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Results: 1 to 20 of 7432

2.

Inverse agonist activity at GAL4-fused ERRalpha (unknown origin) transfected in african green monkey CV1 cells at 1 uM after 24 hrs by luciferase reporter gene assay relative to control

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
3.

Ratio of kaempferol IC50 to compound IC50 for human GAL4-DBD-fused ERRalpha-LBD transcriptional activity

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
4.

Inhibition of ERRalpha in human MCF7 cells assessed as downregulation of PDK4 mRNA expression at 2.5 to 10 uM after 48 hrs by RT-PCR analysis

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
5.

Inhibition of ERRalpha in human MCF7 cells assessed as downregulation of MCAD mRNA expression at 2.5 to 10 uM after 48 hrs by RT-PCR analysis

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
6.

Inhibition of ERRalpha in human MCF7 cells assessed as downregulation of PDK4 expression after 24 hrs by Western blot analysis

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
7.

Inhibition of ERRalpha in human MCF7 cells assessed as downregulation of MCAD expression after 24 hrs by Western blot analysis

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
8.
9.

Inverse agonist activity at human GAL4-DBD-fused ERRalpha-LBD transfected in human HepG2 cells assessed as disruption of interaction with PGC-1alpha after 24 hrs by dual luciferase reporter gene assay [Confirmatory]

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
10.

Displacement of [3H]E2 from human recombinant ERalpha receptor after overnight incubation by liquid scintillation counting analysis [Confirmatory]

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
11.

Displacement of [3H]E2 from human recombinant ERalpha receptor after overnight incubation by liquid scintillation counting analysis relative to 17beta-estradiol

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
12.

Antagonist activity at ERalpha receptor in human MCF7 cells assessed as inhibition of cell growth after 6 days by crystal violet staining method [Confirmatory]

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
13.

Agonist activity at ERalpha receptor in human MCF7 cells assessed as stimulation of cell proliferation after 6 days by crystal violet staining method

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
14.

Agonist activity at ERalpha receptor in human MCF7 cells assessed as activation of ERalpha-based transcription at 100 nM after 20 to 24 hrs by luciferase reporter gene assay

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
15.

Agonist activity at ERalpha receptor in human MCF7 cells assessed as activation of ERalpha-based transcription at 1 nM after 20 to 24 hrs by luciferase reporter gene assay

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
16.

Agonist activity at ERalpha receptor in human HeLa cells assessed as activation of ERalpha-based transcription at 100 nM after 20 to 24 hrs by luciferase reporter gene assay

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
17.

Agonist activity at ERalpha receptor in human HeLa cells assessed as activation of ERalpha-based transcription at 1 nM after 20 to 24 hrs by luciferase reporter gene assay

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
18.

Agonist activity at ERalpha receptor in human HepG2 cells assessed as activation of ERalpha-based transcription at 100 nM after 20 to 24 hrs by luciferase reporter gene assay

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
19.

Antagonist activity at ERalpha receptor in human HeLa cells assessed as inhibition of E2-induced response after 20 to 24 hrs by luciferase reporter gene assay

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1
20.

Partial agonist activity at ERalpha receptor in human HeLa cells assessed as activation of ERalpha-based transcription at 100 nM after 20 to 24 hrs by luciferase reporter gene assay

Source:
ChEMBL
Protein Target:
Steroid hormone receptor ERR1; Estrogen receptor-like 1; Estrogen-related receptor alpha; ERR-alpha; Nuclear receptor subfamily 3 group B member 1

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