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Items: 1 to 20 of 847

1.

Design, synthesis, and structure-activity relationship studies of 4-quinolinyl- and 9-acrydinylhydrazones as potent antimalarial agents.

Fattorusso C, Campiani G, Kukreja G, Persico M, Butini S, Romano MP, Altarelli M, Ros S, Brindisi M, Savini L, Novellino E, Nacci V, Fattorusso E, Parapini S, Basilico N, Taramelli D, Yardley V, Croft S, Borriello M, Gemma S.

J Med Chem. 2008 Mar 13;51(5):1333-43. doi: 10.1021/jm7012375. Epub 2008 Feb 16.

PMID:
18278859
2.

Synthesis of N1-arylidene-N2-quinolyl- and N2-acrydinylhydrazones as potent antimalarial agents active against CQ-resistant P. falciparum strains.

Gemma S, Kukreja G, Fattorusso C, Persico M, Romano MP, Altarelli M, Savini L, Campiani G, Fattorusso E, Basilico N, Taramelli D, Yardley V, Butini S.

Bioorg Med Chem Lett. 2006 Oct 15;16(20):5384-8. Epub 2006 Aug 4.

PMID:
16890433
3.

Synthesis and in vitro and in vivo antimalarial activity of new 4-anilinoquinolines.

Delarue S, Girault S, Maes L, Debreu-Fontaine MA, Labaeïd M, Grellier P, Sergheraert C.

J Med Chem. 2001 Aug 16;44(17):2827-33.

PMID:
11495593
4.

Synthesis and in vitro and in vivo antimalarial activity of N1-(7-chloro-4-quinolyl)-1,4-bis(3-aminopropyl)piperazine derivatives.

Ryckebusch A, Deprez-Poulain R, Maes L, Debreu-Fontaine MA, Mouray E, Grellier P, Sergheraert C.

J Med Chem. 2003 Feb 13;46(4):542-57.

PMID:
12570376
5.

Synthesis of some cryptolepine analogues, assessment of their antimalarial and cytotoxic activities, and consideration of their antimalarial mode of action.

Onyeibor O, Croft SL, Dodson HI, Feiz-Haddad M, Kendrick H, Millington NJ, Parapini S, Phillips RM, Seville S, Shnyder SD, Taramelli D, Wright CW.

J Med Chem. 2005 Apr 7;48(7):2701-9.

PMID:
15801861
6.

Probing the role of the covalent linkage of ferrocene into a chloroquine template.

Biot C, Daher W, Ndiaye CM, Melnyk P, Pradines B, Chavain N, Pellet A, Fraisse L, Pelinski L, Jarry C, Brocard J, Khalife J, Forfar-Bares I, Dive D.

J Med Chem. 2006 Jul 27;49(15):4707-14.

PMID:
16854077
7.

4-anilinoquinoline triazines: a novel class of hybrid antimalarial agents.

Kumar A, Srivastava K, Kumar SR, Siddiqi MI, Puri SK, Sexana JK, Chauhan PM.

Eur J Med Chem. 2011 Feb;46(2):676-90. doi: 10.1016/j.ejmech.2010.12.003. Epub 2010 Dec 9.

PMID:
21194812
8.

Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline.

Delarue-Cochin S, Grellier P, Maes L, Mouray E, Sergheraert C, Melnyk P.

Eur J Med Chem. 2008 Oct;43(10):2045-55. doi: 10.1016/j.ejmech.2007.11.003. Epub 2007 Nov 19.

PMID:
18226428
9.

A prodrug form of a Plasmodium falciparum glutathione reductase inhibitor conjugated with a 4-anilinoquinoline.

Davioud-Charvet E, Delarue S, Biot C, Schwöbel B, Boehme CC, Müssigbrodt A, Maes L, Sergheraert C, Grellier P, Schirmer RH, Becker K.

J Med Chem. 2001 Nov 22;44(24):4268-76.

PMID:
11708927
10.

In vitro efficiency of new acridyl derivatives against Plasmodium falciparum.

Guetzoyan L, Ramiandrasoa F, Dorizon H, Desprez C, Bridoux A, Rogier C, Pradines B, Perrée-Fauvet M.

Bioorg Med Chem. 2007 May 1;15(9):3278-89. Epub 2007 Feb 16.

PMID:
17339112
11.

Synthesis and evaluation of sulfonylurea derivatives as novel antimalarials.

León C, Rodrigues J, Gamboa de Domínguez N, Charris J, Gut J, Rosenthal PJ, Domínguez JN.

Eur J Med Chem. 2007 Jun;42(6):735-42. Epub 2007 Jan 14.

PMID:
17321641
12.

Antimalarial dual drugs based on potent inhibitors of glutathione reductase from Plasmodium falciparum.

Friebolin W, Jannack B, Wenzel N, Furrer J, Oeser T, Sanchez CP, Lanzer M, Yardley V, Becker K, Davioud-Charvet E.

J Med Chem. 2008 Mar 13;51(5):1260-77. doi: 10.1021/jm7009292. Epub 2008 Feb 9.

PMID:
18260613
13.

Synthesis and antimalarial evaluation of novel isocryptolepine derivatives.

Whittell LR, Batty KT, Wong RP, Bolitho EM, Fox SA, Davis TM, Murray PE.

Bioorg Med Chem. 2011 Dec 15;19(24):7519-25. doi: 10.1016/j.bmc.2011.10.037. Epub 2011 Oct 20.

PMID:
22055713
14.

Ligand-based virtual screening and in silico design of new antimalarial compounds using nonstochastic and stochastic total and atom-type quadratic maps.

Marrero-Ponce Y, Iyarreta-Veitía M, Montero-Torres A, Romero-Zaldivar C, Brandt CA, Avila PE, Kirchgatter K, Machado Y.

J Chem Inf Model. 2005 Jul-Aug;45(4):1082-100.

PMID:
16045304
15.

Clotrimazole scaffold as an innovative pharmacophore towards potent antimalarial agents: design, synthesis, and biological and structure-activity relationship studies.

Gemma S, Campiani G, Butini S, Kukreja G, Coccone SS, Joshi BP, Persico M, Nacci V, Fiorini I, Novellino E, Fattorusso E, Taglialatela-Scafati O, Savini L, Taramelli D, Basilico N, Parapini S, Morace G, Yardley V, Croft S, Coletta M, Marini S, Fattorusso C.

J Med Chem. 2008 Mar 13;51(5):1278-94. doi: 10.1021/jm701247k. Epub 2008 Feb 16.

PMID:
18278860
16.

Bisquinolines. 2. Antimalarial N,N-bis(7-chloroquinolin-4-yl)heteroalkanediamines.

Vennerstrom JL, Ager AL Jr, Dorn A, Andersen SL, Gerena L, Ridley RG, Milhous WK.

J Med Chem. 1998 Oct 22;41(22):4360-4.

PMID:
9784111
17.

Design and synthesis of new antimalarial agents from 4-aminoquinoline.

Solomon VR, Puri SK, Srivastava K, Katti SB.

Bioorg Med Chem. 2005 Mar 15;13(6):2157-65.

PMID:
15727868
18.

Mapping antimalarial pharmacophores as a useful tool for the rapid discovery of drugs effective in vivo: design, construction, characterization, and pharmacology of metaquine.

Dascombe MJ, Drew MG, Morris H, Wilairat P, Auparakkitanon S, Moule WA, Alizadeh-Shekalgourabi S, Evans PG, Lloyd M, Dyas AM, Carr P, Ismail FM.

J Med Chem. 2005 Aug 25;48(17):5423-36.

PMID:
16107142
19.
20.
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