Display Settings:

Format
Items per page
Sort by

Send to:

Choose Destination

Results: 1 to 20 of 17756

1.

Inhibition of human SIK [Confirmatory]

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
2.

Inhibition of human SIK assessed as residual activity at 1 uM relative to control

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
3.

Competitive binding affinity to SNF1LK (unknown origin) at 10 uM in presence of ATP relative to control

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
4.

Inhibition of SIK (unknown origin) [Confirmatory]

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
5.

Millipore: Percentage of residual kinase activity of SIK1 at 10uM relative to control. Control inhibitor: Staurosporine at 10.0uM. Buffer: 8 mM MOPS pH 7.0, 0.2 mM EDTA

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
6.

Millipore: Percentage of residual kinase activity of SIK1 at 1uM relative to control. Control inhibitor: Staurosporine at 10.0uM. Buffer: 8 mM MOPS pH 7.0, 0.2 mM EDTA

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
7.

Inhibition of human recombinant SIK expressed in Sf21 cells using CKRREILSRRPSYRK as substrate assessed as residual activity at 1 uM after 90 mins relative to staurosporine

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
8.

Inhibition of human recombinant SIK expressed in Sf21 cells using CREBtide as substrate assessed as residual activity at 1 uM after 90 mins by Cerep assay

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
9.

GSK_PKIS: SNF1LK (SIK) mean inhibition at 1 uM [Nanosyn]

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
10.

GSK_PKIS: SNF1LK (SIK) mean inhibition at 0.1 uM [Nanosyn]

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
11.

Binding constant for SIK kinase domain [Confirmatory]

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
12.

Inhibition of human SIK at 1 uM

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
13.

Inhibition of human SIK at 10 uM after 60 mins by TR-FRET assay

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
14.

Binding constant for SNF1LK kinase domain [Confirmatory]

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
15.

Activity of human SIK at 1 uM

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK1; Salt-inducible kinase 1; SIK-1; Serine/threonine-protein kinase SNF1-like kinase 1; Serine/threonine-protein kinase SNF1LK
16.

Kinase inhibition selectivity assay for compound SID-48409448

Source:
Burnham Center for Chemical Genomics
Protein Targets:
3-phosphoinositide-dependent protein kinase 1 isoform 1 [Homo sapiens]; ...
Total:
314
17.

Kinase Inhibitor Selectivity Profiling Assay

Source:
Ambit Biosciences
Protein Targets:
3-phosphoinositide-dependent protein kinase 1 isoform 1 [Homo sapiens]; ...
Total:
287
18.

Competitive binding affinity to SNF1LK2 (unknown origin) at 10 uM in presence of ATP relative to control

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK2; Qin-induced kinase; Salt-inducible kinase 2; SIK-2; Serine/threonine-protein kinase SNF1-like kinase 2
19.

Competitive binding affinity to QIK (unknown origin) at 10 uM in presence of ATP relative to control

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK2; Qin-induced kinase; Salt-inducible kinase 2; SIK-2; Serine/threonine-protein kinase SNF1-like kinase 2
20.

Inhibition of SNF1LK2 (unknown origin) at 10 uM relative to control

Source:
ChEMBL
Protein Target:
Serine/threonine-protein kinase SIK2; Qin-induced kinase; Salt-inducible kinase 2; SIK-2; Serine/threonine-protein kinase SNF1-like kinase 2

Display Settings:

Format
Items per page
Sort by

Send to:

Choose Destination

Supplemental Content

Refine your results

• What's this?

Actions on your results

Find related data

Recent activity

Your browsing activity is empty.

Activity recording is turned off.

Turn recording back on

See more...
Write to the Help Desk