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Results: 1 to 20 of 100

1.

Virtual and biomolecular screening converge on a selective agonist for GPR30.

Bologa CG, Revankar CM, Young SM, Edwards BS, Arterburn JB, Kiselyov AS, Parker MA, Tkachenko SE, Savchuck NP, Sklar LA, Oprea TI, Prossnitz ER.

Nat Chem Biol. 2006 Apr;2(4):207-12. Epub 2006 Mar 5.

PMID:
16520733
[PubMed - indexed for MEDLINE]
2.

Synthetic estrogen derivatives demonstrate the functionality of intracellular GPR30.

Revankar CM, Mitchell HD, Field AS, Burai R, Corona C, Ramesh C, Sklar LA, Arterburn JB, Prossnitz ER.

ACS Chem Biol. 2007 Aug 17;2(8):536-44. Epub 2007 Jul 27.

PMID:
17655271
[PubMed - indexed for MEDLINE]
3.

A transmembrane intracellular estrogen receptor mediates rapid cell signaling.

Revankar CM, Cimino DF, Sklar LA, Arterburn JB, Prossnitz ER.

Science. 2005 Mar 11;307(5715):1625-30. Epub 2005 Feb 10.

PMID:
15705806
[PubMed - indexed for MEDLINE]
Free Article
4.

GPR30: a novel therapeutic target in estrogen-related disease.

Prossnitz ER, Sklar LA, Oprea TI, Arterburn JB.

Trends Pharmacol Sci. 2008 Mar;29(3):116-23. doi: 10.1016/j.tips.2008.01.001. Epub 2008 Feb 11.

PMID:
18262661
[PubMed - indexed for MEDLINE]
5.

G protein-coupled receptor 30 (GPR30) mediates gene expression changes and growth response to 17beta-estradiol and selective GPR30 ligand G-1 in ovarian cancer cells.

Albanito L, Madeo A, Lappano R, Vivacqua A, Rago V, Carpino A, Oprea TI, Prossnitz ER, Musti AM, Andò S, Maggiolini M.

Cancer Res. 2007 Feb 15;67(4):1859-66.

PMID:
17308128
[PubMed - indexed for MEDLINE]
Free Article
6.

A new membrane G protein-coupled receptor (GPR30) is involved in the cardiac effects of 17beta-estradiol in the male rat.

Filice E, Recchia AG, Pellegrino D, Angelone T, Maggiolini M, Cerra MC.

J Physiol Pharmacol. 2009 Dec;60(4):3-10.

PMID:
20065491
[PubMed - indexed for MEDLINE]
Free Article
7.

GPR30: a seven-transmembrane-spanning estrogen receptor that triggers EGF release.

Filardo EJ, Thomas P.

Trends Endocrinol Metab. 2005 Oct;16(8):362-7. Review.

PMID:
16125968
[PubMed - indexed for MEDLINE]
8.

Binding and activation of the seven-transmembrane estrogen receptor GPR30 by environmental estrogens: a potential novel mechanism of endocrine disruption.

Thomas P, Dong J.

J Steroid Biochem Mol Biol. 2006 Dec;102(1-5):175-9. Epub 2006 Nov 7.

PMID:
17088055
[PubMed - indexed for MEDLINE]
9.

In vivo effects of a GPR30 antagonist.

Dennis MK, Burai R, Ramesh C, Petrie WK, Alcon SN, Nayak TK, Bologa CG, Leitao A, Brailoiu E, Deliu E, Dun NJ, Sklar LA, Hathaway HJ, Arterburn JB, Oprea TI, Prossnitz ER.

Nat Chem Biol. 2009 Jun;5(6):421-7. doi: 10.1038/nchembio.168.

PMID:
19430488
[PubMed - indexed for MEDLINE]
Free PMC Article
10.

Identification of ligands with bicyclic scaffolds provides insights into mechanisms of estrogen receptor subtype selectivity.

Hsieh RW, Rajan SS, Sharma SK, Guo Y, DeSombre ER, Mrksich M, Greene GL.

J Biol Chem. 2006 Jun 30;281(26):17909-19. Epub 2006 Apr 28.

PMID:
16648639
[PubMed - indexed for MEDLINE]
Free Article
11.

G protein-coupled receptor 30 localizes to the endoplasmic reticulum and is not activated by estradiol.

Otto C, Rohde-Schulz B, Schwarz G, Fuchs I, Klewer M, Brittain D, Langer G, Bader B, Prelle K, Nubbemeyer R, Fritzemeier KH.

Endocrinology. 2008 Oct;149(10):4846-56. doi: 10.1210/en.2008-0269. Epub 2008 Jun 19.

PMID:
18566127
[PubMed - indexed for MEDLINE]
12.

Estrogenic G protein-coupled receptor 30 signaling is involved in regulation of endometrial carcinoma by promoting proliferation, invasion potential, and interleukin-6 secretion via the MEK/ERK mitogen-activated protein kinase pathway.

He YY, Cai B, Yang YX, Liu XL, Wan XP.

Cancer Sci. 2009 Jun;100(6):1051-61. doi: 10.1111/j.1349-7006.2009.01148.x. Epub 2009 Mar 9.

PMID:
19432902
[PubMed - indexed for MEDLINE]
13.

Differential effects of 17beta-estradiol on function and expression of estrogen receptor alpha, estrogen receptor beta, and GPR30 in arteries and veins of patients with atherosclerosis.

Haas E, Meyer MR, Schurr U, Bhattacharya I, Minotti R, Nguyen HH, Heigl A, Lachat M, Genoni M, Barton M.

Hypertension. 2007 Jun;49(6):1358-63. Epub 2007 Apr 23.

PMID:
17452498
[PubMed - indexed for MEDLINE]
Free Article
14.

Involvement of estrogen receptor variant ER-alpha36, not GPR30, in nongenomic estrogen signaling.

Kang L, Zhang X, Xie Y, Tu Y, Wang D, Liu Z, Wang ZY.

Mol Endocrinol. 2010 Apr;24(4):709-21. doi: 10.1210/me.2009-0317. Epub 2010 Mar 2.

PMID:
20197310
[PubMed - indexed for MEDLINE]
Free PMC Article
15.

What does an orphan G-protein-coupled receptor have to do with estrogen?

Rae JM, Johnson MD.

Breast Cancer Res. 2005;7(6):243-4. Epub 2005 Sep 29.

PMID:
16280047
[PubMed - indexed for MEDLINE]
Free PMC Article
16.

Beneficial role of the GPR30 agonist G-1 in an animal model of multiple sclerosis.

Blasko E, Haskell CA, Leung S, Gualtieri G, Halks-Miller M, Mahmoudi M, Dennis MK, Prossnitz ER, Karpus WJ, Horuk R.

J Neuroimmunol. 2009 Sep 29;214(1-2):67-77. doi: 10.1016/j.jneuroim.2009.06.023. Epub 2009 Aug 6.

PMID:
19664827
[PubMed - indexed for MEDLINE]
Free PMC Article
17.

Evaluation of ligand selectivity using reporter cell lines stably expressing estrogen receptor alpha or beta.

Escande A, Pillon A, Servant N, Cravedi JP, Larrea F, Muhn P, Nicolas JC, Cavaillès V, Balaguer P.

Biochem Pharmacol. 2006 May 14;71(10):1459-69. Epub 2006 Mar 22.

PMID:
16554039
[PubMed - indexed for MEDLINE]
18.

A critical review of fundamental controversies in the field of GPR30 research.

Langer G, Bader B, Meoli L, Isensee J, Delbeck M, Noppinger PR, Otto C.

Steroids. 2010 Aug-Sep;75(8-9):603-10. doi: 10.1016/j.steroids.2009.12.006. Epub 2009 Dec 23. Review.

PMID:
20034504
[PubMed - indexed for MEDLINE]
19.
20.

The unfolding stories of GPR30, a new membrane-bound estrogen receptor.

Maggiolini M, Picard D.

J Endocrinol. 2010 Feb;204(2):105-14. doi: 10.1677/JOE-09-0242. Epub 2009 Sep 18. Review.

PMID:
19767412
[PubMed - indexed for MEDLINE]
Free Article

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