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Results: 1 to 20 of 101

1.

Build/couple/pair strategy for the synthesis of stereochemically diverse macrolactams via head-to-tail cyclization.

Fitzgerald ME, Mulrooney CA, Duvall JR, Wei J, Suh BC, Akella LB, Vrcic A, Marcaurelle LA.

ACS Comb Sci. 2012 Feb 13;14(2):89-96. doi: 10.1021/co200161z. Epub 2012 Jan 17.

PMID:
22252910
[PubMed - indexed for MEDLINE]
Free PMC Article
2.

Synthesis of a stereochemically diverse library of medium-sized lactams and sultams via S(N)Ar cycloetherification.

Gerard B, Duvall JR, Lowe JT, Murillo T, Wei J, Akella LB, Marcaurelle LA.

ACS Comb Sci. 2011 Jul 11;13(4):365-74. doi: 10.1021/co2000218. Epub 2011 Apr 28.

PMID:
21526820
[PubMed - indexed for MEDLINE]
Free PMC Article
3.

Diversity-oriented synthesis of 13- to 18-membered macrolactams via ring-closing metathesis.

Dandapani S, Lowe JT, Comer E, Marcaurelle LA.

J Org Chem. 2011 Oct 7;76(19):8042-8. doi: 10.1021/jo2011957. Epub 2011 Aug 29.

PMID:
21875084
[PubMed - indexed for MEDLINE]
4.

An aldol-based build/couple/pair strategy for the synthesis of medium- and large-sized rings: discovery of macrocyclic histone deacetylase inhibitors.

Marcaurelle LA, Comer E, Dandapani S, Duvall JR, Gerard B, Kesavan S, Lee MD 4th, Liu H, Lowe JT, Marie JC, Mulrooney CA, Pandya BA, Rowley A, Ryba TD, Suh BC, Wei J, Young DW, Akella LB, Ross NT, Zhang YL, Fass DM, Reis SA, Zhao WN, Haggarty SJ, Palmer M, Foley MA.

J Am Chem Soc. 2010 Dec 1;132(47):16962-76. doi: 10.1021/ja105119r. Epub 2010 Nov 10.

PMID:
21067169
[PubMed - indexed for MEDLINE]
Free PMC Article
5.

Giant macrolactams based on β-sheet peptides.

Cheng PN, Nowick JS.

J Org Chem. 2011 May 6;76(9):3166-73. doi: 10.1021/jo102598n. Epub 2011 Apr 15.

PMID:
21452877
[PubMed - indexed for MEDLINE]
Free PMC Article
6.

Recent applications of ring-closing metathesis in the synthesis of lactams and macrolactams.

Hassan HM.

Chem Commun (Camb). 2010 Dec 28;46(48):9100-6. doi: 10.1039/c0cc03122d. Epub 2010 Nov 12. Review.

PMID:
21076746
[PubMed - indexed for MEDLINE]
7.

Multicomponent macrocyclization reactions (MCMRs) employing highly reactive acyl ketene and nitrile oxide intermediates.

Knapp JM, Fettinger JC, Kurth MJ.

Org Lett. 2011 Sep 2;13(17):4732-5. doi: 10.1021/ol202024a. Epub 2011 Aug 9.

PMID:
21827181
[PubMed - indexed for MEDLINE]
Free PMC Article
8.

Design and synthesis of 1,2,3-triazole-fused chiral medium-ring benzo-heterocycles, scaffolds mimicking benzolactams.

Das Adhikary N, Chattopadhyay P.

J Org Chem. 2012 Jun 15;77(12):5399-405. doi: 10.1021/jo3004327. Epub 2012 Jun 6.

PMID:
22647142
[PubMed - indexed for MEDLINE]
9.

Synthesis of a novel suppressor of beta-cell apoptosis via diversity-oriented synthesis.

Chou DH, Duvall JR, Gerard B, Liu H, Pandya BA, Suh BC, Forbeck EM, Faloon P, Wagner BK, Marcaurelle LA.

ACS Med Chem Lett. 2011 Sep 8;2(9):698-702.

PMID:
21927648
[PubMed]
Free PMC Article
10.

Solid-phase synthesis of peptide thioureas and thiazole-containing macrocycles through Ru-catalyzed ring-closing metathesis.

Cohrt AE, Nielsen TE.

ACS Comb Sci. 2014 Feb 10;16(2):71-7. doi: 10.1021/co400102v. Epub 2014 Jan 17.

PMID:
24377264
[PubMed - indexed for MEDLINE]
11.

Systematic study of the synthesis of macrocyclic dipeptide beta-turn mimics possessing 8-, 9-, and 10- membered rings by ring-closing metathesis.

Kaul R, Surprenant S, Lubell WD.

J Org Chem. 2005 May 13;70(10):3838-44. Erratum in: J Org Chem. 2005 Jun 10;70(12):4901-2.

PMID:
15876068
[PubMed - indexed for MEDLINE]
12.

Efficient synthesis and astonishing supramolecular architectures of several symmetric macrolactams.

Baillargeon P, Bernard S, Gauthier D, Skouta R, Dory YL.

Chemistry. 2007;13(33):9223-35.

PMID:
17886846
[PubMed - indexed for MEDLINE]
13.

Application of a sparse matrix design strategy to the synthesis of dos libraries.

Akella LB, Marcaurelle LA.

ACS Comb Sci. 2011 Jul 11;13(4):357-64. doi: 10.1021/co200020j. Epub 2011 Apr 28.

PMID:
21526822
[PubMed - indexed for MEDLINE]
Free PMC Article
14.

Using cross-metathesis to couple L-phenylalanine to a macrocyclic lactam.

Enholm E, Low T.

J Org Chem. 2006 Mar 17;71(6):2272-6.

PMID:
16526773
[PubMed - indexed for MEDLINE]
15.

A diversity-oriented synthesis approach to macrocycles via oxidative ring expansion.

Kopp F, Stratton CF, Akella LB, Tan DS.

Nat Chem Biol. 2012 Mar 11;8(4):358-65. doi: 10.1038/nchembio.911.

PMID:
22406518
[PubMed - indexed for MEDLINE]
Free PMC Article
16.

Radical photocyclization route for macrocyclic lactone ring expansion and conversion to macrocyclic lactams and ketones.

Nishikawa K, Yoshimi Y, Maeda K, Morita T, Takahashi I, Itou T, Inagaki S, Hatanaka M.

J Org Chem. 2013 Jan 18;78(2):582-9. doi: 10.1021/jo3024126. Epub 2013 Jan 8.

PMID:
23253018
[PubMed - indexed for MEDLINE]
17.

Sequence of intramolecular carbonylation and asymmetric hydrogenation reactions: highly regio- and enantioselective synthesis of medium ring tricyclic lactams.

Lu SM, Alper H.

J Am Chem Soc. 2008 May 21;130(20):6451-5. doi: 10.1021/ja7111417. Epub 2008 Apr 30.

PMID:
18444651
[PubMed - indexed for MEDLINE]
18.
19.

A versatile approach toward the ansamycin antibiotics.

Peng W, Blagg BS.

Org Lett. 2006 Mar 2;8(5):975-8.

PMID:
16494488
[PubMed - indexed for MEDLINE]
20.

A ring-closing metathesis-based approach to the synthesis of (+)-tetrabenazine.

Johannes M, Altmann KH.

Org Lett. 2012 Jul 20;14(14):3752-5. doi: 10.1021/ol301612q. Epub 2012 Jun 28.

PMID:
22742980
[PubMed - indexed for MEDLINE]
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