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Results: 1 to 20 of 345

1.

Inhibition of recombinant human PCAF catalytic domain (492 to 658 aa) using histone H3 at 100 uM after 1 hr by radiochemical assay in presence of [acetyl-3H]-acetyl coenzyme A

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
2.

Inhibition of PCAF bromodomain (unknown origin) assessed as inhibition of PCAF BRD tat-AcK50 peptide interaction by ELISA

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
3.

Binding affinity to PCAF bromodomain (unknown origin) assessed as change in melting temperature at 10 uM by differential scanning fluorimetric analysis

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
4.

Inhibition of human recombinant N-terminal His-tagged PCAF histone acetyltransferase catalytic domain expressed in Escherichia coli BL21 D3 using biotinylated histone H3 as substrate at 50 uM after 10 mins by TR-FRET analysis relative to control

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
5.

Inhibition of human recombinant N-terminal His-tagged PCAF histone acetyltransferase catalytic domain expressed in Escherichia coli BL21 D3 using biotinylated histone H3 as substrate after 10 mins by TR-FRET analysis relative to control

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
6.

Inhibition of PCAF bromodomain (unknown origin)-HIV-Tak50ac interaction

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
7.

Inhibition of human recombinant histone acetyltransferase PCAF assessed as acetylation of histone H3 at 0.15 to 0.6 mM

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
8.

Binding affinity to PCAF bromodomain (unknown origin) assessed as change in melting temperature at 10 uM by differential scanning fluorimetric analysis

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
9.

Inhibition of PCAF (unknown origin) using histone H3 derived peptide as substrate after 20 mins by fluorescence assay

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
10.

Inhibition of PCAF (unknown origin) using histone H3 derived peptide as substrate at 10'-6 to 10'-3 M after 20 mins by fluorescence assay

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
11.

Competitive inhibition of PCAF (unknown origin) using histone H3 derived peptide as substrate after 20 mins by fluorescence assay

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
12.

Displacement of fluorescein-labeled MS239 from recombinant human PCAF after 1 hr by fluorescence anisotropy assay

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
13.

Inhibition of human recombinant His-tagged PCAF HAT domain expressed in Escherichia coli BL21(DE3) cells using [14C]Ac-AoA and histone H4 as substrate at >200 uM after 5 mins by scintillation counting

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
14.

Inhibition of human recombinant His-tagged PCAF HAT domain expressed in Escherichia coli BL21(DE3) cells using [14C]Ac-AoA and histone H4 as substrate after 5 mins by scintillation counting

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
15.

Inhibition of human recombinant His-tagged PCAF HAT domain expressed in Escherichia coli BL21(DE3) cells using [14C]Ac-AoA and histone H4 as substrate at 200 uM after 5 mins by scintillation counting

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
16.

Inhibition of human recombinant KAT2B using histone H4 peptide as substrate at 50 uM after 2 hrs

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
17.

Increase of human recombinant KAT2B acetylation activity using histone H4 peptide as substrate at 50 uM after 2 hrs

Source:
ChEMBL
Protein Target:
Histone acetyltransferase KAT2B; Histone acetyltransferase PCAF; Histone acetylase PCAF; Lysine acetyltransferase 2B; P300/CBP-associated factor; P/CAF
18.
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