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Items: 1 to 20 of 82

1.

Molecular basis of agonism and antagonism in the oestrogen receptor.

Brzozowski AM, Pike AC, Dauter Z, Hubbard RE, Bonn T, Engström O, Ohman L, Greene GL, Gustafsson JA, Carlquist M.

Nature. 1997 Oct 16;389(6652):753-8.

PMID:
9338790
2.

Structural aspects of agonism and antagonism in the oestrogen receptor.

Pike AC, Brzozowski AM, Walton J, Hubbard RE, Bonn T, Gustafsson JA, Carlquist M.

Biochem Soc Trans. 2000;28(4):396-400. Review.

PMID:
10961927
3.

Structural insights into the mode of action of a pure antiestrogen.

Pike AC, Brzozowski AM, Walton J, Hubbard RE, Thorsell AG, Li YL, Gustafsson JA, Carlquist M.

Structure. 2001 Feb 7;9(2):145-53.

4.

Structure of the ligand-binding domain of oestrogen receptor beta in the presence of a partial agonist and a full antagonist.

Pike AC, Brzozowski AM, Hubbard RE, Bonn T, Thorsell AG, Engström O, Ljunggren J, Gustafsson JA, Carlquist M.

EMBO J. 1999 Sep 1;18(17):4608-18.

5.

Structural characterization of a subtype-selective ligand reveals a novel mode of estrogen receptor antagonism.

Shiau AK, Barstad D, Radek JT, Meyers MJ, Nettles KW, Katzenellenbogen BS, Katzenellenbogen JA, Agard DA, Greene GL.

Nat Struct Biol. 2002 May;9(5):359-64.

PMID:
11953755
6.

Molecular mechanisms of estrogen action: selective ligands and receptor pharmacology.

Katzenellenbogen BS, Choi I, Delage-Mourroux R, Ediger TR, Martini PG, Montano M, Sun J, Weis K, Katzenellenbogen JA.

J Steroid Biochem Mol Biol. 2000 Nov 30;74(5):279-85. Review.

PMID:
11162936
7.
8.

Novel structural templates for estrogen-receptor ligands and prospects for combinatorial synthesis of estrogens.

Fink BE, Mortensen DS, Stauffer SR, Aron ZD, Katzenellenbogen JA.

Chem Biol. 1999 Apr;6(4):205-19.

9.

Structural insights into the mechanisms of agonism and antagonism in oestrogen receptor isoforms.

Hubbard RE, Pike AC, Brzozowski AM, Walton J, Bonn T, Gustafsson JA, Carlquist M.

Eur J Cancer. 2000 Sep;36 Suppl 4:S17-8.

PMID:
11056300
10.

X-ray crystal structures of the estrogen-related receptor-gamma ligand binding domain in three functional states reveal the molecular basis of small molecule regulation.

Wang L, Zuercher WJ, Consler TG, Lambert MH, Miller AB, Orband-Miller LA, McKee DD, Willson TM, Nolte RT.

J Biol Chem. 2006 Dec 8;281(49):37773-81. Epub 2006 Sep 21.

11.

Molecular determinants of tissue selectivity in estrogen receptor modulators.

Grese TA, Sluka JP, Bryant HU, Cullinan GJ, Glasebrook AL, Jones CD, Matsumoto K, Palkowitz AD, Sato M, Termine JD, Winter MA, Yang NN, Dodge JA.

Proc Natl Acad Sci U S A. 1997 Dec 9;94(25):14105-10.

12.

A structural biologist's view of the oestrogen receptor.

Pike AC, Brzozowski AM, Hubbard RE.

J Steroid Biochem Mol Biol. 2000 Nov 30;74(5):261-8. Review.

PMID:
11162934
13.

Crystal structure of a mutant hERalpha ligand-binding domain reveals key structural features for the mechanism of partial agonism.

Gangloff M, Ruff M, Eiler S, Duclaud S, Wurtz JM, Moras D.

J Biol Chem. 2001 May 4;276(18):15059-65. Epub 2001 Feb 6.

15.
16.

An estrogen receptor basis for raloxifene action in bone.

Bryant HU, Glasebrook AL, Yang NN, Sato M.

J Steroid Biochem Mol Biol. 1999 Apr-Jun;69(1-6):37-44. Review.

PMID:
10418979
17.

Identification of an estrogen response element activated by metabolites of 17beta-estradiol and raloxifene.

Yang NN, Venugopalan M, Hardikar S, Glasebrook A.

Science. 1996 Aug 30;273(5279):1222-5. Erratum in: Science. 1997 Feb 28;275(5304):1249.

PMID:
8703055
18.

The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen.

Shiau AK, Barstad D, Loria PM, Cheng L, Kushner PJ, Agard DA, Greene GL.

Cell. 1998 Dec 23;95(7):927-37.

19.

Novel modes of oestrogen receptor agonism and antagonism by hydroxylated and chlorinated biphenyls, revealed by conformation-specific peptide recognition patterns.

Sumbayev VV, Jensen JK, Hansen JA, Andreasen PA.

Mol Cell Endocrinol. 2008 Jun 11;287(1-2):30-9. doi: 10.1016/j.mce.2008.02.004. Epub 2008 Feb 13.

PMID:
18343567
20.
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