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Similar articles for PubMed (Select 19804380)

1.

Relative positioning of diazepam in the benzodiazepine-binding-pocket of GABA receptors.

Tan KR, Baur R, Charon S, Goeldner M, Sigel E.

J Neurochem. 2009 Dec;111(5):1264-73. doi: 10.1111/j.1471-4159.2009.06419.x. Epub 2009 Oct 5.

PMID:
19804380
2.
3.

On the benzodiazepine binding pocket in GABAA receptors.

Berezhnoy D, Nyfeler Y, Gonthier A, Schwob H, Goeldner M, Sigel E.

J Biol Chem. 2004 Jan 30;279(5):3160-8. Epub 2003 Nov 11.

4.

Covalent modification of GABAA receptor isoforms by a diazepam analogue provides evidence for a novel benzodiazepine binding site that prevents modulation by these drugs.

Baur R, Tan KR, Lüscher BP, Gonthier A, Goeldner M, Sigel E.

J Neurochem. 2008 Sep;106(6):2353-63. doi: 10.1111/j.1471-4159.2008.05574.x. Epub 2008 Jul 15.

PMID:
18643789
5.

Flavan-3-ol derivatives are positive modulators of GABA(A) receptors with higher efficacy for the alpha(2) subtype and anxiolytic action in mice.

Fernandez SP, Mewett KN, Hanrahan JR, Chebib M, Johnston GA.

Neuropharmacology. 2008 Oct;55(5):900-7. doi: 10.1016/j.neuropharm.2008.06.069. Epub 2008 Jul 9.

PMID:
18657554
7.
8.

Two neighboring residues of loop A of the alpha1 subunit point towards the benzodiazepine binding site of GABAA receptors.

Tan KR, Baur R, Gonthier A, Goeldner M, Sigel E.

FEBS Lett. 2007 Oct 2;581(24):4718-22. Epub 2007 Sep 6.

10.

Benzodiazepine actions mediated by specific gamma-aminobutyric acid(A) receptor subtypes.

Rudolph U, Crestani F, Benke D, Brünig I, Benson JA, Fritschy JM, Martin JR, Bluethmann H, Möhler H.

Nature. 1999 Oct 21;401(6755):796-800. Erratum in: Nature 2000 Apr 6;404(6778):629.

PMID:
10548105
12.

Pharmacological modulation of the diazepam-insensitive recombinant gamma-aminobutyric acidA receptors alpha 4 beta 2 gamma 2 and alpha 6 beta 2 gamma 2.

Knoflach F, Benke D, Wang Y, Scheurer L, Lüddens H, Hamilton BJ, Carter DB, Mohler H, Benson JA.

Mol Pharmacol. 1996 Nov;50(5):1253-61.

PMID:
8913357
13.
14.

Relative positioning of classical benzodiazepines to the γ2-subunit of GABAA receptors.

Middendorp SJ, Hurni E, Schönberger M, Stein M, Pangerl M, Trauner D, Sigel E.

ACS Chem Biol. 2014 Aug 15;9(8):1846-53. doi: 10.1021/cb500186a. Epub 2014 Jul 1.

PMID:
24918742
16.

The anxioselective agent 7-(2-chloropyridin-4-yl)pyrazolo-[1,5-a]-pyrimidin-3-yl](pyridin-2-yl)methanone (DOV 51892) is more efficacious than diazepam at enhancing GABA-gated currents at alpha1 subunit-containing GABAA receptors.

Popik P, Kostakis E, Krawczyk M, Nowak G, Szewczyk B, Krieter P, Chen Z, Russek SJ, Gibbs TT, Farb DH, Skolnick P, Lippa AS, Basile AS.

J Pharmacol Exp Ther. 2006 Dec;319(3):1244-52. Epub 2006 Sep 13.

18.

Individually monitoring ligand-induced changes in the structure of the GABAA receptor at benzodiazepine binding site and non-binding-site interfaces.

Sharkey LM, Czajkowski C.

Mol Pharmacol. 2008 Jul;74(1):203-12. doi: 10.1124/mol.108.044891. Epub 2008 Apr 18.

19.
20.

A closer look at the high affinity benzodiazepine binding site on GABAA receptors.

Sigel E, Lüscher BP.

Curr Top Med Chem. 2011;11(2):241-6. Review.

PMID:
21189125
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