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Items: 1 to 20 of 724

1.

Synthesis of methoxypoly(ethylene glycol) carbonate prodrugs of zidovudine and penetration through human skin in vitro.

N'da DD, Breytenbach JC.

J Pharm Pharmacol. 2009 Jun;61(6):721-31. doi: 10.1211/jpp.61.06.0004.

PMID:
19505362
2.

Synthesis and in vitro transdermal penetration of methoxypoly(ethylene glycol) carbonate derivatives of stavudine.

N'Da DD, Breytenbach JC, Legoabe LJ, Breytenbach JW.

Med Chem. 2009 Nov;5(6):497-506.

PMID:
19673696
3.

Synthesis and in vitro human skin penetration of oligo- and polymeric ethylene glycol carbonates of zidovudine and stavudine.

N'Da DD, Breytenbach JC, Breytenbach JW.

Arzneimittelforschung. 2010;60(9):575-82. doi: 10.1055/s-0031-1296328.

PMID:
21117502
4.

Synthesis and in vitro transdermal penetration of methoxypoly(ethylene glycol) carbonate and carbamate derivatives of lamivudine (3TC).

van Heerden J, Breytenbach JC, N'Da DD, Breytenbach JW, du Preez JL.

Med Chem. 2010 Mar;6(2):91-9.

PMID:
20158460
5.

Dipeptide derivatives of AZT: synthesis, chemical stability, activation in human plasma, hPEPT1 affinity, and antiviral activity.

Santos C, Morais J, Gouveia L, de Clercq E, Pannecouque C, Nielsen CU, Steffansen B, Moreira R, Gomes P.

ChemMedChem. 2008 Jun;3(6):970-8. doi: 10.1002/cmdc.200800012.

PMID:
18389514
6.

Novel approaches for designing 5'-O-ester prodrugs of 3'-azido-2', 3'-dideoxythymidine (AZT).

Parang K, Wiebe LI, Knaus EE.

Curr Med Chem. 2000 Oct;7(10):995-1039. Review.

PMID:
10911016
7.

New 3'-azido-3'-deoxythymidin-5'-yl O-(4-hydroxyalkyl or -alkenyl or -alkylepoxide) carbonate prodrugs: synthesis and anti-HIV evaluation.

Vlieghe P, Clerc T, Pannecouque C, Witvrouw M, De Clercq E, Salles JP, Kraus JL.

J Med Chem. 2001 Aug 30;44(18):3014-21.

PMID:
11520210
8.

New 3'-azido-3'-deoxythymidin-5'-yl O-(omega-hydroxyalkyl) carbonate prodrugs: synthesis and anti-HIV evaluation.

Vlieghe P, Bihel F, Clerc T, Pannecouque C, Witvrouw M, De Clercq E, Salles JP, Chermann JC, Kraus JL.

J Med Chem. 2001 Mar 1;44(5):777-86.

PMID:
11262088
9.

Enhanced delivery of zidovudine through rat and human skin via ester prodrugs.

Seki T, Kawaguchi T, Juni K.

Pharm Res. 1990 Sep;7(9):948-52.

PMID:
2235895
10.

Self-assembled drug delivery systems. Part 4. In vitro/in vivo studies of the self-assemblies of cholesteryl-phosphonyl zidovudine.

Jin Y, Xing L, Tian Y, Li M, Gao C, Du L, Dong J, Chen H.

Int J Pharm. 2009 Oct 20;381(1):40-8. doi: 10.1016/j.ijpharm.2009.07.024. Epub 2009 Jul 29. Erratum in: Int J Pharm. 2010 Sep 15;397(1-2):231.

PMID:
19646518
11.

Synthesis, in vitro and in vivo release kinetics, and anti-HIV activity of a sustained-release prodrug (mPEG-AZT) of 3'-azido-3'-deoxythymidine (AZT, Zidovudine).

Li W, Chang Y, Zhan P, Zhang N, Liu X, Pannecouque C, De Clercq E.

ChemMedChem. 2010 Nov 8;5(11):1893-8. doi: 10.1002/cmdc.201000352.

PMID:
20936623
12.

Transdermal delivery system for zidovudine: in vitro, ex vivo and in vivo evaluation.

Narishetty ST, Panchagnula R.

Biopharm Drug Dispos. 2004 Jan;25(1):9-20.

PMID:
14716748
13.

Enhanced transdermal delivery of AZT (Zidovudine) using iontophoresis and penetration enhancer.

Oh SY, Jeong SY, Park TG, Lee JH.

J Control Release. 1998 Feb 12;51(2-3):161-8.

PMID:
9685913
14.
15.

Synthesis of piperazinylalkyl ester prodrugs of ketorolac and their in vitro evaluation for transdermal delivery.

Qandil A, Al-Nabulsi S, Al-Taani B, Tashtoush B.

Drug Dev Ind Pharm. 2008 Oct;34(10):1054-63. doi: 10.1080/03639040801946681 .

PMID:
18608464
16.

Synthesis and transdermal permeation of novel N4-methoxypoly(ethylene glycol) carbamates of cytarabine.

Legoabe LJ, N'Da DD, Breytenbach JC, du Preez JL, du Plessis J.

Drug Dev Ind Pharm. 2010 Dec;36(12):1477-85. doi: 10.3109/03639045.2010.488646. Epub 2010 Jun 19.

PMID:
20560790
17.

Combination strategies to enhance transdermal permeation of zidovudine (AZT).

Thomas NS, Panchagnula R.

Pharmazie. 2003 Dec;58(12):895-8.

PMID:
14703969
18.
19.

Enhanced delivery of AZT to macrophages via acetylated LDL.

Hu J, Liu H, Wang L.

J Control Release. 2000 Dec 3;69(3):327-35.

PMID:
11102673
20.

Human skin permeation of branched-chain 3-0-alkyl ester and carbonate prodrugs of naltrexone.

Vaddi HK, Hamad MO, Chen J, Banks SL, Crooks PA, Stinchcomb AL.

Pharm Res. 2005 May;22(5):758-65. Epub 2005 May 17.

PMID:
15906171
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