Similar articles for PMID: 17826100

Year	Number of Results
1980	1
1982	1
1996	1
1997	2
1998	1
2000	3
2001	3
2002	1
2003	1
2004	6
2005	1
2006	6
2007	3
2008	4
2009	5
2010	5
2011	3
2012	6
2013	2
2014	4
2015	6
2016	2
2019	2
2024	0

1

Discovery of platelet-type 12-human lipoxygenase selective inhibitors by high-throughput screening of structurally diverse libraries.

Deschamps JD, Gautschi JT, Whitman S, Johnson TA, Gassner NC, Crews P, Holman TR. Deschamps JD, et al. Bioorg Med Chem. 2007 Nov 15;15(22):6900-8. doi: 10.1016/j.bmc.2007.08.015. Epub 2007 Aug 22. Bioorg Med Chem. 2007. PMID: 17826100 Free PMC article.

2

Structure-activity relationship studies of flavonoids as potent inhibitors of human platelet 12-hLO, reticulocyte 15-hLO-1, and prostate epithelial 15-hLO-2.

Vasquez-Martinez Y, Ohri RV, Kenyon V, Holman TR, Sepúlveda-Boza S. Vasquez-Martinez Y, et al. Bioorg Med Chem. 2007 Dec 1;15(23):7408-25. doi: 10.1016/j.bmc.2007.07.036. Epub 2007 Aug 22. Bioorg Med Chem. 2007. PMID: 17869117 Free PMC article.

3

Novel human lipoxygenase inhibitors discovered using virtual screening with homology models.

Kenyon V, Chorny I, Carvajal WJ, Holman TR, Jacobson MP. Kenyon V, et al. J Med Chem. 2006 Feb 23;49(4):1356-63. doi: 10.1021/jm050639j. J Med Chem. 2006. PMID: 16480270

4

Discovery of potent and selective inhibitors of human reticulocyte 15-lipoxygenase-1.

Rai G, Kenyon V, Jadhav A, Schultz L, Armstrong M, Jameson JB, Hoobler E, Leister W, Simeonov A, Holman TR, Maloney DJ. Rai G, et al. J Med Chem. 2010 Oct 28;53(20):7392-404. doi: 10.1021/jm1008852. J Med Chem. 2010. PMID: 20866075 Free PMC article.

5

Baicalein is a potent in vitro inhibitor against both reticulocyte 15-human and platelet 12-human lipoxygenases.

Deschamps JD, Kenyon VA, Holman TR. Deschamps JD, et al. Bioorg Med Chem. 2006 Jun 15;14(12):4295-301. doi: 10.1016/j.bmc.2006.01.057. Epub 2006 Feb 24. Bioorg Med Chem. 2006. PMID: 16500106

6

Redox inactivation of human 15-lipoxygenase by marine-derived meroditerpenes and synthetic chromanes: archetypes for a unique class of selective and recyclable inhibitors.

Cichewicz RH, Kenyon VA, Whitman S, Morales NM, Arguello JF, Holman TR, Crews P. Cichewicz RH, et al. J Am Chem Soc. 2004 Nov 17;126(45):14910-20. doi: 10.1021/ja046082z. J Am Chem Soc. 2004. PMID: 15535718

7

Selective Small Molecule Inhibitors of 12-Human Lipoxygenase (12-hLO).

Rai G, Jadhav A, Schultz L, Kenyon V, Leister W, Simeonov A, Holman TR, Maloney DJ. Rai G, et al. 2009 Nov 30 [updated 2011 Mar 25]. In: Probe Reports from the NIH Molecular Libraries Program [Internet]. Bethesda (MD): National Center for Biotechnology Information (US); 2010–. 2009 Nov 30 [updated 2011 Mar 25]. In: Probe Reports from the NIH Molecular Libraries Program [Internet]. Bethesda (MD): National Center for Biotechnology Information (US); 2010–. PMID: 21735604 Free Books & Documents. Review.

8

Identification of 6-benzyloxysalicylates as a novel class of inhibitors of 15-lipoxygenase-1.

Eleftheriadis N, Thee S, te Biesebeek J, van der Wouden P, Baas BJ, Dekker FJ. Eleftheriadis N, et al. Eur J Med Chem. 2015 Apr 13;94:265-75. doi: 10.1016/j.ejmech.2015.03.007. Epub 2015 Mar 5. Eur J Med Chem. 2015. PMID: 25771032

9

2-arylalkyl-substituted anthracenones as inhibitors of 12-lipoxygenase enzymes. 1. Structure-activity relationships of the terminal aryl ring.

Müller K, Altmann R, Prinz H. Müller K, et al. Eur J Med Chem. 2001 Jun;36(6):569-75. doi: 10.1016/s0223-5234(01)01248-x. Eur J Med Chem. 2001. PMID: 11525848

10

Discovery of potent and selective inhibitors of human platelet-type 12- lipoxygenase.

Kenyon V, Rai G, Jadhav A, Schultz L, Armstrong M, Jameson JB 2nd, Perry S, Joshi N, Bougie JM, Leister W, Taylor-Fishwick DA, Nadler JL, Holinstat M, Simeonov A, Maloney DJ, Holman TR. Kenyon V, et al. J Med Chem. 2011 Aug 11;54(15):5485-97. doi: 10.1021/jm2005089. Epub 2011 Jul 8. J Med Chem. 2011. PMID: 21739938 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Results by year

Text availability

Article attribute

Article type

Publication date

62 results

Results by year