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Similar articles for PubMed (Select 21741131)

1.

Targeting the human malaria parasite Plasmodium falciparum: in vitro identification of a new antiplasmodial hit in 4-phenoxy-2-trichloromethylquinazoline series.

Castera-Ducros C, Azas N, Verhaeghe P, Hutter S, Garrigue P, Dumètre A, Mbatchi L, Laget M, Remusat V, Sifredi F, Rault S, Rathelot P, Vanelle P.

Eur J Med Chem. 2011 Sep;46(9):4184-91. doi: 10.1016/j.ejmech.2011.06.021. Epub 2011 Jun 23.

PMID:
21741131
2.

4-Thiophenoxy-2-trichloromethyquinazolines display in vitro selective antiplasmodial activity against the human malaria parasite Plasmodium falciparum.

Verhaeghe P, Dumètre A, Castera-Ducros C, Hutter S, Laget M, Fersing C, Prieri M, Yzombard J, Sifredi F, Rault S, Rathelot P, Vanelle P, Azas N.

Bioorg Med Chem Lett. 2011 Oct 1;21(19):6003-6. doi: 10.1016/j.bmcl.2011.06.113. Epub 2011 Jul 2.

PMID:
21852132
3.

Synthesis and in vitro antiplasmodial evaluation of 4-anilino-2-trichloromethylquinazolines.

Verhaeghe P, Azas N, Hutter S, Castera-Ducros C, Laget M, Dumètre A, Gasquet M, Reboul JP, Rault S, Rathelot P, Vanelle P.

Bioorg Med Chem. 2009 Jul 1;17(13):4313-22. doi: 10.1016/j.bmc.2009.05.022. Epub 2009 May 15.

PMID:
19482476
4.

A new synthetic route to original sulfonamide derivatives in 2-trichloromethylquinazoline series: a structure-activity relationship study of antiplasmodial activity.

Primas N, Verhaeghe P, Cohen A, Kieffer C, Dumètre A, Hutter S, Rault S, Rathelot P, Azas N, Vanelle P.

Molecules. 2012 Jul 5;17(7):8105-17. doi: 10.3390/molecules17078105.

5.

Synthesis and antiplasmodial activity of new 4-aryl-2-trichloromethylquinazolines.

Verhaeghe P, Azas N, Gasquet M, Hutter S, Ducros C, Laget M, Rault S, Rathelot P, Vanelle P.

Bioorg Med Chem Lett. 2008 Jan 1;18(1):396-401. Epub 2007 Oct 17.

PMID:
17981462
6.

Original quinazoline derivatives displaying antiplasmodial properties.

Kabri Y, Azas N, Dumètre A, Hutter S, Laget M, Verhaeghe P, Gellis A, Vanelle P.

Eur J Med Chem. 2010 Feb;45(2):616-22. doi: 10.1016/j.ejmech.2009.11.005. Epub 2009 Nov 6.

PMID:
19926173
7.

Synthesis and in vitro evaluation of 4-trichloromethylpyrrolo[1,2-a]quinoxalines as new antiplasmodial agents.

Primas N, Suzanne P, Verhaeghe P, Hutter S, Kieffer C, Laget M, Cohen A, Broggi J, Lancelot JC, Lesnard A, Dallemagne P, Rathelot P, Rault S, Vanelle P, Azas N.

Eur J Med Chem. 2014 Aug 18;83:26-35. doi: 10.1016/j.ejmech.2014.06.014. Epub 2014 Jun 10.

PMID:
24946216
8.
9.

Dibenzylideneacetone analogues as novel Plasmodium falciparum inhibitors.

Aher RB, Wanare G, Kawathekar N, Kumar RR, Kaushik NK, Sahal D, Chauhan VS.

Bioorg Med Chem Lett. 2011 May 15;21(10):3034-6. doi: 10.1016/j.bmcl.2011.03.037. Epub 2011 Apr 12.

PMID:
21493068
10.

Cryptolepine analogues containing basic aminoalkyl side-chains at C-11: synthesis, antiplasmodial activity, and cytotoxicity.

Lavrado J, Paulo A, Gut J, Rosenthal PJ, Moreira R.

Bioorg Med Chem Lett. 2008 Feb 15;18(4):1378-81. doi: 10.1016/j.bmcl.2008.01.015. Epub 2008 Jan 9.

PMID:
18207399
11.

Preparation and antiprotozoal evaluation of promising β-carboline alkaloids.

Gellis A, Dumètre A, Lanzada G, Hutter S, Ollivier E, Vanelle P, Azas N.

Biomed Pharmacother. 2012 Jul;66(5):339-47. doi: 10.1016/j.biopha.2011.12.006. Epub 2012 Feb 17.

PMID:
22397756
12.

Search for new pharmacophores for antimalarial activity. Part II: synthesis and antimalarial activity of new 6-ureido-4-anilinoquinazolines.

Madapa S, Tusi Z, Mishra A, Srivastava K, Pandey SK, Tripathi R, Puri SK, Batra S.

Bioorg Med Chem. 2009 Jan 1;17(1):222-34. doi: 10.1016/j.bmc.2008.11.005. Epub 2008 Nov 8.

PMID:
19041250
13.

Synthesis and evaluation of febrifugine analogues as potential antimalarial agents.

Zhu S, Meng L, Zhang Q, Wei L.

Bioorg Med Chem Lett. 2006 Apr 1;16(7):1854-8. Epub 2006 Jan 24.

14.

Antimalarial acridines: synthesis, in vitro activity against P. falciparum and interaction with hematin.

Guetzoyan L, Yu XM, Ramiandrasoa F, Pethe S, Rogier C, Pradines B, Cresteil T, Perrée-Fauvet M, Mahy JP.

Bioorg Med Chem. 2009 Dec 1;17(23):8032-9. doi: 10.1016/j.bmc.2009.10.005. Epub 2009 Oct 9.

PMID:
19879150
15.

Synthesis, structural characterization and biological evaluation of novel stilbene derivatives as potential antimalarial agents.

Jung M, Park WH, Jung JC, Lim E, Lee Y, Oh S, Moon HI.

Chem Biol Drug Des. 2009 Mar;73(3):346-54. doi: 10.1111/j.1747-0285.2009.00775.x.

PMID:
19207471
16.

Evaluation of substituted phenalenone analogues as antiplasmodial agents.

Gutiérrez D, Flores N, Abad-Grillo T, McNaughton-Smith G.

Exp Parasitol. 2013 Oct;135(2):456-8. doi: 10.1016/j.exppara.2013.08.008. Epub 2013 Aug 25.

PMID:
23985373
17.

Synthesis of novel substituted 1,3-diaryl propenone derivatives and their antimalarial activity in vitro.

Mishra N, Arora P, Kumar B, Mishra LC, Bhattacharya A, Awasthi SK, Bhasin VK.

Eur J Med Chem. 2008 Jul;43(7):1530-5. Epub 2007 Sep 29.

PMID:
17977622
18.

Synthesis, cytotoxicity, and antiplasmodial and antitrypanosomal activity of new neocryptolepine derivatives.

Jonckers TH, van Miert S, Cimanga K, Bailly C, Colson P, De Pauw-Gillet MC, van den Heuvel H, Claeys M, Lemière F, Esmans EL, Rozenski J, Quirijnen L, Maes L, Dommisse R, Lemière GL, Vlietinck A, Pieters L.

J Med Chem. 2002 Aug 1;45(16):3497-508.

PMID:
12139461
19.

Modifications of the chemical structure of terpenes in antiplasmodial and antifungal drug research.

Olagnier D, Costes P, Berry A, Linas MD, Urrutigoity M, Dechy-Cabaret O, Benoit-Vical F.

Bioorg Med Chem Lett. 2007 Nov 15;17(22):6075-8. Epub 2007 Sep 18.

PMID:
17904365
20.

Karavilagenin C derivatives as antimalarials.

Ramalhete C, Lopes D, Molnár J, Mulhovo S, Rosário VE, Ferreira MJ.

Bioorg Med Chem. 2011 Jan 1;19(1):330-8. doi: 10.1016/j.bmc.2010.11.015. Epub 2010 Nov 11.

PMID:
21129980
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