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Results: 1 to 20 of 211

1.

Design, synthesis, and biological evaluation of new cinnamic derivatives as antituberculosis agents.

De P, Koumba Yoya G, Constant P, Bedos-Belval F, Duran H, Saffon N, Daffé M, Baltas M.

J Med Chem. 2011 Mar 10;54(5):1449-61. doi: 10.1021/jm101510d. Epub 2011 Feb 10.

PMID:
21309577
[PubMed - indexed for MEDLINE]
2.

Synthesis, biological evaluation, and structure-activity relationships for 5-[(E)-2-arylethenyl]-3-isoxazolecarboxylic acid alkyl ester derivatives as valuable antitubercular chemotypes.

Pieroni M, Lilienkampf A, Wan B, Wang Y, Franzblau SG, Kozikowski AP.

J Med Chem. 2009 Oct 22;52(20):6287-96. doi: 10.1021/jm900513a.

PMID:
19757815
[PubMed - indexed for MEDLINE]
3.

Synthesis and antimycobacterial evaluation of new trans-cinnamic acid hydrazide derivatives.

Carvalho SA, da Silva EF, de Souza MV, Lourenço MC, Vicente FR.

Bioorg Med Chem Lett. 2008 Jan 15;18(2):538-41. Epub 2007 Nov 28.

PMID:
18068364
[PubMed - indexed for MEDLINE]
4.

Synthesis and evaluation of a novel series of pseudo-cinnamic derivatives as antituberculosis agents.

Yoya GK, Bedos-Belval F, Constant P, Duran H, Daffé M, Baltas M.

Bioorg Med Chem Lett. 2009 Jan 15;19(2):341-3. doi: 10.1016/j.bmcl.2008.11.082. Epub 2008 Nov 27.

PMID:
19084396
[PubMed - indexed for MEDLINE]
5.

Structure-activity relationships for a series of quinoline-based compounds active against replicating and nonreplicating Mycobacterium tuberculosis.

Lilienkampf A, Mao J, Wan B, Wang Y, Franzblau SG, Kozikowski AP.

J Med Chem. 2009 Apr 9;52(7):2109-18. doi: 10.1021/jm900003c.

PMID:
19271749
[PubMed - indexed for MEDLINE]
6.

Synthesis, antitubercular activity, and SAR study of N-substituted-phenylamino-5-methyl-1H-1,2,3-triazole-4-carbohydrazides.

Jordão AK, Sathler PC, Ferreira VF, Campos VR, de Souza MC, Castro HC, Lannes A, Lourenco A, Rodrigues CR, Bello ML, Lourenco MC, Carvalho GS, Almeida MC, Cunha AC.

Bioorg Med Chem. 2011 Sep 15;19(18):5605-11. doi: 10.1016/j.bmc.2011.07.035. Epub 2011 Jul 24.

PMID:
21840219
[PubMed - indexed for MEDLINE]
Free Article
7.

Design, synthesis and antimycobacterial evaluation of novel 3-substituted-N-aryl-6,7-dimethoxy-3a,4-dihydro-3H-indeno[1,2-c]pyrazole-2-carboxamide analogues.

Ahsan MJ, Samy JG, Dutt KR, Agrawal UK, Yadav BS, Vyas S, Kaur R, Yadav G.

Bioorg Med Chem Lett. 2011 Aug 1;21(15):4451-3. doi: 10.1016/j.bmcl.2011.06.018. Epub 2011 Jun 17.

PMID:
21733688
[PubMed - indexed for MEDLINE]
8.

Clubbed triazoles: a novel approach to antitubercular drugs.

Shiradkar M, Suresh Kumar GV, Dasari V, Tatikonda S, Akula KC, Shah R.

Eur J Med Chem. 2007 Jun;42(6):807-16. Epub 2006 Dec 15.

PMID:
17239490
[PubMed - indexed for MEDLINE]
9.

[Development of antituberculous drugs: current status and future prospects].

Tomioka H, Namba K.

Kekkaku. 2006 Dec;81(12):753-74. Review. Japanese.

PMID:
17240921
[PubMed - indexed for MEDLINE]
10.

Novel molecular hybrids of cinnamic acids and guanylhydrazones as potential antitubercular agents.

Bairwa R, Kakwani M, Tawari NR, Lalchandani J, Ray MK, Rajan MG, Degani MS.

Bioorg Med Chem Lett. 2010 Mar 1;20(5):1623-5. doi: 10.1016/j.bmcl.2010.01.031. Epub 2010 Jan 20.

PMID:
20138519
[PubMed - indexed for MEDLINE]
11.

Schiff bases of indoline-2,3-dione (isatin) derivatives and nalidixic acid carbohydrazide, synthesis, antitubercular activity and pharmacophoric model building.

Aboul-Fadl T, Bin-Jubair FA, Aboul-Wafa O.

Eur J Med Chem. 2010 Oct;45(10):4578-86. doi: 10.1016/j.ejmech.2010.07.020. Epub 2010 Aug 8.

PMID:
20696500
[PubMed - indexed for MEDLINE]
12.

Rational design of 5-phenyl-3-isoxazolecarboxylic acid ethyl esters as growth inhibitors of Mycobacterium tuberculosis. a potent and selective series for further drug development.

Lilienkampf A, Pieroni M, Wan B, Wang Y, Franzblau SG, Kozikowski AP.

J Med Chem. 2010 Jan 28;53(2):678-88. doi: 10.1021/jm901273n.

PMID:
20000577
[PubMed - indexed for MEDLINE]
13.

Synthesis and preliminary in vitro evaluation of antimycobacterial activity of new pyrrolo[1,2-a] quinoxaline-carboxylic acid hydrazide derivatives.

Guillon J, Reynolds RC, Leger JM, Guie MA, Massip S, Dallemagne P, Jarry C.

J Enzyme Inhib Med Chem. 2004 Dec;19(6):489-95.

PMID:
15662953
[PubMed - indexed for MEDLINE]
14.

Four hydrazide compounds that inhibit the growth of mycobacterium tuberculosis.

Bartzatt R, Cirillo SL, Cirillo JD.

Physiol Chem Phys Med NMR. 2008;40:55-65.

PMID:
20070040
[PubMed - indexed for MEDLINE]
15.

Thiosemicarbazones, semicarbazones, dithiocarbazates and hydrazide/hydrazones: anti-Mycobacterium tuberculosis activity and cytotoxicity.

Pavan FR, da S Maia PI, Leite SR, Deflon VM, Batista AA, Sato DN, Franzblau SG, Leite CQ.

Eur J Med Chem. 2010 May;45(5):1898-905. doi: 10.1016/j.ejmech.2010.01.028. Epub 2010 Jan 28.

PMID:
20163897
[PubMed - indexed for MEDLINE]
16.

Synthesis, tuberculosis inhibitory activity, and SAR study of N-substituted-phenyl-1,2,3-triazole derivatives.

Costa MS, Boechat N, Rangel EA, da Silva Fde C, de Souza AM, Rodrigues CR, Castro HC, Junior IN, Lourenço MC, Wardell SM, Ferreira VF.

Bioorg Med Chem. 2006 Dec 15;14(24):8644-53. Epub 2006 Sep 1.

PMID:
16949290
[PubMed - indexed for MEDLINE]
17.

[Prospects for development of new antituberculous drugs].

Tomioka H.

Kekkaku. 2002 Aug;77(8):573-84. Japanese.

PMID:
12235850
[PubMed - indexed for MEDLINE]
18.

Synthesis and antituberculosis activity of some N-pyridyl-N'-thiazolylhydrazine derivatives.

Turan-Zitouni G, Kaplancikli ZA, Ozdemir A.

Eur J Med Chem. 2010 May;45(5):2085-8. doi: 10.1016/j.ejmech.2010.01.017. Epub 2010 Jan 20.

PMID:
20149489
[PubMed - indexed for MEDLINE]
19.

Synthesis and antituberculosis activity of new hydrazide derivatives.

Kaplancikli ZA, Turan-Zitouni G, Ozdemir A, Teulade JC.

Arch Pharm (Weinheim). 2008 Nov;341(11):721-4. doi: 10.1002/ardp.200800048.

PMID:
18720343
[PubMed - indexed for MEDLINE]
20.

Design, synthesis and antitubercular evaluation of novel series of N-[4-(piperazin-1-yl)phenyl]cinnamamide derivatives.

Patel KN, Telvekar VN.

Eur J Med Chem. 2014 Mar 21;75:43-56. doi: 10.1016/j.ejmech.2014.01.024. Epub 2014 Jan 25.

PMID:
24530490
[PubMed - indexed for MEDLINE]

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