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Results: 1 to 20 of 111

1.

1-(2-Aminoethyl)-3-(arylsulfonyl)-1H-pyrrolopyridines are 5-HT(6) receptor ligands.

Bernotas RC, Antane SA, Lenicek SE, Haydar SN, Robichaud AJ, Harrison BL, Zhang GM, Smith D, Coupet J, Schechter LE.

Bioorg Med Chem Lett. 2009 Dec 15;19(24):6935-8. doi: 10.1016/j.bmcl.2009.10.067. Epub 2009 Oct 20.

PMID:
19884004
[PubMed - indexed for MEDLINE]
2.

Novel 1-(azacyclyl)-3-arylsulfonyl-1H-pyrrolo[2,3-b]pyridines as 5-HT6 agonists and antagonists.

Elokdah H, Li D, McFarlane G, Bernotas RC, Robichaud AJ, Magolda RL, Zhang GM, Smith D, Schechter LE.

Bioorg Med Chem. 2007 Sep 15;15(18):6208-26. Epub 2007 Jun 14.

PMID:
17624788
[PubMed - indexed for MEDLINE]
3.

3-(Arylsulfonyl)-1-(azacyclyl)-1H-indoles are 5-HT(6) receptor modulators.

Bernotas RC, Antane S, Shenoy R, Le VD, Chen P, Harrison BL, Robichaud AJ, Zhang GM, Smith D, Schechter LE.

Bioorg Med Chem Lett. 2010 Mar 1;20(5):1657-60. doi: 10.1016/j.bmcl.2010.01.073. Epub 2010 Jan 21.

PMID:
20138763
[PubMed - indexed for MEDLINE]
4.

Novel 1-aminoethyl-3-arylsulfonyl-1H-pyrrolo[2,3-b]pyridines are potent 5-HT(6) agonists.

Bernotas RC, Lenicek S, Antane S, Cole DC, Harrison BL, Robichaud AJ, Zhang GM, Smith D, Platt B, Lin Q, Li P, Coupet J, Rosenzweig-Lipson S, Beyer CE, Schechter LE.

Bioorg Med Chem. 2009 Jul 15;17(14):5153-63. doi: 10.1016/j.bmc.2009.05.055. Epub 2009 May 29.

PMID:
19523834
[PubMed - indexed for MEDLINE]
5.

1-(2-Aminoethyl)-3-(arylsulfonyl)-1H-indoles as novel 5-HT6 receptor ligands.

Bernotas R, Lenicek S, Antane S, Zhang GM, Smith D, Coupet J, Harrison B, Schechter LE.

Bioorg Med Chem Lett. 2004 Nov 15;14(22):5499-502.

PMID:
15482912
[PubMed - indexed for MEDLINE]
6.

Pyrroloquinoxaline derivatives as high-affinity and selective 5-HT(3) receptor agonists: synthesis, further structure-activity relationships, and biological studies.

Campiani G, Morelli E, Gemma S, Nacci V, Butini S, Hamon M, Novellino E, Greco G, Cagnotto A, Goegan M, Cervo L, Dalla Valle F, Fracasso C, Caccia S, Mennini T.

J Med Chem. 1999 Oct 21;42(21):4362-79.

PMID:
10543880
[PubMed - indexed for MEDLINE]
7.

The putative <<silent>> 5-HT(1A) receptor antagonist, WAY 100635, has inverse agonist properties at cloned human 5-HT(1A) receptors.

Cosi C, Koek W.

Eur J Pharmacol. 2000 Jul 28;401(1):9-15.

PMID:
10915831
[PubMed - indexed for MEDLINE]
8.

Specific labelling of serotonin 5-HT(1B) receptors in rat frontal cortex with the novel, phenylpiperazine derivative, [3H]GR125,743. A pharmacological characterization.

Millan MJ, Newman-Tancredi A, Lochon S, Touzard M, Aubry S, Audinot V.

Pharmacol Biochem Behav. 2002 Apr;71(4):589-98.

PMID:
11888550
[PubMed - indexed for MEDLINE]
9.

1,2,5-Thiadiazole derivatives are potent and selective ligands at human 5-HT1A receptors.

Sabb AL, Vogel RL, Kelly MG, Palmer Y, Smith DL, Andree TH, Schechter LE.

Bioorg Med Chem Lett. 2001 Apr 23;11(8):1069-71.

PMID:
11327592
[PubMed - indexed for MEDLINE]
10.

Synthesis and structure-affinity relationships of novel N-(1-ethyl-4-methylhexahydro-1,4-diazepin-6-yl)pyridine-3-carboxamides with potent serotonin 5-HT3 and dopamine D2 receptor antagonistic activity.

Hirokawa Y, Fujiwara I, Suzuki K, Harada H, Yoshikawa T, Yoshida N, Kato S.

J Med Chem. 2003 Feb 27;46(5):702-15.

PMID:
12593651
[PubMed - indexed for MEDLINE]
11.

2,3-Dihydro-2-oxo-1H-benzimidazole-1-carboxamides with selective affinity for the 5-HT(4) receptor: synthesis and structure-affinity and structure-activity relationships of a new series of partial agonist and antagonist derivatives.

Tapia I, Alonso-Cires L, López-Tudanca PL, Mosquera R, Labeaga L, Innerárity A, Orjales A.

J Med Chem. 1999 Jul 29;42(15):2870-80.

PMID:
10425096
[PubMed - indexed for MEDLINE]
12.

Novel 2-aminotetralin and 3-aminochroman derivatives as selective serotonin 5-HT7 receptor agonists and antagonists.

Holmberg P, Sohn D, Leideborg R, Caldirola P, Zlatoidsky P, Hanson S, Mohell N, Rosqvist S, Nordvall G, Johansson AM, Johansson R.

J Med Chem. 2004 Jul 29;47(16):3927-30.

PMID:
15267230
[PubMed - indexed for MEDLINE]
13.

1-(Arylsulfonyl)-2,3-dihydro-1H-quinolin-4-one derivatives as 5-HT(6) serotonin receptor ligands.

Park CM, Choi JI, Choi JH, Kim SY, Park WK, Seong CM.

Bioorg Med Chem Lett. 2011 Jan 15;21(2):698-703. doi: 10.1016/j.bmcl.2010.12.007. Epub 2010 Dec 8.

PMID:
21190848
[PubMed - indexed for MEDLINE]
14.

Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).

Glennon RA.

J Med Chem. 2003 Jul 3;46(14):2795-812. Review. No abstract available.

PMID:
12825922
[PubMed - indexed for MEDLINE]
15.

Structure-affinity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agents.

Leopoldo M, Berardi F, Colabufo NA, Contino M, Lacivita E, Niso M, Perrone R, Tortorella V.

J Med Chem. 2004 Dec 16;47(26):6616-24.

PMID:
15588097
[PubMed - indexed for MEDLINE]
16.

Synthesis of new serotonin 5-HT7 receptor ligands. Determinants of 5-HT7/5-HT1A receptor selectivity.

Medina RA, Sallander J, Benhamú B, Porras E, Campillo M, Pardo L, López-Rodríguez ML.

J Med Chem. 2009 Apr 23;52(8):2384-92. doi: 10.1021/jm8014553.

PMID:
19326916
[PubMed - indexed for MEDLINE]
17.

Synthesis and molecular modeling of new 1-aryl-3-[4-arylpiperazin-1-yl]-1-propane derivatives with high affinity at the serotonin transporter and at 5-HT(1A) receptors.

Orús L, Pérez-Silanes S, Oficialdegui AM, Martínez-Esparza J, Del Castillo JC, Mourelle M, Langer T, Guccione S, Donzella G, Krovat EM, Poptodorov K, Lasheras B, Ballaz S, Hervías I, Tordera R, Del Río J, Monge A.

J Med Chem. 2002 Sep 12;45(19):4128-39.

PMID:
12213056
[PubMed - indexed for MEDLINE]
18.

2-Substituted tryptamines: agents with selectivity for 5-HT(6) serotonin receptors.

Glennon RA, Lee M, Rangisetty JB, Dukat M, Roth BL, Savage JE, McBride A, Rauser L, Hufeisen S, Lee DK.

J Med Chem. 2000 Mar 9;43(5):1011-8.

PMID:
10715164
[PubMed - indexed for MEDLINE]
19.

Active conformation of some arylpiperazine postsynaptic 5-HT(1A) receptor antagonists.

Paluchowska MH, Bojarski AJ, Charakchieva-Minol S, Wesołowska A.

Eur J Med Chem. 2002 Apr;37(4):273-83.

PMID:
11960662
[PubMed - indexed for MEDLINE]
20.

Arylpiperazine derivatives acting at 5-HT(1A) receptors.

López-Rodríguez ML, Ayala D, Benhamú B, Morcillo MJ, Viso A.

Curr Med Chem. 2002 Feb;9(4):443-69. Review.

PMID:
11945120
[PubMed - indexed for MEDLINE]

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