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Results: 19

1.

Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranes [Confirmatory]

Source:
ChEMBL
Protein Target:
C-C motif chemokine 2; HC11; Monocyte chemoattractant protein 1; Monocyte chemotactic and activating factor; MCAF; Monocyte chemotactic protein 1; MCP-1; Monocyte secretory protein JE; Small-inducible cytokine A2
2.

Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membrane at 1 uM relative to control

Source:
ChEMBL
Protein Target:
C-C motif chemokine 2; HC11; Monocyte chemoattractant protein 1; Monocyte chemotactic and activating factor; MCAF; Monocyte chemotactic protein 1; MCP-1; Monocyte secretory protein JE; Small-inducible cytokine A2
3.

Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membrane assessed as kinetic rate index at Ki by dual-point competition association assay relative to control

Source:
ChEMBL
Protein Target:
C-C motif chemokine 2; HC11; Monocyte chemoattractant protein 1; Monocyte chemotactic and activating factor; MCAF; Monocyte chemotactic protein 1; MCP-1; Monocyte secretory protein JE; Small-inducible cytokine A2
4.

Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membrane assessed as residence time

Source:
ChEMBL
Protein Target:
C-C motif chemokine 2; HC11; Monocyte chemoattractant protein 1; Monocyte chemotactic and activating factor; MCAF; Monocyte chemotactic protein 1; MCP-1; Monocyte secretory protein JE; Small-inducible cytokine A2
5.

Displacement of [3H]INCB3344 from human CCR2 receptor expressed in human U2OS cell membranes by saturation binding assay [Confirmatory]

Source:
ChEMBL
Protein Target:
C-C motif chemokine 2; HC11; Monocyte chemoattractant protein 1; Monocyte chemotactic and activating factor; MCAF; Monocyte chemotactic protein 1; MCP-1; Monocyte secretory protein JE; Small-inducible cytokine A2
6.

Displacement of [3H]INCB3344 from human CCR2 receptor expressed in human U2OS cell membranes [Confirmatory]

Source:
ChEMBL
Protein Target:
C-C motif chemokine 2; HC11; Monocyte chemoattractant protein 1; Monocyte chemotactic and activating factor; MCAF; Monocyte chemotactic protein 1; MCP-1; Monocyte secretory protein JE; Small-inducible cytokine A2
7.

Displacement of [3H]INCB3344 from human CCR2 receptor expressed in human U2OS cell membranes assessed as association and dissociation of radioligand [Confirmatory]

Source:
ChEMBL
Protein Target:
C-C motif chemokine 2; HC11; Monocyte chemoattractant protein 1; Monocyte chemotactic and activating factor; MCAF; Monocyte chemotactic protein 1; MCP-1; Monocyte secretory protein JE; Small-inducible cytokine A2
8.

Displacement of [3H]INCB3344 from human CCR2 receptor expressed in human U2OS cell membranes assessed as association and dissociation of compound by competition association assay [Confirmatory]

Source:
ChEMBL
Protein Target:
C-C motif chemokine 2; HC11; Monocyte chemoattractant protein 1; Monocyte chemotactic and activating factor; MCAF; Monocyte chemotactic protein 1; MCP-1; Monocyte secretory protein JE; Small-inducible cytokine A2
9.

Inhibition of MCP1-mediated human THP cell migration [Confirmatory]

Source:
ChEMBL
Protein Target:
C-C motif chemokine 2; HC11; Monocyte chemoattractant protein 1; Monocyte chemotactic and activating factor; MCAF; Monocyte chemotactic protein 1; MCP-1; Monocyte secretory protein JE; Small-inducible cytokine A2
12.

Experimentally measured binding affinity data (Ki) for protein-ligand complexes derived from PDB

Source:
Shanghai Institute of Organic Chemistry
Protein Targets:
Chain 1, E. Coli (Lacz) Beta-Galactosidase (R599a) In Complex With D- Galctopyranosyl-1-One; ...
Total:
3355
13.
14.
15.

Summary of the probe development effort to identify inhibitors of sialic acid acetylesterase (SIAE) [Summary]

Source:
The Scripps Research Institute Molecular Screening Center
Protein Target:
Sialate O-acetylesterase; H-Lse; Sialic acid-specific 9-O-acetylesterase [Homo sapiens]
16.
17.
19.

70S ribosome inhibitor

Source:
ChEMBL
Protein Targets:
30S ribosomal protein S1; ...
Total:
57

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