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Results: 11

PubMed Links for Books (Select 2510508)

1.

Identification and optimization of inhibitors of Trypanosomal cysteine proteases: cruzain, rhodesain, and TbCatB.

Mott BT, Ferreira RS, Simeonov A, Jadhav A, Ang KK, Leister W, Shen M, Silveira JT, Doyle PS, Arkin MR, McKerrow JH, Inglese J, Austin CP, Thomas CJ, Shoichet BK, Maloney DJ.

J Med Chem. 2010 Jan 14;53(1):52-60. doi: 10.1021/jm901069a.

2.

Development of potent purine-derived nitrile inhibitors of the trypanosomal protease TbcatB.

Mallari JP, Shelat AA, Obrien T, Caffrey CR, Kosinski A, Connelly M, Harbut M, Greenbaum D, McKerrow JH, Guy RK.

J Med Chem. 2008 Feb 14;51(3):545-52. doi: 10.1021/jm070760l. Epub 2008 Jan 4.

PMID:
18173229
4.

A common allosteric site and mechanism in caspases.

Scheer JM, Romanowski MJ, Wells JA.

Proc Natl Acad Sci U S A. 2006 May 16;103(20):7595-600. Epub 2006 May 8.

5.

Caspase inhibitors: a pharmaceutical industry perspective.

Linton SD.

Curr Top Med Chem. 2005;5(16):1697-717. Review.

PMID:
16375749
6.

Crystal structures of a ligand-free and malonate-bound human caspase-1: implications for the mechanism of substrate binding.

Romanowski MJ, Scheer JM, O'Brien T, McDowell RS.

Structure. 2004 Aug;12(8):1361-71.

PMID:
15296730
7.

Inflammatory caspases: linking an intracellular innate immune system to autoinflammatory diseases.

Martinon F, Tschopp J.

Cell. 2004 May 28;117(5):561-74. Review.

PMID:
15163405
8.

Novel, nonpeptidic cyanamides as potent and reversible inhibitors of human cathepsins K and L.

Falgueyret JP, Oballa RM, Okamoto O, Wesolowski G, Aubin Y, Rydzewski RM, Prasit P, Riendeau D, Rodan SB, Percival MD.

J Med Chem. 2001 Jan 4;44(1):94-104.

PMID:
11141092
9.

Peptide based interleukin-1 beta converting enzyme (ICE) inhibitors: synthesis, structure activity relationships and crystallographic study of the ICE-inhibitor complex.

Okamoto Y, Anan H, Nakai E, Morihira K, Yonetoku Y, Kurihara H, Sakashita H, Terai Y, Takeuchi M, Shibanuma T, Isomura Y.

Chem Pharm Bull (Tokyo). 1999 Jan;47(1):11-21.

PMID:
9987822
10.

Structure and mechanism of interleukin-1 beta converting enzyme.

Wilson KP, Black JA, Thomson JA, Kim EE, Griffith JP, Navia MA, Murcko MA, Chambers SP, Aldape RA, Raybuck SA, et al.

Nature. 1994 Jul 28;370(6487):270-5.

PMID:
8035875
11.

Peptide aldehydes and nitriles as transition state analog inhibitors of cysteine proteases.

Dufour E, Storer AC, Ménard R.

Biochemistry. 1995 Jul 18;34(28):9136-43.

PMID:
7619812
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