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Serotonin Receptors in Neurobiology
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Serotonin Receptors in Neurobiology
Chattopadhyay
Amitabha
Center for Cellular and Molecular Biology, Hyderabad, India
CRC Press, Taylor & Francis Group
0-8493-3977-4
978-0-8493-3977-6
2007
© 2007
Taylor & Francis Group, LLC
Frontiers in Neuroscience
Table of Contents
Series Preface
Preface
Editor
Contributors
1 Quantitative Imaging of Serotonin Autofluorescence with Multiphoton Microscopy
S. K. Kaushalya and Sudipta Maiti
INTRODUCTION
MULTIPHOTON MICROSCOPY
OPTICAL SETUP
IMAGING SEROTONIN AND OTHER MONOAMINES IN LIVE NEURONS
REFERENCES
2 Monitoring Receptor-Mediated Changes of Intracellular cAMP Level by Using Ion Channels and Fluorescent Proteins as Biosensors
Evgeni G. Ponimaskin, Martin Heine, Andre Zeug, Tatyana Voyno-Yasenetskaya, and Petrus S. Salonikidis
INTRODUCTION
MONITORING OF RECEPTOR MEDIATED cAMP CHANGES IN LIVING CELLS BY ELECTROPHYSIOLOGICAL APPROACH
FÖRSTER RESONANCE ENERGY TRANSFER (FRET)-BASED cAMP SENSOR
REFERENCES
3 Membrane Organization and Dynamics of the Serotonin
1A
Receptor Monitored Using Fluorescence Microscopic Approaches
Shanti Kalipatnapu, Thomas J. Pucadyil, and Amitabha Chattopadhyay
RELEVANCE OF MEMBRANE ORGANIZATION AND DYNAMICS TO PROTEIN FUNCTION
THE SEROTONIN
1A
RECEPTOR
MEMBRANE ORGANIZATION OF THE SEROTONIN
1A
RECEPTOR MONITORED USING DETERGENT INSOLUBILITY
MEMBRANE DYNAMICS OF THE SEROTONIN
1A
RECEPTOR
CONCLUSION
REFERENCES
4 Calmodulin Is a 5-HT Receptor-Interacting and Regulatory Protein
Justin N. Turner, Sonya D. Coaxum, Andrew K. Gelasco, Maria N. Garnovskaya, and John R. Raymond
INTRODUCTION
5-HT RECEPTORS AND CALMODULIN
CONCLUSIONS
REFERENCES
5 Identification of Novel Transcriptional Regulators in the Nervous System
Federico Remes-Lenicov, Kirsten X. Jacobsen, Anastasia Rogaeva, Margaret Czesak, Mahmoud Hadjighasem, Mireille Daigle, and Paul R. Albert
INTRODUCTION
IDENTIFICATION OF TRANSCRIPTION START SITE
PROMOTER CHARACTERIZATION
IDENTIFICATION OF DNA ELEMENTS
IDENTIFICATION OF DNA BINDING PROTEINS
TRANSCRIPTION FACTOR ACTIVITY
SUMMARY: TRANSCRIPTIONAL APPROACH TO DISCOVERY
REFERENCES
6 Serotonin 2A (5-HT
2A
) Receptor Function: Ligand-Dependent Mechanisms and Pathways
Ishier Raote, Aditi Bhattacharya, and Mitradas M. Panicker
LOCALIZATION OF 5-HT
2A
MRNA AND RECEPTOR PROTEIN IN THE BRAIN
INTRACELLULAR SIGNALING CASCADES ACTIVATED BY THE 5-HT
2A
RECEPTOR
INTRACELLULAR LOCALIZATION OF THE 5-HT
2A
RECEPTOR
INTRACELLULAR TRAFFICKING OF THE 5-HT
2A
RECEPTOR
LONG-TERM REGULATION OF 5-HT
2A
RECEPTOR
CONCLUSION
REFERENCES
7 The 5-HT
1A
Receptor: A Signaling Hub Linked to Emotional Balance
Probal Banerjee, Mukti Mehta, and Baishali Kanjilal
INTRODUCTION
DISTRIBUTION AND ONTOGENY OF THE 5-HT
1A
-R
PRESYNAPTIC AND POSTSYNAPTIC 5-HT
1A
-R AND THEIR SIGNALING EFFECTS
ABERRANT 5-HT
1A
-R EXPRESSION AND DISEASES
THERAPEUTIC AGENTS THAT FUNCTION BY REGULATING 5-HT
1A
-R SIGNALING
RECENT ADVANCEMENT THROUGH THE USE OF THE SNRIs
ROLE OF 5-HT
1A
-R IN THE IMMUNE SYSTEM AND CANCER
REQUIRED FUTURE STUDIES TO UNRAVEL MECHANISMS OF 5-HT
1A
-R SIGNALING
EXAMPLES OF SOME STUDIES AND POSSIBLE STRATEGIES
CONCLUDING REMARKS
EXPERIMENTAL PROCEDURES
REFERENCES
8 Do Limits of Neuronal Plasticity Represent an Opportunity for Mental Diseases, Such as Addiction to Food and Illegal Drugs? Use and Utilities of Serotonin Receptor Knock-Out Mice
Valerie Compan
INTRODUCTION
HUMAN 5-HT RECEPTOR GENE POLYMORPHISMS AND ADDICTIONS TO FOOD AND ILLEGAL DRUGS
KNOCK-OUT OF 5-HT RECEPTORS CLASSICALLY REQUIRED ENVIRONMENTAL CHALLENGES TO PRODUCE MALADAPTIVE BEHAVIOR
5-HT RECEPTOR KNOCK-OUT MICE AND ADAPTIVE CHANGES IN CENTRAL SEROTONINERGIC SYSTEMS
CONCLUSION
REFERENCES
9 Use of Mice with Targeted Genetic Inactivation in the Serotonergic System for the Study of Anxiety
Miklos Toth
ROLE OF THE 5-HT SYSTEM IN MODULATING ANXIETY STATES
MICE WITH TARGETED GENETIC INACTIVATION IN THE SEROTONERGIC SYSTEM FOR THE STUDY OF ANXIETY
BEHAVIORAL TESTS FOR ANXIETY
MICE WITH GENETIC INACTIVATION OF 5-HT RECEPTORS AND THE 5-HT TRANSPORTER
SUMMARY
REFERENCES
Copyright © 2007
Taylor & Francis Group, LLC
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