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    Org Biomol Chem. 2012 Mar 7;10(9):1870-6. Epub 2012 Jan 25.

    Enantioselective synthesis of the carbocyclic nucleoside (-)-abacavir.

    Source

    iThemba Pharmaceuticals PTY (Ltd.), Gauteng, South Africa.

    Abstract

    An enantiopure β-lactam with a suitably disposed electron withdrawing group on nitrogen, participated in a π-allylpalladium mediated reaction with 2,6-dichloropurine tetrabutylammonium salt to afford an advanced cis-1,4-substituted cyclopentenoid with both high regio- and stereoselectivity. This advanced intermediate was successfully manipulated to the total synthesis of (-)-Abacavir.

    PMID:
    22274412
    [PubMed - in process]

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