Sato Y, Kobayashi Y, Komazaki H, Saito M.

J Pharmacol Sci. 2008 May;107(1):66-79. Epub 2008 Apr 29.

PMID:
18446005
[PubMed - indexed for MEDLINE]
Free Article
7.

Muscarinic cholinergic and histamine H1 receptor binding of phenothiazine drug metabolites.

Hals PA, Hall H, Dahl SG.

Life Sci. 1988;43(5):405-12.

PMID:
2899826
[PubMed - indexed for MEDLINE]
8.

Constitutive activity of the histamine H(1) receptor reveals inverse agonism of histamine H(1) receptor antagonists.

Bakker RA, Wieland K, Timmerman H, Leurs R.

Eur J Pharmacol. 2000 Jan 3;387(1):R5-7.

PMID:
10633171
[PubMed - indexed for MEDLINE]
9.

[Substituted 2,3,4,5-tetrahydro-1H-gamma-carbolines: new antagonists of histamine H1 receptors].

Ivashchenko AV, Mit'kin OD, Okun' IM, Salimov RM, Fedotov IuA.

Eksp Klin Farmakol. 2010 Nov;73(11):25-9. Russian.

PMID:
21254595
[PubMed - indexed for MEDLINE]
10.

Emedastine: a potent, high affinity histamine H1-receptor-selective antagonist for ocular use: receptor binding and second messenger studies.

Sharif NA, Su SX, Yanni JM.

J Ocul Pharmacol. 1994 Winter;10(4):653-64.

PMID:
7714409
[PubMed - indexed for MEDLINE]
11.
12.

Studies on the novel antiallergic agent HSR-609: its penetration into the central nervous system in mice and guinea pigs and its selectivity for the histamine H1-receptor.

Kakiuchi M, Ohashi T, Musoh K, Kawamura K, Morikawa K, Kato H.

Jpn J Pharmacol. 1997 Apr;73(4):291-8.

PMID:
9165365
[PubMed - indexed for MEDLINE]
Free Article
13.

Unique binding pocket for KW-4679 in the histamine H1 receptor.

Nonaka H, Otaki S, Ohshima E, Kono M, Kase H, Ohta K, Fukui H, Ichimura M.

Eur J Pharmacol. 1998 Mar 12;345(1):111-7.

PMID:
9593602
[PubMed - indexed for MEDLINE]
14.

Stereochemical diversity-oriented conformational restriction strategy. Development of potent histamine H3 and/or H4 receptor antagonists with an imidazolylcyclopropane structure.

Watanabe M, Kazuta Y, Hayashi H, Yamada S, Matsuda A, Shuto S.

J Med Chem. 2006 Sep 7;49(18):5587-96.

PMID:
16942032
[PubMed - indexed for MEDLINE]
15.

Synthesis and structure-activity relationship of tricyclic carboxylic acids as novel anti-histamines.

Kubota K, Kurebayashi H, Miyachi H, Tobe M, Onishi M, Isobe Y.

Bioorg Med Chem. 2011 May 1;19(9):3005-21. doi: 10.1016/j.bmc.2011.03.003. Epub 2011 Mar 11.

PMID:
21470866
[PubMed - indexed for MEDLINE]
16.

Food-deprived activity stress decreased the activity of the histaminergic neuron system in rats.

Endou M, Yanai K, Sakurai E, Fukudo S, Hongo M, Watanabe T.

Brain Res. 2001 Feb 9;891(1-2):32-41.

PMID:
11164807
[PubMed - indexed for MEDLINE]
17.

Synthesis and pharmacological identification of neutral histamine H1-receptor antagonists.

Govoni M, Bakker RA, van de Wetering I, Smit MJ, Menge WM, Timmerman H, Elz S, Schunack W, Leurs R.

J Med Chem. 2003 Dec 18;46(26):5812-24.

PMID:
14667234
[PubMed - indexed for MEDLINE]
18.

Crystal structure-based virtual screening for fragment-like ligands of the human histamine H(1) receptor.

de Graaf C, Kooistra AJ, Vischer HF, Katritch V, Kuijer M, Shiroishi M, Iwata S, Shimamura T, Stevens RC, de Esch IJ, Leurs R.

J Med Chem. 2011 Dec 8;54(23):8195-206. doi: 10.1021/jm2011589. Epub 2011 Nov 7.

PMID:
22007643
[PubMed - indexed for MEDLINE]
Free PMC Article
19.

Preclinical pharmacology of bilastine, a new selective histamine H1 receptor antagonist: receptor selectivity and in vitro antihistaminic activity.

Corcóstegui R, Labeaga L, Innerárity A, Berisa A, Orjales A.

Drugs R D. 2005;6(6):371-84.

PMID:
16274260
[PubMed - indexed for MEDLINE]
20.

Identification of a dual histamine H1/H3 receptor ligand based on the H1 antagonist chlorpheniramine.

Aslanian R, Mutahi Mw, Shih NY, Piwinski JJ, West R, Williams SM, She S, Wu RL, Hey JA.

Bioorg Med Chem Lett. 2003 Jun 16;13(12):1959-61.

PMID:
12781173
[PubMed - indexed for MEDLINE]

Display Settings:

Format
Items per page
Sort by

Send to:

Choose Destination

Supplemental Content

Write to the Help Desk