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    Org Biomol Chem. 2008 Jul 21;6(14):2507-15. Epub 2008 May 9.

    Towards sequence selective DNA binding: design, synthesis and DNA binding studies of novel bis-porphyrin peptidic nanostructures.

    Source

    Département de chimie and CREFSIP, Faculté des sciences et de génie, Université Laval, Québec, Québec, Canada.

    Abstract

    A new series of peptidic nanostructures bearing two intercalating moieties was designed and synthesized to achieve selective recognition of DNA sequences. A cationic porphyrin was attached to a glutamic acid side chain and the latter introduced into a peptidic sequence by standard solid-phase peptide synthesis methodology. Conformation of the hydrosoluble peptidic structures bearing two cationic porphyrins was studied by circular dichroism. Using UV-visible spectroscopy and induced circular dichroism, we demonstrate that the compounds are fully intercalated upon binding to double-stranded DNA and that the compounds exhibit a tremendous preference for GC over AT sequences for intercalation.

    PMID:
    18600271
    [PubMed - indexed for MEDLINE]

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