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Results: 1 to 20 of 100

1.

Conformationally-restricted amino acid analogues bearing a distal sulfonic acid show selective inhibition of system x(c)(-) over the vesicular glutamate transporter.

Etoga JL, Ahmed SK, Patel S, Bridges RJ, Thompson CM.

Bioorg Med Chem Lett. 2010 Apr 15;20(8):2680-3. doi: 10.1016/j.bmcl.2009.10.020. Epub 2009 Oct 12.

PMID:
20303751
[PubMed - indexed for MEDLINE]
Free PMC Article
2.

Inhibitor of the glutamate vesicular transporter (VGLUT).

Thompson CM, Davis E, Carrigan CN, Cox HD, Bridges RJ, Gerdes JM.

Curr Med Chem. 2005;12(18):2041-56. Review.

PMID:
16101493
[PubMed - indexed for MEDLINE]
3.

Synthesis and preliminary evaluation of trans-3,4-conformationally-restricted glutamate and pyroglutamate analogues as novel EAAT2 inhibitors.

Denton T, Seib T, Bridges R, Thompson C.

Bioorg Med Chem Lett. 2002 Nov 4;12(21):3209-13.

PMID:
12372536
[PubMed - indexed for MEDLINE]
4.

Use of the hydantoin isostere to produce inhibitors showing selectivity toward the vesicular glutamate transporter versus the obligate exchange transporter system x(c)(-).

Ahmed SK, Etoga JL, Patel SA, Bridges RJ, Thompson CM.

Bioorg Med Chem Lett. 2011 Jul 15;21(14):4358-62. doi: 10.1016/j.bmcl.2011.05.018. Epub 2011 May 14.

PMID:
21669531
[PubMed - indexed for MEDLINE]
Free PMC Article
5.

Synthesis and in vitro pharmacology of substituted quinoline-2,4-dicarboxylic acids as inhibitors of vesicular glutamate transport.

Carrigan CN, Bartlett RD, Esslinger CS, Cybulski KA, Tongcharoensirikul P, Bridges RJ, Thompson CM.

J Med Chem. 2002 May 23;45(11):2260-76.

PMID:
12014964
[PubMed - indexed for MEDLINE]
7.

Uptake of L-glutamate into synaptic vesicles: competitive inhibition by dyes with biphenyl and amino- and sulphonic acid-substituted naphthyl groups.

Roseth S, Fykse EM, Fonnum F.

Biochem Pharmacol. 1998 Nov 1;56(9):1243-9.

PMID:
9802337
[PubMed - indexed for MEDLINE]
8.

Expression of the vesicular glutamate transporters during development indicates the widespread corelease of multiple neurotransmitters.

Boulland JL, Qureshi T, Seal RP, Rafiki A, Gundersen V, Bergersen LH, Fremeau RT Jr, Edwards RH, Storm-Mathisen J, Chaudhry FA.

J Comp Neurol. 2004 Dec 13;480(3):264-80.

PMID:
15515175
[PubMed - indexed for MEDLINE]
9.

The SLC32 transporter, a key protein for the synaptic release of inhibitory amino acids.

Gasnier B.

Pflugers Arch. 2004 Feb;447(5):756-9. Epub 2003 May 16. Review.

PMID:
12750892
[PubMed - indexed for MEDLINE]
10.

Identification of selective norbornane-type aspartate analogue inhibitors of the glutamate transporter 1 (GLT-1) from the chemical universe generated database (GDB).

Luethi E, Nguyen KT, Bürzle M, Blum LC, Suzuki Y, Hediger M, Reymond JL.

J Med Chem. 2010 Oct 14;53(19):7236-50. doi: 10.1021/jm100959g.

PMID:
20812729
[PubMed - indexed for MEDLINE]
11.

Effects of L-glutamate transport inhibition by a conformationally restricted glutamate analogue (2S,1'S,2'R)-2-(carboxycyclopropyl)glycine (L-CCG III) on metabolism in brain tissue in vitro analysed by NMR spectroscopy.

Moussa Cel-H, Mitrovic AD, Vandenberg RJ, Provis T, Rae C, Bubb WA, Balcar VJ.

Neurochem Res. 2002 Feb;27(1-2):27-35.

PMID:
11926273
[PubMed - indexed for MEDLINE]
12.
13.

Inhibition by folded isomers of L-2-(carboxycyclopropyl)glycine of glutamate uptake via the human glutamate transporter hGluT-1.

Yamashita H, Kawakami H, Zhang YX, Hagiwara T, Tanaka K, Nakamura S.

Eur J Pharmacol. 1995 Apr 28;289(2):387-90.

PMID:
7621914
[PubMed - indexed for MEDLINE]
14.

Human vesicular glutamate transporters functionally complement EAT-4 in C. elegans.

Lee D, Jung S, Ryu J, Ahnn J, Ha I.

Mol Cells. 2008 Feb 29;25(1):50-4.

PMID:
18319613
[PubMed - indexed for MEDLINE]
Free Article
15.

Tetrapeptide inhibitors of the glutamate vesicular transporter (VGLUT).

Patel SA, Nagy JO, Bolstad ED, Gerdes JM, Thompson CM.

Bioorg Med Chem Lett. 2007 Sep 15;17(18):5125-8. Epub 2007 Jul 26.

PMID:
17662605
[PubMed - indexed for MEDLINE]
Free PMC Article
16.

Molecular identification and characterisation of the glycine transporter (GLYT1) and the glutamine/glutamate transporter (ASCT2) in the rat lens.

Lim J, Lorentzen KA, Kistler J, Donaldson PJ.

Exp Eye Res. 2006 Aug;83(2):447-55. Epub 2006 Apr 25.

PMID:
16635486
[PubMed - indexed for MEDLINE]
17.

N-methyl-D-aspartate autoreceptors respond to low and high agonist concentrations by facilitating, respectively, exocytosis and carrier-mediated release of glutamate in rat hippocampus.

Luccini E, Musante V, Neri E, Raiteri M, Pittaluga A.

J Neurosci Res. 2007 Dec;85(16):3657-65.

PMID:
17671992
[PubMed - indexed for MEDLINE]
18.

Vesicular glutamate transporter acts as a metabolic regulator.

Moriyama Y, Omote H.

Biol Pharm Bull. 2008 Oct;31(10):1844-6. Review.

PMID:
18827340
[PubMed - indexed for MEDLINE]
Free Article
19.

Synthesis, molecular modeling studies, and preliminary pharmacological characterization of all possible 2-(2'-sulfonocyclopropyl)glycine stereoisomers as conformationally constrained L-homocysteic acid analogs.

Pellicciari R, Marinozzi M, Macchiarulo A, Fulco MC, Gafarova J, Serpi M, Giorgi G, Nielsen S, Thomsen C.

J Med Chem. 2007 Sep 20;50(19):4630-41. Epub 2007 Aug 29.

PMID:
17725337
[PubMed - indexed for MEDLINE]
20.

Plasma membrane and vesicular glutamate transporter mRNAs/proteins in hypothalamic neurons that regulate body weight.

Collin M, Bäckberg M, Ovesjö ML, Fisone G, Edwards RH, Fujiyama F, Meister B.

Eur J Neurosci. 2003 Sep;18(5):1265-78. Erratum in: Eur J Neurosci. 2003 Sep;18(6):1717.

PMID:
12956725
[PubMed - indexed for MEDLINE]

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