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Results: 1 to 20 of 101

1.

Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. 5. Opioid receptor binding properties of N-((4'-phenyl)-phenethyl) analogues of 8-CAC.

VanAlstine MA, Wentland MP, Cohen DJ, Bidlack JM.

Bioorg Med Chem Lett. 2007 Dec 1;17(23):6516-20. Epub 2007 Sep 29.

PMID:
17935988
[PubMed - indexed for MEDLINE]
Free PMC Article
2.

Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. 4. Opioid receptor binding properties of 8-[N-(4'-phenyl)-phenethyl)carboxamido] analogues of cyclazocine and ethylketocycalzocine.

Wentland MP, VanAlstine M, Kucejko R, Lou R, Cohen DJ, Parkhill AL, Bidlack JM.

J Med Chem. 2006 Sep 7;49(18):5635-9.

PMID:
16942039
[PubMed - indexed for MEDLINE]
3.

Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. Part 6: Opioid receptor binding properties of cyclic variants of 8-carboxamidocyclazocine.

Wentland MP, Sun X, Cohen DJ, Bidlack JM.

Bioorg Med Chem. 2008 May 15;16(10):5653-64. doi: 10.1016/j.bmc.2008.03.066. Epub 2008 Mar 30.

PMID:
18417347
[PubMed - indexed for MEDLINE]
Free PMC Article
4.

Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. Part 7: syntheses and opioid receptor properties of cyclic variants of cyclazocine.

Wentland MP, Lu Q, Ganorkar R, Zhang SZ, Jo S, Cohen DJ, Bidlack JM.

Bioorg Med Chem Lett. 2009 Jan 15;19(2):365-8. doi: 10.1016/j.bmcl.2008.11.076. Epub 2008 Nov 24.

PMID:
19091564
[PubMed - indexed for MEDLINE]
5.

Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. Part 8. High affinity ligands for opioid receptors in the picomolar Ki range: oxygenated N-(2-[1,1'-biphenyl]-4-ylethyl) analogues of 8-CAC.

Wentland MP, Jo S, Gargano JM, VanAlstine MA, Cohen DJ, Bidlack JM.

Bioorg Med Chem Lett. 2012 Dec 15;22(24):7340-4. doi: 10.1016/j.bmcl.2012.10.081. Epub 2012 Oct 27.

PMID:
23142613
[PubMed - indexed for MEDLINE]
Free PMC Article
6.

8-Carboxamidocyclazocine analogues: redefining the structure-activity relationships of 2,6-methano-3-benzazocines.

Wentland MP, Lou R, Ye Y, Cohen DJ, Richardson GP, Bidlack JM.

Bioorg Med Chem Lett. 2001 Mar 12;11(5):623-6.

PMID:
11266156
[PubMed - indexed for MEDLINE]
7.

Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. Part 2: 8-formamidocyclazocine analogues.

Wentland MP, Sun X, Ye Y, Lou R, Bidlack JM.

Bioorg Med Chem Lett. 2003 Jun 2;13(11):1911-4.

PMID:
12749896
[PubMed - indexed for MEDLINE]
8.

Probes for narcotic receptor mediated phenomena. 44. Synthesis of an N-substituted 4-hydroxy-5-(3-hydroxyphenyl)morphan with high affinity and selective μ-antagonist activity.

Iyer MR, Lee YS, Deschamps JR, Dersch CM, Rothman RB, Jacobson AE, Rice KC.

Eur J Med Chem. 2012 Apr;50:44-54. doi: 10.1016/j.ejmech.2012.01.025. Epub 2012 Jan 20.

PMID:
22341895
[PubMed - indexed for MEDLINE]
Free PMC Article
9.

Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. Part 9: Synthesis, characterization and molecular modeling of pyridinyl isosteres of N-BPE-8-CAC (1), a high affinity ligand for opioid receptors.

VanAlstine MA, Wentland MP, Alvarez J, Cao Q, Cohen DJ, Knapp BI, Bidlack JM.

Bioorg Med Chem Lett. 2013 Apr 1;23(7):2128-33. doi: 10.1016/j.bmcl.2013.01.117. Epub 2013 Feb 8.

PMID:
23434225
[PubMed - indexed for MEDLINE]
Free PMC Article
10.

Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. Part 3: 8-Thiocarboxamido and 8-thioformamido derivatives of cyclazocine.

Wentland MP, Sun X, Bu Y, Lou R, Cohen DJ, Bidlack JM.

Bioorg Med Chem Lett. 2005 May 16;15(10):2547-51.

PMID:
15863314
[PubMed - indexed for MEDLINE]
11.

Novel diastereomeric opioid tetrapeptides exhibit differing pharmacological activity profiles.

Ioja E, Tourwé D, Kertész I, Tóth G, Borsodi A, Benyhe S.

Brain Res Bull. 2007 Sep 14;74(1-3):119-29. Epub 2007 Jun 8.

PMID:
17683797
[PubMed - indexed for MEDLINE]
12.

Syntheses and opioid receptor binding affinities of 8-amino-2,6-methano-3-benzazocines.

Wentland MP, Ye Y, Cioffi CL, Lou R, Zhou Q, Xu G, Duan W, Dehnhardt CM, Sun X, Cohen DJ, Bidlack JM.

J Med Chem. 2003 Feb 27;46(5):838-49.

PMID:
12593663
[PubMed - indexed for MEDLINE]
13.

8-Carboxamidocyclazocine: a long-acting, novel benzomorphan.

Bidlack JM, Cohen DJ, McLaughlin JP, Lou R, Ye Y, Wentland MP.

J Pharmacol Exp Ther. 2002 Jul;302(1):374-80.

PMID:
12065740
[PubMed - indexed for MEDLINE]
Free Article
14.

Effects of the substitution of Phe4 in the opioid peptide [D-Ala8]dynorphin A-(1-11)NH2.

Vig BS, Zheng MQ, Murray TF, Aldrich JV.

J Med Chem. 2003 Sep 11;46(19):4002-8.

PMID:
12954053
[PubMed - indexed for MEDLINE]
15.

8-Aminocyclazocine analogues: synthesis and structure-activity relationships.

Wentland MP, Xu G, Cioffi CL, Ye Y, Duan W, Cohen DJ, Colasurdo AM, Bidlack JM.

Bioorg Med Chem Lett. 2000 Jan 17;10(2):183-7.

PMID:
10673107
[PubMed - indexed for MEDLINE]
16.
17.

High-affinity carbamate analogues of morphinan at opioid receptors.

Peng X, Knapp BI, Bidlack JM, Neumeyer JL.

Bioorg Med Chem Lett. 2007 Mar 15;17(6):1508-11. Epub 2007 Jan 17.

PMID:
17276685
[PubMed - indexed for MEDLINE]
Free PMC Article
18.

Synthesis and opioid activity of enantiomeric N-substituted 2,3,4,4a,5,6,7,7a-octahydro-1H-benzofuro[3,2-e]isoquinolines.

Hsin LW, Chang LT, Rothman RB, Dersch CM, Fishback JA, Matsumoto RR.

J Med Chem. 2010 Feb 11;53(3):1392-6. doi: 10.1021/jm901503e.

PMID:
20055417
[PubMed - indexed for MEDLINE]
19.

Antipodal alpha-N-(methyl through decyl)-N-normetazocines (5,9 alpha-dimethyl-2'-hydroxy-6,7-benzomorphans): in vitro and in vivo properties.

May EL, Aceto MD, Bowman ER, Bentley C, Martin BR, Harris LS, Medzihradsky F, Mattson MV, Jacobson AE.

J Med Chem. 1994 Sep 30;37(20):3408-18.

PMID:
7932569
[PubMed - indexed for MEDLINE]
20.

Opioid ligand binding sites in the spinal cord of the guinea-pig.

Zarr GD, Werling LL, Brown SR, Cox BM.

Neuropharmacology. 1986 May;25(5):471-80.

PMID:
3016586
[PubMed - indexed for MEDLINE]

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