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Selectivity interaction (hFSH antagonism assay) EUB0000340a FSHR
Assay data:1 Tested
SummaryRelated BioAssays by Target
Selectivity interaction (hFSH antagonism experiment) EUB0000240b FSHR
Cell-based assay (FSH Antagonism)
PRESTO-Tango GPCRome screening (FSHR)
Agonist activity at human FSHR expressed in CHO-K1 cells at 20 uM by PathHunter beta-arrestin assay relative to control
Assay data:8 Tested
SummaryPubMed CitationRelated BioAssays by Target
Antagonist activity at human FSHR expressed in CHO-K1 cells by PathHunter beta-arrestin assay
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Antagonist activity at human FSHR expressed in CHO-K1 cells at 20 uM by PathHunter beta-arrestin assay relative to control
Antagonist activity at human follicle stimulating hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed by agonist solution addition and measured after 120 mins by cell based TR-FRET assay
Assay data:5 Tested
Human FSH receptor (Glycoprotein hormone receptors)
Assay data:3 Active, 3 Tested
Positive allosteric modulation of human FSHR expressed in rat granulocytes assessed as FSH-induced estradiol production after 72 hrs by radioimmunossay
Assay data:3 Active, 4 Activity ≤ 1 µM, 4 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Positive allosteric modulation of FSHR (unknown origin) expressed in CHO cells assessed as FSH-induced cAMP accumulation incubated for 1 hr by HTRF assay
Assay data:6 Active, 6 Activity ≤ 1 µM, 6 Tested
Positive allosteric modulation of human FSH receptor expressed in CHO cells assessed as effect on FSH-induced cAMP accumulation at 50 uM after 1 hr by HTRF assay relative to FSH
Assay data:6 Tested
Positive allosteric modulation of human FSH receptor expressed in CHO cells assessed as effect on FSH-induced cAMP accumulation at 12 uM after 1 hr by HTRF assay relative to FSH
Positive allosteric modulation of human FSH receptor expressed in CHO cells assessed as effect on FSH-induced cAMP accumulation after 1 hr by HTRF assay
Assay data:23 Tested
Agonist activity at FSHR (unknown origin) at 10 uM after 90 to 180 mins by beta-arrestin assay relative to control
Antagonist activity at FSHR (unknown origin) at 10 uM after 3 to 5 hrs by beta-arrestin assay relative to control
Allosteric activation of human FSH receptor
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
Agonist activity at human FSH receptor by aromatase-based assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Agonist activity at human FSH receptor by cAMP-based assay
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