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Items: 1 to 20 of 97

1.

Synthesis of [4-(2-hydroxyphenyl)thiazol-2-yl]methanones as potential bioisosteres of salicylidene acylhydrazides.

Hillgren JM, Dahlgren MK, To TM, Elofsson M.

Molecules. 2010 Aug 31;15(9):6019-34. doi: 10.3390/molecules15096019.

2.

Synthesis of 2-(2-aminopyrimidine)-2,2-difluoroethanols as potential bioisosters of salicylidene acylhydrazides.

Dahlgren MK, Oberg CT, Wallin EA, Janson PG, Elofsson M.

Molecules. 2010 Jun 21;15(6):4423-38. doi: 10.3390/molecules15064423.

3.

Synthesis and antimicrobial activity of novel 2-thiazolylimino-5-arylidene-4-thiazolidinones.

Vicini P, Geronikaki A, Anastasia K, Incerti M, Zani F.

Bioorg Med Chem. 2006 Jun 1;14(11):3859-64. Epub 2006 Feb 20.

PMID:
16488614
4.

Synthesis and in vitro antibacterial activity of 3-[N-methyl-N-(3-methyl-1,3-thiazolium-2-yl)aminolmethyl cephalosporin derivatives.

Kim SH, Son H, Nam G, Chi DY, Kim JH.

Bioorg Med Chem Lett. 2000 Jun 5;10(11):1143-5.

PMID:
10866367
5.

Statistical molecular design of a focused salicylidene acylhydrazide library and multivariate QSAR of inhibition of type III secretion in the Gram-negative bacterium Yersinia.

Dahlgren MK, Zetterström CE, Gylfe S, Linusson A, Elofsson M.

Bioorg Med Chem. 2010 Apr 1;18(7):2686-703. doi: 10.1016/j.bmc.2010.02.022. Epub 2010 Feb 18.

PMID:
20219378
6.

Combinatorial approach toward synthesis of small molecule libraries as bacterial transglycosylase inhibitors.

Shih HW, Chen KT, Chen SK, Huang CY, Cheng TJ, Ma C, Wong CH, Cheng WC.

Org Biomol Chem. 2010 Jun 7;8(11):2586-93. doi: 10.1039/c000622j. Epub 2010 Mar 29.

PMID:
20485795
7.

Design, synthesis and biological evaluation of novel thiazole derivatives as potent FabH inhibitors.

Lv PC, Wang KR, Yang Y, Mao WJ, Chen J, Xiong J, Zhu HL.

Bioorg Med Chem Lett. 2009 Dec 1;19(23):6750-4. doi: 10.1016/j.bmcl.2009.09.111. Epub 2009 Oct 2.

PMID:
19836235
8.

Identification of aryl 2-aminoimidazoles as biofilm inhibitors in Gram-negative bacteria.

Bunders CA, Richards JJ, Melander C.

Bioorg Med Chem Lett. 2010 Jun 15;20(12):3797-800. doi: 10.1016/j.bmcl.2010.04.042. Epub 2010 Apr 18.

PMID:
20466544
9.

Virulence blockers as alternatives to antibiotics: type III secretion inhibitors against Gram-negative bacteria.

Keyser P, Elofsson M, Rosell S, Wolf-Watz H.

J Intern Med. 2008 Jul;264(1):17-29. doi: 10.1111/j.1365-2796.2008.01941.x. Epub 2008 Apr 3.

10.
11.

Synthesis and in vitro antibacterial activities of 3-thiazol-4-yl-1-carba-1-dethiacephalosporins.

Hornback WJ, Munroe JE, Counter FT.

J Antibiot (Tokyo). 1994 Sep;47(9):1052-64.

13.

[Synthesis of derivatives of 2-(2-amino-1,3- thiazol-4-yl)-2-hydroxyiminoacetic acid].

Shiliaeva SV, Gorbunova SM.

Antibiot Khimioter. 1988 Sep;33(9):714-8. Review. Russian. No abstract available.

PMID:
3064724
14.

Synthesis and biological evaluation of some 2,4,5-trisubstituted thiazole derivatives as potential antimicrobial and anticancer agents.

Al-Saadi MS, Faidallah HM, Rostom SA.

Arch Pharm (Weinheim). 2008 Jul;341(7):424-34. doi: 10.1002/ardp.200800026.

PMID:
18574850
15.

Synthesis and antibiotic activity of a small molecules library of 1,2,3-triazole derivatives.

Aufort M, Herscovici J, Bouhours P, Moreau N, Girard C.

Bioorg Med Chem Lett. 2008 Feb 1;18(3):1195-8. Epub 2007 Dec 4.

PMID:
18086525
17.

Solution-phase synthesis of a combinatorial library of 3-[4-(coumarin-3-yl)-1,3-thiazol-2-ylcarbamoyl]propanoic acid amides.

Zhuravel IO, Kovalenko SM, Vlasov SV, Chernykh VP.

Molecules. 2005 Feb 28;10(2):444-56.

18.

Synthesis of some bioactive 2-bromo-5-methoxy-N'-[4-(aryl)-1,3-thiazol-2-yl]benzohydrazide derivatives.

Vijaya Raj KK, Narayana B, Ashalatha BV, Suchetha Kumari N, Sarojini BK.

Eur J Med Chem. 2007 Mar;42(3):425-9. Epub 2006 Oct 30.

PMID:
17074422
19.

Synthesis, anti-bacterial and anti-fungal activities of some novel Schiff bases containing 2,4-disubstituted thiazole ring.

Bharti SK, Nath G, Tilak R, Singh SK.

Eur J Med Chem. 2010 Feb;45(2):651-60. doi: 10.1016/j.ejmech.2009.11.008. Epub 2009 Nov 6.

PMID:
19932927
20.

Solution versus fluorous versus solid-phase synthesis of 2,5-disubstituted 1,3-azoles. Preliminary antibacterial activity studies.

Sanz-Cervera JF, Blasco R, Piera J, Cynamon M, Ibáñez I, Murguía M, Fustero S.

J Org Chem. 2009 Dec 4;74(23):8988-96. doi: 10.1021/jo9016265.

PMID:
19894729
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