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    Fertil Steril. 2010 Oct;94(5):1632-8.e1. Epub 2010 Jan 4.

    Antiproliferative effects of anastrozole, methotrexate, and 5-fluorouracil on endometriosis in vitro and in vivo.

    Source

    Faculté de Médecine, Université Paris Descartes, EA 1833, ERTi, AP-HP Hôpital Cochin, Paris, France.

    Abstract

    OBJECTIVE:

    To investigate the effects of antiproliferative drugs (anastrozole, methotrexate, and 5-fluorouracil [5-FU]) on the proliferation of endometriotic cells in vitro and in vivo.

    DESIGN:

    Ex vivo study on human endometrial and endometriotic cells in culture; establishment of a murine model using mice implanted with human endometriosis.

    SETTING:

    University research center.

    PATIENT(S):

    Ten patients with ovarian endometrioma, 10 patients with deep infiltrating endometriosis, and 10 patients without endometriosis.

    INTERVENTION(S):

    Stromal and epithelial cells were extracted from endometrial and endometriotic biopsies from patients with endometriosis and from patients without endometriosis. Cells were treated in vitro with anastrozole, methotrexate, progesterone, or 5-FU. Human endometriotic lesions were implanted in nude mice. Mice were treated with 5-FU or phosphate-buffered saline during 4 weeks before sacrifice and extraction of the endometriotic implants.

    MAIN OUTCOME MEASURE(S):

    Stromal and epithelial cell proliferation and pathology score of endometriotic implants.

    RESULT(S):

    Although anastrozole, methotrexate, and progesterone were ineffective, 5-FU significantly decreased the proliferation of endometriotic cells in vitro and controlled the growth of both cells from ovarian endometrioma and deep infiltrating endometriosis.

    CONCLUSION(S):

    Considering common features between endometriotic cells and tumor cells, the use of 5-FU could be an option in the management of severe endometriosis.

    Copyright © 2010 American Society for Reproductive Medicine. Published by Elsevier Inc. All rights reserved.

    PMID:
    20045515
    [PubMed - indexed for MEDLINE]

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