Selective Inhibition of BET Protein Domains Has Functional Relevance

Cancer Discov. 2020 May;10(5):637. doi: 10.1158/2159-8290.CD-RW2020-048. Epub 2020 Mar 27.

Abstract

Inhibition of BET protein bromodomains BD1 and BD2 produces unique phenotypes in disease models.

Publication types

  • Comment

MeSH terms

  • Humans
  • Neoplasms*
  • Protein Domains
  • Transcription Factors*

Substances

  • Transcription Factors