Interaction of barbiturates with dihydropicrotoxinin binding sites related to the GABA receptor-ionophore system

Life Sci. 1978 May 8;22(18):1643-51. doi: 10.1016/0024-3205(78)90061-9.
No abstract available

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Aminobutyrates / metabolism*
  • Animals
  • Barbiturates / metabolism*
  • Binding Sites
  • Brain / metabolism*
  • Ionophores / metabolism
  • Male
  • Membranes / metabolism
  • Picrotoxin / analogs & derivatives*
  • Rats
  • Receptors, Drug / metabolism*
  • Receptors, Neurotransmitter / physiology
  • Structure-Activity Relationship
  • gamma-Aminobutyric Acid / metabolism*

Substances

  • Aminobutyrates
  • Barbiturates
  • Ionophores
  • Receptors, Drug
  • Receptors, Neurotransmitter
  • Picrotoxin
  • dihydropicrotoxinin
  • gamma-Aminobutyric Acid