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Items: 1 to 20 of 136

1.

Synthesis and biochemical evaluation of novel and potent inhibitors of the enzyme oestrone sulphatase (ES).

Ahmed S, James K, Owen CP, Patel CK.

J Steroid Biochem Mol Biol. 2002 Apr;80(4-5):419-27.

PMID:
11983489
3.

Hydrophobicity, a physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES).

Ahmed S, James K, Owen CP, Patel CK, Patel M.

Bioorg Med Chem Lett. 2001 Sep 17;11(18):2525-8.

PMID:
11549461
4.

Novel inhibitors of the enzyme estrone sulfatase (ES).

Ahmed S, James K, Owen CP, Patel CK, Patel M.

Bioorg Med Chem Lett. 2001 Mar 26;11(6):841-4.

PMID:
11277533
5.

Potent active site-directed inhibition of steroid sulphatase by tricyclic coumarin-based sulphamates.

Woo LL, Purohit A, Malini B, Reed MJ, Potter BV.

Chem Biol. 2000 Oct;7(10):773-91.

6.

Evidence for the mechanism of the irreversible inhibition of oestrone sulphatase (ES) by aminosulphonate based compounds.

Ahmed S, Owen CP, James K, Patel CK, Sampson L.

J Steroid Biochem Mol Biol. 2002 Apr;80(4-5):429-40.

PMID:
11983490
7.

Design, synthesis and biochemical evaluation of AC ring mimics as novel inhibitors of the enzyme estrone sulfatase (ES).

Ahmed S, James K, Owen CP.

J Steroid Biochem Mol Biol. 2002 Nov;82(4-5):425-35.

PMID:
12589950
9.
10.

Steroidal and nonsteroidal sulfamates as potent inhibitors of steroid sulfatase.

Woo LW, Howarth NM, Purohit A, Hejaz HA, Reed MJ, Potter BV.

J Med Chem. 1998 Mar 26;41(7):1068-83.

PMID:
9544207
11.

Determination and use of a transition state for the enzyme estrone sulfatase (ES) from a proposed reaction mechanism.

Ahmed S, James K, Owen CP, Patel CK, Patel MB.

Bioorg Med Chem Lett. 2001 Dec 3;11(23):3001-5.

PMID:
11714597
12.

Design, synthesis and biochemical evaluation of AC ring mimics as novel inhibitors of the enzyme estrone sulfatase (ES).

Ahmed S, James K, Owen CP, Patel CK.

Bioorg Med Chem Lett. 2002 May 20;12(10):1343-6.

PMID:
11992773
13.

2-difluoromethyloestrone 3-O-sulphamate, a highly potent steroid sulphatase inhibitor.

Reed JE, Woo LW, Robinson JJ, Leblond B, Leese MP, Purohit A, Reed MJ, Potter BV.

Biochem Biophys Res Commun. 2004 Apr 23;317(1):169-75.

PMID:
15047163
14.

Measurement of oestrone sulphatase activity in white blood cells to monitor in vivo inhibition of steroid sulphatase activity by oestrone-3-O-sulphamate.

Purohit A, Froome VA, Wang DY, Potter BV, Reed MJ.

J Steroid Biochem Mol Biol. 1997 May;62(1):45-51.

PMID:
9366497
15.

The development of A-ring modified analogues of oestrone-3-O-sulphamate as potent steroid sulphatase inhibitors with reduced oestrogenicity.

Purohit A, Vernon KA, Hummelinck AE, Woo LW, Hejaz HA, Potter BV, Reed MJ.

J Steroid Biochem Mol Biol. 1998 Mar;64(5-6):269-75.

PMID:
9618028
16.
17.
18.

In vivo inhibition of oestrone sulphatase and dehydroepiandrosterone sulphatase by oestrone-3-O-sulphamate.

Purohit A, Williams GJ, Roberts CJ, Potter BV, Reed MJ.

Int J Cancer. 1995 Sep 27;63(1):106-11.

PMID:
7558436
19.

Structure-activity relationship study of steroidal and nonsteroidal inhibitors of the enzyme estrone sulfatase.

Ahmed S, James K, Sampson L, Mastri C.

Biochem Biophys Res Commun. 1999 Jan 27;254(3):811-5.

PMID:
9920822
20.

Acid dissociation constant, a potential physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES).

Ahmed S, Owen CP, James K, Patel CK, Patel M.

Bioorg Med Chem Lett. 2001 Apr 9;11(7):899-902.

PMID:
11294387
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