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Results: 1 to 20 of 126

1.

Derivation of a possible transition-state for the reaction catalysed by the enzyme estrone Sulfatase (ES).

Ahmed S, James K.

Bioorg Med Chem Lett. 1999 Jun 21;9(12):1645-50.

PMID:
10397493
[PubMed - indexed for MEDLINE]
2.

Determination and use of a transition state for the enzyme estrone sulfatase (ES) from a proposed reaction mechanism.

Ahmed S, James K, Owen CP, Patel CK, Patel MB.

Bioorg Med Chem Lett. 2001 Dec 3;11(23):3001-5.

PMID:
11714597
[PubMed - indexed for MEDLINE]
3.
4.
5.

Estrone sulfatase: probing structural requirements for substrate and inhibitor recognition.

Anderson C, Freeman J, Lucas LH, Farley M, Dalhoumi H, Widlanski TS.

Biochemistry. 1997 Mar 4;36(9):2586-94. Erratum in: Biochemistry 1997 Sep 23;36(38):11542.

PMID:
9054565
[PubMed - indexed for MEDLINE]
6.

Structure-activity relationship study of steroidal and nonsteroidal inhibitors of the enzyme estrone sulfatase.

Ahmed S, James K, Sampson L, Mastri C.

Biochem Biophys Res Commun. 1999 Jan 27;254(3):811-5.

PMID:
9920822
[PubMed - indexed for MEDLINE]
7.

Estrone 3-sulfate mimics, inhibitors of estrone sulfatase activity: homology model construction and docking studies.

Howarth NM, Purohit A, Robinson JJ, Vicker N, Reed MJ, Potter BV.

Biochemistry. 2002 Dec 17;41(50):14801-14.

PMID:
12475228
[PubMed - indexed for MEDLINE]
9.

Synthesis and biochemical evaluation of novel and potent inhibitors of the enzyme oestrone sulphatase (ES).

Ahmed S, James K, Owen CP, Patel CK.

J Steroid Biochem Mol Biol. 2002 Apr;80(4-5):419-27.

PMID:
11983489
[PubMed - indexed for MEDLINE]
10.

Synthesis and sulfatase inhibitory activities of non-steroidal estrone sulfatase inhibitors.

Li PK, Milano S, Kluth L, Rhodes ME.

J Steroid Biochem Mol Biol. 1996 Sep;59(1):41-8.

PMID:
9009236
[PubMed - indexed for MEDLINE]
11.

Hydrophobicity, a physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES).

Ahmed S, James K, Owen CP, Patel CK, Patel M.

Bioorg Med Chem Lett. 2001 Sep 17;11(18):2525-8.

PMID:
11549461
[PubMed - indexed for MEDLINE]
12.

Design, synthesis and biochemical evaluation of AC ring mimics as novel inhibitors of the enzyme estrone sulfatase (ES).

Ahmed S, James K, Owen CP, Patel CK.

Bioorg Med Chem Lett. 2002 May 20;12(10):1343-6.

PMID:
11992773
[PubMed - indexed for MEDLINE]
13.

Novel inhibitors of the enzyme estrone sulfatase (ES).

Ahmed S, James K, Owen CP, Patel CK, Patel M.

Bioorg Med Chem Lett. 2001 Mar 26;11(6):841-4.

PMID:
11277533
[PubMed - indexed for MEDLINE]
14.

Three-dimensional structures of sulfatases.

Ghosh D.

Methods Enzymol. 2005;400:273-93. Review.

PMID:
16399355
[PubMed - indexed for MEDLINE]
15.

Design, synthesis and biochemical evaluation of AC ring mimics as novel inhibitors of the enzyme estrone sulfatase (ES).

Ahmed S, James K, Owen CP.

J Steroid Biochem Mol Biol. 2002 Nov;82(4-5):425-35.

PMID:
12589950
[PubMed - indexed for MEDLINE]
16.

Estrone sulfonates as inhibitors of estrone sulfatase.

Howarth NM, Purohit A, Reed MJ, Potter BV.

Steroids. 1997 Apr;62(4):346-50.

PMID:
9090794
[PubMed - indexed for MEDLINE]
17.

17 alpha-alkyl- or 17 alpha-substituted benzyl-17 beta-estradiols: a new family of estrone-sulfatase inhibitors.

Poirier D, Boivin RP.

Bioorg Med Chem Lett. 1998 Jul 21;8(14):1891-6.

PMID:
9873454
[PubMed - indexed for MEDLINE]
18.

Inhibition of estrone sulfatase (ES) by alkyl and cycloalkyl ester derivatives of 4-[(aminosulfonyl)oxy] benzoic acid.

Patel CK, Owen CP, Ahmed S.

Bioorg Med Chem Lett. 2004 Feb 9;14(3):605-9.

PMID:
14741252
[PubMed - indexed for MEDLINE]
19.

Docking studies of sulphamate inhibitors of estrone sulphatase in human carbonic anhydrase II.

Vicker N, Ho Y, Robinson J, Woo LL, Purohit A, Reed MJ, Potter BV.

Bioorg Med Chem Lett. 2003 Mar 10;13(5):863-5.

PMID:
12617909
[PubMed - indexed for MEDLINE]
20.

Strong inhibition of estrone-3-sulfatase activity by pregnenolone 16alpha-carbonitrile but not by several analogs lacking a 16alpha-nitrile group.

Zhu BT, Kosh JW, Fu J, Cai MX, Xu S, Conney AH.

Steroids. 2000 Sep;65(9):521-7.

PMID:
10978731
[PubMed - indexed for MEDLINE]

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