Similar articles for PMID: 19282189

Year	Number of Results
1958	2
1967	1
1968	1
1974	1
1982	3
1987	1
1988	1
1990	2
1991	1
1992	1
1994	1
1998	1
2000	1
2002	1
2003	1
2004	6
2005	11
2006	18
2007	8
2008	31
2009	92
2010	10
2011	15
2012	13
2013	12
2014	17
2015	9
2016	5
2017	6
2018	4
2019	4
2020	3
2022	2
2024	0

1

Discovery of potent and orally active 3-alkoxy-5-phenoxy-N-thiazolyl benzamides as novel allosteric glucokinase activators.

Iino T, Tsukahara D, Kamata K, Sasaki K, Ohyama S, Hosaka H, Hasegawa T, Chiba M, Nagata Y, Eiki J, Nishimura T. Iino T, et al. Bioorg Med Chem. 2009 Apr 1;17(7):2733-43. doi: 10.1016/j.bmc.2009.02.038. Epub 2009 Feb 25. Bioorg Med Chem. 2009. PMID: 19282189

2

Structure-activity relationships of 3,5-disubstituted benzamides as glucokinase activators with potent in vivo efficacy.

Iino T, Hashimoto N, Sasaki K, Ohyama S, Yoshimoto R, Hosaka H, Hasegawa T, Chiba M, Nagata Y, Eiki J, Nishimura T. Iino T, et al. Bioorg Med Chem. 2009 Jun 1;17(11):3800-9. doi: 10.1016/j.bmc.2009.04.040. Epub 2009 Apr 24. Bioorg Med Chem. 2009. PMID: 19427223

3

Discovery and structure-activity relationships of a novel class of quinazoline glucokinase activators.

Iino T, Sasaki Y, Bamba M, Mitsuya M, Ohno A, Kamata K, Hosaka H, Maruki H, Futamura M, Yoshimoto R, Ohyama S, Sasaki K, Chiba M, Ohtake N, Nagata Y, Eiki J, Nishimura T. Iino T, et al. Bioorg Med Chem Lett. 2009 Oct 1;19(19):5531-8. doi: 10.1016/j.bmcl.2009.08.064. Epub 2009 Aug 21. Bioorg Med Chem Lett. 2009. PMID: 19726182

4

Identification of novel and potent 2-amino benzamide derivatives as allosteric glucokinase activators.

Nishimura T, Iino T, Mitsuya M, Bamba M, Watanabe H, Tsukahara D, Kamata K, Sasaki K, Ohyama S, Hosaka H, Futamura M, Nagata Y, Eiki J. Nishimura T, et al. Bioorg Med Chem Lett. 2009 Mar 1;19(5):1357-60. doi: 10.1016/j.bmcl.2009.01.053. Epub 2009 Jan 21. Bioorg Med Chem Lett. 2009. PMID: 19188063

5

Design, synthesis, and pharmacological evaluation of benzamide derivatives as glucokinase activators.

Mao W, Ning M, Liu Z, Zhu Q, Leng Y, Zhang A. Mao W, et al. Bioorg Med Chem. 2012 May 1;20(9):2982-91. doi: 10.1016/j.bmc.2012.03.008. Epub 2012 Mar 8. Bioorg Med Chem. 2012. PMID: 22459213

6

Discovery of 3-(4-methanesulfonylphenoxy)-N-[1-(2-methoxy-ethoxymethyl)-1H-pyrazol-3-yl]-5-(3-methylpyridin-2-yl)-benzamide as a novel glucokinase activator (GKA) for the treatment of type 2 diabetes mellitus.

Park K, Lee BM, Hyun KH, Lee DH, Choi HH, Kim H, Chong W, Kim KB, Nam SY. Park K, et al. Bioorg Med Chem. 2014 Apr 1;22(7):2280-93. doi: 10.1016/j.bmc.2014.02.009. Epub 2014 Feb 17. Bioorg Med Chem. 2014. PMID: 24588963

7

Discovery of novel 3,6-disubstituted 2-pyridinecarboxamide derivatives as GK activators.

Mitsuya M, Kamata K, Bamba M, Watanabe H, Sasaki Y, Sasaki K, Ohyama S, Hosaka H, Nagata Y, Eiki J, Nishimura T. Mitsuya M, et al. Bioorg Med Chem Lett. 2009 May 15;19(10):2718-21. doi: 10.1016/j.bmcl.2009.03.137. Epub 2009 Mar 29. Bioorg Med Chem Lett. 2009. PMID: 19362831

8

Discovery of novel 2-(pyridine-2-yl)-1H-benzimidazole derivatives as potent glucokinase activators.

Ishikawa M, Nonoshita K, Ogino Y, Nagae Y, Tsukahara D, Hosaka H, Maruki H, Ohyama S, Yoshimoto R, Sasaki K, Nagata Y, Eiki J, Nishimura T. Ishikawa M, et al. Bioorg Med Chem Lett. 2009 Aug 1;19(15):4450-4. doi: 10.1016/j.bmcl.2009.05.038. Epub 2009 May 18. Bioorg Med Chem Lett. 2009. PMID: 19540111

9

SAR, pharmacokinetics, safety, and efficacy of glucokinase activating 2-(4-sulfonylphenyl)-N-thiazol-2-ylacetamides: discovery of PSN-GK1.

Bertram LS, Black D, Briner PH, Chatfield R, Cooke A, Fyfe MC, Murray PJ, Naud F, Nawano M, Procter MJ, Rakipovski G, Rasamison CM, Reynet C, Schofield KL, Shah VK, Spindler F, Taylor A, Turton R, Williams GM, Wong-Kai-In P, Yasuda K. Bertram LS, et al. J Med Chem. 2008 Jul 24;51(14):4340-5. doi: 10.1021/jm8003202. Epub 2008 Jun 28. J Med Chem. 2008. PMID: 18588279

10

Design, synthesis and biological evaluation of novel thiazol-2-yl benzamide derivatives as glucokinase activators.

Charaya N, Pandita D, Grewal AS, Lather V. Charaya N, et al. Comput Biol Chem. 2018 Apr;73:221-229. doi: 10.1016/j.compbiolchem.2018.02.018. Epub 2018 Feb 27. Comput Biol Chem. 2018. PMID: 29518630

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