Format
Items per page
Sort by

Send to:

Choose Destination

Results: 1 to 20 of 259

1.

Synthesis, characterization, and first successful monkey imaging studies of metabotropic glutamate receptor subtype 5 (mGluR5) PET radiotracers.

Hamill TG, Krause S, Ryan C, Bonnefous C, Govek S, Seiders TJ, Cosford ND, Roppe J, Kamenecka T, Patel S, Gibson RE, Sanabria S, Riffel K, Eng W, King C, Yang X, Green MD, O'Malley SS, Hargreaves R, Burns HD.

Synapse. 2005 Jun 15;56(4):205-16.

PMID:
15803497
[PubMed - indexed for MEDLINE]
2.

Screening cascade and development of potential Positron Emission Tomography radiotracers for mGluR5: in vitro and in vivo characterization.

Patel S, Ndubizu O, Hamill T, Chaudhary A, Burns HD, Hargreaves R, Gibson RE.

Mol Imaging Biol. 2005 Jul-Aug;7(4):314-23.

PMID:
16080024
[PubMed - indexed for MEDLINE]
3.

Synthesis, characterization, and monkey PET studies of [¹⁸F]MK-1312, a PET tracer for quantification of mGluR1 receptor occupancy by MK-5435.

Hostetler ED, Eng W, Joshi AD, Sanabria-Bohórquez S, Kawamoto H, Ito S, O'Malley S, Krause S, Ryan C, Patel S, Williams M, Riffel K, Suzuki G, Ozaki S, Ohta H, Cook J, Burns HD, Hargreaves R.

Synapse. 2011 Feb;65(2):125-35. doi: 10.1002/syn.20826.

PMID:
20524178
[PubMed - indexed for MEDLINE]
4.

Species differences in mGluR5 binding sites in mammalian central nervous system determined using in vitro binding with [18F]F-PEB.

Patel S, Hamill TG, Connolly B, Jagoda E, Li W, Gibson RE.

Nucl Med Biol. 2007 Nov;34(8):1009-17. Epub 2007 Sep 19.

PMID:
17998106
[PubMed - indexed for MEDLINE]
5.

Inverse agonist histamine H3 receptor PET tracers labelled with carbon-11 or fluorine-18.

Hamill TG, Sato N, Jitsuoka M, Tokita S, Sanabria S, Eng W, Ryan C, Krause S, Takenaga N, Patel S, Zeng Z, Williams D Jr, Sur C, Hargreaves R, Burns HD.

Synapse. 2009 Dec;63(12):1122-32. doi: 10.1002/syn.20689.

PMID:
19670309
[PubMed - indexed for MEDLINE]
6.

In vitro and in vivo evaluation of [18F]-FDEGPECO as a PET tracer for imaging the metabotropic glutamate receptor subtype 5 (mGluR5).

Wanger-Baumann CA, Mu L, Honer M, Belli S, Alf MF, Schubiger PA, Krämer SD, Ametamey SM.

Neuroimage. 2011 Jun 1;56(3):984-91. doi: 10.1016/j.neuroimage.2011.03.024. Epub 2011 Mar 21.

PMID:
21406237
[PubMed - indexed for MEDLINE]
7.

Radiolabeling and in vitro and in vivo evaluation of [18F]-FE-DABP688 as a PET radioligand for the metabotropic glutamate receptor subtype 5.

Honer M, Stoffel A, Kessler LJ, Schubiger PA, Ametamey SM.

Nucl Med Biol. 2007 Nov;34(8):973-80. Epub 2007 Sep 19.

PMID:
17998101
[PubMed - indexed for MEDLINE]
8.

Synthesis, characterization, and monkey positron emission tomography (PET) studies of [18F]Y1-973, a PET tracer for the neuropeptide Y Y1 receptor.

Hostetler ED, Sanabria-Bohórquez S, Fan H, Zeng Z, Gantert L, Williams M, Miller P, O'Malley S, Kameda M, Ando M, Sato N, Ozaki S, Tokita S, Ohta H, Williams D, Sur C, Cook JJ, Burns HD, Hargreaves R.

Neuroimage. 2011 Feb 14;54(4):2635-42. doi: 10.1016/j.neuroimage.2010.11.014. Epub 2010 Nov 13.

PMID:
21078401
[PubMed - indexed for MEDLINE]
9.

Radiosynthesis and preclinical evaluation of 11C-ABP688 as a probe for imaging the metabotropic glutamate receptor subtype 5.

Ametamey SM, Kessler LJ, Honer M, Wyss MT, Buck A, Hintermann S, Auberson YP, Gasparini F, Schubiger PA.

J Nucl Med. 2006 Apr;47(4):698-705.

PMID:
16595505
[PubMed - indexed for MEDLINE]
Free Article
10.

Synthesis, radiolabeling, in vitro and in vivo evaluation of [18F]-FPECMO as a positron emission tomography radioligand for imaging the metabotropic glutamate receptor subtype 5.

Lucatelli C, Honer M, Salazar JF, Ross TL, Schubiger PA, Ametamey SM.

Nucl Med Biol. 2009 Aug;36(6):613-22. doi: 10.1016/j.nucmedbio.2009.03.005.

PMID:
19647167
[PubMed - indexed for MEDLINE]
11.

Methoxyphenylethynyl, methoxypyridylethynyl and phenylethynyl derivatives of pyridine: synthesis, radiolabeling and evaluation of new PET ligands for metabotropic glutamate subtype 5 receptors.

Yu M, Tueckmantel W, Wang X, Zhu A, Kozikowski AP, Brownell AL.

Nucl Med Biol. 2005 Aug;32(6):631-40.

PMID:
16026710
[PubMed - indexed for MEDLINE]
12.

Synthesis and simple 18F-labeling of 3-fluoro-5-(2-(2-(fluoromethyl)thiazol-4-yl)ethynyl)benzonitrile as a high affinity radioligand for imaging monkey brain metabotropic glutamate subtype-5 receptors with positron emission tomography.

Siméon FG, Brown AK, Zoghbi SS, Patterson VM, Innis RB, Pike VW.

J Med Chem. 2007 Jul 12;50(14):3256-66. Epub 2007 Jun 16.

PMID:
17571866
[PubMed - indexed for MEDLINE]
13.

PET imaging studies in rhesus monkey with the cannabinoid-1 (CB1) receptor ligand [11C]CB-119.

Hamill TG, Lin LS, Hagmann W, Liu P, Jewell J, Sanabria S, Eng W, Ryan C, Fong TM, Connolly B, Vanko A, Hargreaves R, Goulet MT, Burns HD.

Mol Imaging Biol. 2009 Jul-Aug;11(4):246-52. doi: 10.1007/s11307-008-0194-8. Epub 2009 Jan 7.

PMID:
19130142
[PubMed - indexed for MEDLINE]
14.

Human PET studies of metabotropic glutamate receptor subtype 5 with 11C-ABP688.

Ametamey SM, Treyer V, Streffer J, Wyss MT, Schmidt M, Blagoev M, Hintermann S, Auberson Y, Gasparini F, Fischer UC, Buck A.

J Nucl Med. 2007 Feb;48(2):247-52.

PMID:
17268022
[PubMed - indexed for MEDLINE]
Free Article
15.

Synthesis and preliminary biological evaluation of 3-[(18)F]fluoro-5-(2-pyridinylethynyl)benzonitrile as a PET radiotracer for imaging metabotropic glutamate receptor subtype 5.

Wang JQ, Tueckmantel W, Zhu A, Pellegrino D, Brownell AL.

Synapse. 2007 Dec;61(12):951-61.

PMID:
17787003
[PubMed - indexed for MEDLINE]
16.

Characterization of 1-(2-[18F] fluoro-3-pyridyl)-4-(2-isopropyl-1-oxo- isoindoline-5-yl)-5-methyl-1H-1,2,3-triazole, a PET ligand for imaging the metabotropic glutamate receptor type 1 in rat and monkey brains.

Fujinaga M, Maeda J, Yui J, Hatori A, Yamasaki T, Kawamura K, Kumata K, Yoshida Y, Nagai Y, Higuchi M, Suhara T, Fukumura T, Zhang MR.

J Neurochem. 2012 Apr;121(1):115-24. doi: 10.1111/j.1471-4159.2011.07348.x. Epub 2011 Jul 1.

PMID:
21668889
[PubMed - indexed for MEDLINE]
18.

Synthesis and characterization of two PET radioligands for the metabotropic glutamate 1 (mGlu1) receptor.

Huang Y, Narendran R, Bischoff F, Guo N, Bae SA, Hwang DR, Lesage AS, Laruelle M.

Synapse. 2012 Dec;66(12):1002-14. doi: 10.1002/syn.21606. Epub 2012 Sep 29. Erratum in: Synapse. 2013 Feb;67(2):109.

PMID:
22927303
[PubMed - indexed for MEDLINE]
19.

Syntheses and pharmacological characterization of novel thiazole derivatives as potential mGluR5 PET ligands.

Baumann CA, Mu L, Wertli N, Krämer SD, Honer M, Schubiger PA, Ametamey SM.

Bioorg Med Chem. 2010 Aug 15;18(16):6044-54. doi: 10.1016/j.bmc.2010.06.070. Epub 2010 Jun 25.

PMID:
20634080
[PubMed - indexed for MEDLINE]
20.

Synthesis and biologic evaluation of a novel serotonin 5-HT1A receptor radioligand, 18F-labeled mefway, in rodents and imaging by PET in a nonhuman primate.

Saigal N, Pichika R, Easwaramoorthy B, Collins D, Christian BT, Shi B, Narayanan TK, Potkin SG, Mukherjee J.

J Nucl Med. 2006 Oct;47(10):1697-706.

PMID:
17015907
[PubMed - indexed for MEDLINE]
Free Article
Format
Items per page
Sort by

Send to:

Choose Destination

Supplemental Content

Write to the Help Desk