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Results: 1 to 20 of 480

1.

Comparison of miniaturized time-resolved fluorescence resonance energy transfer and enzyme-coupled luciferase high-throughput screening assays to discover inhibitors of Rho-kinase II (ROCK-II).

Schröter T, Minond D, Weiser A, Dao C, Habel J, Spicer T, Chase P, Baillargeon P, Scampavia L, Schürer S, Chung C, Mader C, Southern M, Tsinoremas N, LoGrasso P, Hodder P.

J Biomol Screen. 2008 Jan;13(1):17-28. doi: 10.1177/1087057107310806.

PMID:
18227223
[PubMed - indexed for MEDLINE]
2.

Discovery of novel scaffolds for Rho kinase 2 inhibitor through TRFRET-based high throughput screening assay.

Oh KS, Mun J, Cho JE, Lee S, Yi KY, Lim CJ, Lee JS, Park WJ, Lee BH.

Comb Chem High Throughput Screen. 2013 Jan;16(1):37-46.

PMID:
22934984
[PubMed - indexed for MEDLINE]
3.

Fluorescence polarization and time-resolved fluorescence resonance energy transfer techniques for PI3K assays.

Horiuchi KY, Ma H.

Methods Mol Biol. 2009;572:161-76. doi: 10.1007/978-1-60761-244-5_10.

PMID:
20694691
[PubMed - indexed for MEDLINE]
4.

Readout technologies for highly miniaturized kinase assays applicable to high-throughput screening in a 1536-well format.

Klumpp M, Boettcher A, Becker D, Meder G, Blank J, Leder L, Forstner M, Ottl J, Mayr LM.

J Biomol Screen. 2006 Sep;11(6):617-33. Epub 2006 Jun 7.

PMID:
16760365
[PubMed - indexed for MEDLINE]
5.
6.

Development and applications of a broad-coverage, TR-FRET-based kinase binding assay platform.

Lebakken CS, Riddle SM, Singh U, Frazee WJ, Eliason HC, Gao Y, Reichling LJ, Marks BD, Vogel KW.

J Biomol Screen. 2009 Sep;14(8):924-35. doi: 10.1177/1087057109339207. Epub 2009 Jun 29.

PMID:
19564447
[PubMed - indexed for MEDLINE]
7.

Development and implementation of a miniaturized high-throughput time-resolved fluorescence energy transfer assay to identify small molecule inhibitors of polo-like kinase 1.

Sharlow ER, Leimgruber S, Shun TY, Lazo JS.

Assay Drug Dev Technol. 2007 Dec;5(6):723-35. doi: 10.1089/adt.2007.102.

PMID:
18181689
[PubMed - indexed for MEDLINE]
8.

Miniaturization of intracellular calcium functional assays to 1536-well plate format using a fluorometric imaging plate reader.

Hodder P, Mull R, Cassaday J, Berry K, Strulovici B.

J Biomol Screen. 2004 Aug;9(5):417-26.

PMID:
15296641
[PubMed - indexed for MEDLINE]
9.

A high-throughput, nonisotopic, competitive binding assay for kinases using nonselective inhibitor probes (ED-NSIP).

Vainshtein I, Silveria S, Kaul P, Rouhani R, Eglen RM, Wang J.

J Biomol Screen. 2002 Dec;7(6):507-14.

PMID:
14599348
[PubMed - indexed for MEDLINE]
10.

Development of high-throughput TR-FRET and AlphaScreen assays for identification of potent inhibitors of PDK1.

Xu Z, Nagashima K, Sun D, Rush T, Northrup A, Andersen JN, Kariv I, Bobkova EV.

J Biomol Screen. 2009 Dec;14(10):1257-62. doi: 10.1177/1087057109349356. Epub .

PMID:
19822882
[PubMed - indexed for MEDLINE]
11.

Identification of novel scaffolds for IκB kinase beta inhibitor via a high-throughput screening TR-FRET assay.

Oh KS, Lee S, Choi JK, Lee BH.

Comb Chem High Throughput Screen. 2010 Nov;13(9):790-7.

PMID:
20615197
[PubMed - indexed for MEDLINE]
12.

Establishment and application of a high throughput model for Rho kinase inhibitors screening based on fluorescence polarization.

Duan W, Sun L, Liu J, Wu X, Zhang L, Yan M.

Biol Pharm Bull. 2006 Jun;29(6):1138-42.

PMID:
16755006
[PubMed - indexed for MEDLINE]
Free Article
13.

Recommendations for the reduction of compound artifacts in time-resolved fluorescence resonance energy transfer assays.

Imbert PE, Unterreiner V, Siebert D, Gubler H, Parker C, Gabriel D.

Assay Drug Dev Technol. 2007 Jun;5(3):363-72.

PMID:
17638536
[PubMed - indexed for MEDLINE]
14.

A time-resolved fluorescence resonance energy transfer assay for high-throughput screening of 14-3-3 protein-protein interaction inhibitors.

Du Y, Fu RW, Lou B, Zhao J, Qui M, Khuri FR, Fu H.

Assay Drug Dev Technol. 2013 Jul;11(6):367-81. doi: 10.1089/adt.2013.507. Epub 2013 Aug 1.

PMID:
23906346
[PubMed - indexed for MEDLINE]
Free PMC Article
15.

A toolbox approach to high-throughput TR-FRET-based SUMOylation and DeSUMOylation assays.

Carlson CB, Horton RA, Vogel KW.

Assay Drug Dev Technol. 2009 Aug;7(4):348-55. doi: 10.1089/adt.2008.0188.

PMID:
19656081
[PubMed - indexed for MEDLINE]
16.

Cellular HTS assays for pharmacological characterization of Na(V)1.7 modulators.

Trivedi S, Dekermendjian K, Julien R, Huang J, Lund PE, Krupp J, Kronqvist R, Larsson O, Bostwick R.

Assay Drug Dev Technol. 2008 Apr;6(2):167-79.

PMID:
18078380
[PubMed - indexed for MEDLINE]
17.

Data concordance from a comparison between filter binding and fluorescence polarization assay formats for identification of ROCK-II inhibitors.

Hubert CL, Sherling SE, Johnston PA, Stancato LF.

J Biomol Screen. 2003 Aug;8(4):399-409.

PMID:
14567792
[PubMed - indexed for MEDLINE]
18.

Development, validation and implementation of immobilized metal affinity for phosphochemicals (IMAP)-based high-throughput screening assays for low-molecular-weight compound libraries.

Sharlow ER, Leimgruber S, Yellow-Duke A, Barrett R, Wang QJ, Lazo JS.

Nat Protoc. 2008;3(8):1350-63. doi: 10.1038/nprot.2008.111.

PMID:
18714303
[PubMed - indexed for MEDLINE]
19.

Identification of inhibitors of bacterial transcription/translation machinery utilizing a miniaturized 1536-well format screen.

Kariv I, Cao H, Marvil PD, Bobkova EV, Bukhtiyarov YE, Yan YP, Patel U, Coudurier L, Chung TD, Oldenburg KR.

J Biomol Screen. 2001 Aug;6(4):233-43.

PMID:
11689123
[PubMed - indexed for MEDLINE]
20.

A dual-readout F2 assay that combines fluorescence resonance energy transfer and fluorescence polarization for monitoring bimolecular interactions.

Du Y, Nikolovska-Coleska Z, Qui M, Li L, Lewis I, Dingledine R, Stuckey JA, Krajewski K, Roller PP, Wang S, Fu H.

Assay Drug Dev Technol. 2011 Aug;9(4):382-93. doi: 10.1089/adt.2010.0292. Epub 2011 Mar 11.

PMID:
21395401
[PubMed - indexed for MEDLINE]
Free PMC Article

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