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Items: 1 to 20 of 333

1.

Indapamide-like benzenesulfonamides as inhibitors of carbonic anhydrases I, II, VII, and XIII.

Čapkauskaitė E, Baranauskienė L, Golovenko D, Manakova E, Gražulis S, Tumkevičius S, Matulis D.

Bioorg Med Chem. 2010 Nov 1;18(21):7357-64. doi: 10.1016/j.bmc.2010.09.016. Epub 2010 Sep 15.

PMID:
20926301
2.

4-[N-(substituted 4-pyrimidinyl)amino]benzenesulfonamides as inhibitors of carbonic anhydrase isozymes I, II, VII, and XIII.

Sūdžius J, Baranauskienė L, Golovenko D, Matulienė J, Michailovienė V, Torresan J, Jachno J, Sukackaitė R, Manakova E, Gražulis S, Tumkevičius S, Matulis D.

Bioorg Med Chem. 2010 Nov 1;18(21):7413-21. doi: 10.1016/j.bmc.2010.09.011. Epub 2010 Sep 8.

PMID:
20889345
3.

Benzenesulfonamides with pyrimidine moiety as inhibitors of human carbonic anhydrases I, II, VI, VII, XII, and XIII.

Čapkauskaitė E, Zubrienė A, Smirnov A, Torresan J, Kišonaitė M, Kazokaitė J, Gylytė J, Michailovienė V, Jogaitė V, Manakova E, Gražulis S, Tumkevičius S, Matulis D.

Bioorg Med Chem. 2013 Nov 15;21(22):6937-47. doi: 10.1016/j.bmc.2013.09.029. Epub 2013 Sep 20.

PMID:
24103428
4.

Inhibition and binding studies of carbonic anhydrase isozymes I, II and IX with benzimidazo[1,2-c][1,2,3]thiadiazole-7-sulphonamides.

Baranauskienė L, Hilvo M, Matulienė J, Golovenko D, Manakova E, Dudutienė V, Michailovienė V, Torresan J, Jachno J, Parkkila S, Maresca A, Supuran CT, Gražulis S, Matulis D.

J Enzyme Inhib Med Chem. 2010 Dec;25(6):863-70. doi: 10.3109/14756360903571685. Epub 2010 Feb 18.

PMID:
20166809
5.

Carbonic anhydrase inhibitors: Synthesis and inhibition of the cytosolic mammalian carbonic anhydrase isoforms I, II and VII with benzene sulfonamides incorporating 4,5,6,7-tetrachlorophthalimide moiety.

Sethi KK, Verma SM, Tanç M, Carta F, Supuran CT.

Bioorg Med Chem. 2013 Sep 1;21(17):5168-74. doi: 10.1016/j.bmc.2013.06.035. Epub 2013 Jun 26.

PMID:
23867389
6.

Identification of 3,4-Dihydroisoquinoline-2(1H)-sulfonamides as potent carbonic anhydrase inhibitors: synthesis, biological evaluation, and enzyme--ligand X-ray studies.

Gitto R, Agnello S, Ferro S, De Luca L, Vullo D, Brynda J, Mader P, Supuran CT, Chimirri A.

J Med Chem. 2010 Mar 25;53(6):2401-8. doi: 10.1021/jm9014026.

PMID:
20170095
7.

Carbonic anhydrase inhibitors: novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II and IX.

Garaj V, Puccetti L, Fasolis G, Winum JY, Montero JL, Scozzafava A, Vullo D, Innocenti A, Supuran CT.

Bioorg Med Chem Lett. 2005 Jun 15;15(12):3102-8.

PMID:
15905091
8.

4-Substituted-2,3,5,6-tetrafluorobenzenesulfonamides as inhibitors of carbonic anhydrases I, II, VII, XII, and XIII.

Dudutienė V, Zubrienė A, Smirnov A, Gylytė J, Timm D, Manakova E, Gražulis S, Matulis D.

Bioorg Med Chem. 2013 Apr 1;21(7):2093-106. doi: 10.1016/j.bmc.2013.01.008. Epub 2013 Jan 16.

PMID:
23394791
9.

Design of [(2-pyrimidinylthio)acetyl]benzenesulfonamides as inhibitors of human carbonic anhydrases.

Čapkauskaitė E, Zubrienė A, Baranauskienė L, Tamulaitienė G, Manakova E, Kairys V, Gražulis S, Tumkevičius S, Matulis D.

Eur J Med Chem. 2012 May;51:259-70. doi: 10.1016/j.ejmech.2012.02.050. Epub 2012 Mar 3.

PMID:
22440859
10.

Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides derived from 4-isothiocyanato-benzolamide.

Cecchi A, Winum JY, Innocenti A, Vullo D, Montero JL, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett. 2004 Dec 6;14(23):5775-80.

PMID:
15501039
11.

Carbonic anhydrase inhibitors: synthesis and inhibition of the human cytosolic isozymes I and II and transmembrane isozymes IX, XII (cancer-associated) and XIV with 4-substituted 3-pyridinesulfonamides.

Brzozowski Z, Sławiński J, Saczewski F, Innocenti A, Supuran CT.

Eur J Med Chem. 2010 Jun;45(6):2396-404. doi: 10.1016/j.ejmech.2010.02.020. Epub 2010 Feb 12.

PMID:
20202722
12.

Carbonic anhydrase inhibitors. Interaction of indapamide and related diuretics with 12 mammalian isozymes and X-ray crystallographic studies for the indapamide-isozyme II adduct.

Temperini C, Cecchi A, Scozzafava A, Supuran CT.

Bioorg Med Chem Lett. 2008 Apr 15;18(8):2567-73. doi: 10.1016/j.bmcl.2008.03.051. Epub 2008 Mar 20.

PMID:
18374572
13.

5-Substituted-(1,2,3-triazol-4-yl)thiophene-2-sulfonamides strongly inhibit human carbonic anhydrases I, II, IX and XII: solution and X-ray crystallographic studies.

Leitans J, Sprudza A, Tanc M, Vozny I, Zalubovskis R, Tars K, Supuran CT.

Bioorg Med Chem. 2013 Sep 1;21(17):5130-8. doi: 10.1016/j.bmc.2013.06.041. Epub 2013 Jun 27.

PMID:
23859774
14.

Carbonic anhydrase inhibitors. Sulfonamide diuretics revisited--old leads for new applications?

Temperini C, Cecchi A, Scozzafava A, Supuran CT.

Org Biomol Chem. 2008 Jul 21;6(14):2499-506. doi: 10.1039/b800767e. Epub 2008 May 29.

PMID:
18600270
15.

Benzimidazo[1,2-c][1,2,3]thiadiazole-7-sulfonamides as inhibitors of carbonic anhydrase.

Dudutiene V, Baranauskiene L, Matulis D.

Bioorg Med Chem Lett. 2007 Jun 15;17(12):3335-8. Epub 2007 Apr 5.

PMID:
17442568
16.

New superacid synthesized (fluorinated) tertiary benzenesulfonamides acting as selective hCA IX inhibitors: toward a new mode of carbonic anhydrase inhibition by sulfonamides.

Métayer B, Mingot A, Vullo D, Supuran CT, Thibaudeau S.

Chem Commun (Camb). 2013 Jul 11;49(54):6015-7. doi: 10.1039/c3cc40858b.

PMID:
23503420
17.

Inhibition pattern of sulfamide-related compounds in binding to carbonic anhydrase isoforms I, II, VII, XII and XIV.

Gavernet L, Gonzalez Funes JL, Palestro PH, Bruno Blanch LE, Estiu GL, Maresca A, Barrios I, Supuran CT.

Bioorg Med Chem. 2013 Mar 15;21(6):1410-8. doi: 10.1016/j.bmc.2012.10.048. Epub 2012 Nov 29.

PMID:
23266178
18.
19.

In vitro inhibition of α-carbonic anhydrase isozymes by some phenolic compounds.

Oztürk Sarikaya SB, Topal F, Sentürk M, Gülçin I, Supuran CT.

Bioorg Med Chem Lett. 2011 Jul 15;21(14):4259-62. doi: 10.1016/j.bmcl.2011.05.071. Epub 2011 May 25.

PMID:
21669522
20.

Carbonic anhydrase inhibitors. Inhibition of the human cytosolic isozyme VII with aromatic and heterocyclic sulfonamides.

Vullo D, Voipio J, Innocenti A, Rivera C, Ranki H, Scozzafava A, Kaila K, Supuran CT.

Bioorg Med Chem Lett. 2005 Feb 15;15(4):971-6.

PMID:
15686895
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