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Mu-Opioid Receptor Binding Assay from US Patent US11845759: "Opioid compounds and uses thereof"
Assay data:7 Active, 7 Activity ≤ 1 µM, 8 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Agonistic activity of the kappa-opioid receptors from US Patent US11643436: "Polypeptide compound, pharmaceutical composition, preparation method and application thereof"
Assay data:10 Active, 10 Activity ≤ 1 nM, 10 Activity ≤ 1 µM, 10 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
KOR beta-Arrestin Agonist and Antagonist Assays from US Patent US11634396: "Opioid receptor modulators"
Assay data:12 Active, 2 Activity ≤ 1 µM, 69 Tested
MOR cAMP Agonist and Antagonist Assays from US Patent US11634396: "Opioid receptor modulators"
Assay data:73 Active, 49 Activity ≤ 1 µM, 312 Tested
Opioid Receptor Binding Assay from US Patent US11534436: "Methods for treating depressive symptoms"
Assay data:39 Active, 32 Activity ≤ 1 nM, 39 Activity ≤ 1 µM, 39 Tested
Opioid Receptor Binding Assay from US Patent US11492374: "Peptides for treatment of medical disorders"
Assay data:7 Active, 6 Activity ≤ 1 nM, 7 Activity ≤ 1 µM, 7 Tested
Displacement of [3H]DAMGO from human mu opioid receptor measured after 2 hrs by competitive binding assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Displacement of [3H]DAMGO from human cloned mu-opioid receptor by radioligand binding assay
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000586a OPRK1
Assay data:1 Tested
SummaryRelated BioAssays by Target
Selectivity interaction (Enzyme panel (ion channels, GPCRs, other targets)) EUB0000196bCl OPRK1
Selectivity interaction (GloSensor assay) EUB0000234b OPRM1
Selectivity interaction (Eurofins Panlabs Discovery Services Panel (enzymes and receptors)) EUB0000234b OPRM1
Selectivity interaction (Enzyme panel (GPCRS, ion channels, and transporters)) EUB0000194b OPRM1
Selectivity interaction (CEREP panel (GPCRS, ion channels, transporters)) EUB0000193b OPRK1
Selectivity interaction (SafetyScreen44? (Eurofins, ion channels, GPCRs, hydrolases, and other enzymes)) EUB0000282b OPRK1
Selectivity interaction (CEREP Wide Ligand screening panel (ion channels, receptors, enzymes)) EUB0000304b OPRM1
Selectivity interaction (CEREP Wide Ligand screening panel (ion channels, receptors, enzymes)) EUB0000304b OPRK1
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000344a OPRK1
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