Selective and enantiospecific acylation of kappa o...[J Med Chem. 1989] - PubMed Result

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1: J Med Chem. 1989 Feb;32(2):281-3.Links

Selective and enantiospecific acylation of kappa opioid receptors by (1S,2S)-trans-2-isothiocyanato-N-methyl-N-[2-(1-pyrrolidinyl) cyclohexy l] benzeneacetamide. Demonstration of kappa receptor heterogeneity.

de Costa BR, Rothman RB, Bykov V, Jacobson AE, Rice KC.

Section on Drug Design and Synthesis, National Institute of Digestive, Diabetes and Kidney Diseases, Bethesda, Maryland 20892.

PMID: 2536435 [PubMed - indexed for MEDLINE]

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Selective and enantiospecific acylation of kappa opioid receptors by (1S,2S)-trans-2-isoth...Selective and enantiospecific acylation of kappa opioid receptors by (1S,2S)-trans-2-isothiocyanato-N-methyl-N-[2-(1-pyrrolidinyl) cyclohexy l] benzeneacetamide. Demonstration of kappa receptor heterogeneity.

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